Compile Data Set for Download or QSAR
Found 104 with Last Name = 'bernardo' and Initial = 'v'
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)copy SMILEScopy InChI
Affinity DataKi:  13nMAssay Description:Inhibition of human recombinant c-Abl by filter-binding assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50343424(1-(2-chloro-2-(4-chlorophenyl)ethyl)-N-(4-fluorobe...)copy SMILEScopy InChI
Affinity DataKi:  80nMAssay Description:Inhibition of human recombinant c-Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K79F5PubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50343427(CHEMBL1775039 | N-Benzyl-1-(2-chloro-2-phenylethyl...)copy SMILEScopy InChI
Affinity DataKi:  90nMAssay Description:Inhibition of human recombinant c-Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K79F5PubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50343430(CHEMBL1775036 | N-(3-Chlorophenyl)-1-(2-chloro-2-p...)copy SMILEScopy InChI
Affinity DataKi:  120nMAssay Description:Inhibition of human recombinant c-Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K79F5PubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50343431(1-(2-Chloro-2-phenylethyl)-6-[(2-morpholin-4-yleth...)copy SMILEScopy InChI
Affinity DataKi:  150nMAssay Description:Inhibition of human recombinant c-Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K79F5PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50343430(CHEMBL1775036 | N-(3-Chlorophenyl)-1-(2-chloro-2-p...)copy SMILEScopy InChI
Affinity DataKi:  190nMAssay Description:Inhibition of human recombinant c-Src by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K79F5PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50343431(1-(2-Chloro-2-phenylethyl)-6-[(2-morpholin-4-yleth...)copy SMILEScopy InChI
Affinity DataKi:  210nMAssay Description:Inhibition of human recombinant c-Src by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K79F5PubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50343421(2-({4-[(2-Phenylethyl)amino]-1-(2-phenylvinyl)-1H-...)copy SMILEScopy InChI
Affinity DataKi:  220nMAssay Description:Inhibition of human recombinant c-Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K79F5PubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50142885(Benzyl-[1-(2-chloro-2-phenyl-ethyl)-6-methylsulfan...)copy SMILEScopy InChI
Affinity DataKi:  260nMAssay Description:Inhibition of human recombinant c-Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K79F5PubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50343429(1-(2-Chloro-2-phenylethyl)-6-[(2-morpholin-4-yleth...)copy SMILEScopy InChI
Affinity DataKi:  270nMAssay Description:Inhibition of human recombinant c-Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K79F5PubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50343426(1-(2-Chloro-2-phenylethyl)-6-[(2-morpholin-4-yleth...)copy SMILEScopy InChI
Affinity DataKi:  340nMAssay Description:Inhibition of human recombinant c-Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K79F5PubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50343425(CHEMBL1775041 | N-(3-Chlorophenyl)-1-(2-chloro-2-p...)copy SMILEScopy InChI
Affinity DataKi:  390nMAssay Description:Inhibition of human recombinant c-Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K79F5PubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50343428(1-(2-Chloro-2-phenylethyl)-N-(4-fluorobenzyl)-6-[(...)copy SMILEScopy InChI
Affinity DataKi:  580nMAssay Description:Inhibition of human recombinant c-Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K79F5PubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50343417(1-[2-Chloro-2-(4-chlorophenyl)ethyl]-N-(pyridin-4-...)copy SMILEScopy InChI
Affinity DataKi:  660nMAssay Description:Inhibition of human recombinant c-Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K79F5PubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50343420(6-(Methylsulfonyl)-1-(2-phenylvinyl)-N-propyl-1H-p...)copy SMILEScopy InChI
Affinity DataKi:  720nMAssay Description:Inhibition of human recombinant c-Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K79F5PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50343419(CHEMBL1775043 | N-Benzyl-1-(2-chloro-2-phenylethyl...)copy SMILEScopy InChI
Affinity DataKi:  740nMAssay Description:Inhibition of human recombinant c-Src by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K79F5PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50343424(1-(2-chloro-2-(4-chlorophenyl)ethyl)-N-(4-fluorobe...)copy SMILEScopy InChI
Affinity DataKi:  800nMAssay Description:Inhibition of human recombinant c-Src by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K79F5PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50343428(1-(2-Chloro-2-phenylethyl)-N-(4-fluorobenzyl)-6-[(...)copy SMILEScopy InChI
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of human recombinant c-Src by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K79F5PubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50343418(1-[2-Chloro-2-(4-chlorophenyl)ethyl]-N-(pyridin-2-...)copy SMILEScopy InChI
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of human recombinant c-Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K79F5PubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50343422(1-[2-Chloro-2-(4-fluorophenyl)ethyl]-N-(pyridin-4-...)copy SMILEScopy InChI
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of human recombinant c-Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K79F5PubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50343419(CHEMBL1775043 | N-Benzyl-1-(2-chloro-2-phenylethyl...)copy SMILEScopy InChI
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of human recombinant c-Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K79F5PubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50343423(1-[2-Chloro-2-(4-fluorophenyl)ethyl]-N-(pyridin-2-...)copy SMILEScopy InChI
Affinity DataKi:  2.10E+3nMAssay Description:Inhibition of human recombinant c-Abl by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K79F5PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50343421(2-({4-[(2-Phenylethyl)amino]-1-(2-phenylvinyl)-1H-...)copy SMILEScopy InChI
Affinity DataKi:  2.40E+3nMAssay Description:Inhibition of human recombinant c-Src by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K79F5PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50343427(CHEMBL1775039 | N-Benzyl-1-(2-chloro-2-phenylethyl...)copy SMILEScopy InChI
Affinity DataKi:  2.90E+3nMAssay Description:Inhibition of human recombinant c-Src by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K79F5PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50343420(6-(Methylsulfonyl)-1-(2-phenylvinyl)-N-propyl-1H-p...)copy SMILEScopy InChI
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of human recombinant c-Src by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K79F5PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50343422(1-[2-Chloro-2-(4-fluorophenyl)ethyl]-N-(pyridin-4-...)copy SMILEScopy InChI
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of human recombinant c-Src by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K79F5PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50142885(Benzyl-[1-(2-chloro-2-phenyl-ethyl)-6-methylsulfan...)copy SMILEScopy InChI
Affinity DataKi:  3.70E+3nMAssay Description:Inhibition of human recombinant c-Src by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K79F5PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50343426(1-(2-Chloro-2-phenylethyl)-6-[(2-morpholin-4-yleth...)copy SMILEScopy InChI
Affinity DataKi:  3.80E+3nMAssay Description:Inhibition of human recombinant c-Src by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K79F5PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50343417(1-[2-Chloro-2-(4-chlorophenyl)ethyl]-N-(pyridin-4-...)copy SMILEScopy InChI
Affinity DataKi:  3.90E+3nMAssay Description:Inhibition of human recombinant c-Src by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K79F5PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50343418(1-[2-Chloro-2-(4-chlorophenyl)ethyl]-N-(pyridin-2-...)copy SMILEScopy InChI
Affinity DataKi:  4.80E+3nMAssay Description:Inhibition of human recombinant c-Src by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K79F5PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50343425(CHEMBL1775041 | N-(3-Chlorophenyl)-1-(2-chloro-2-p...)copy SMILEScopy InChI
Affinity DataKi:  7.60E+3nMAssay Description:Inhibition of human recombinant c-Src by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K79F5PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM50343423(1-[2-Chloro-2-(4-fluorophenyl)ethyl]-N-(pyridin-2-...)copy SMILEScopy InChI
Affinity DataKi:  8.30E+3nMAssay Description:Inhibition of human recombinant c-Src by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K79F5PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
University of Siena

Curated by ChEMBL
LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)copy SMILEScopy InChI
Affinity DataKi:  3.10E+4nMAssay Description:Inhibition of human recombinant c-Src by filter-binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28K79F5PubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50322393((S)-N-((3-amino-1-(5-ethyl-7H-pyrrolo[2,3-d]pyrimi...)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibition of AKT1 after 90 mins by IMAP assayMore data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50322395((S)-N-((3-amino-1-(5-methyl-7H-pyrrolo[2,3-d]pyrim...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Inhibition of AKT1 after 90 mins by IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X580CPubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50322394((S)-N-((3-amino-1-(5-chloro-7H-pyrrolo[2,3-d]pyrim...)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Inhibition of AKT1 after 90 mins by IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X580CPubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50322401((S)-N-((3-amino-1-(5-ethyl-7H-pyrrolo[2,3-d]pyrimi...)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:Inhibition of AKT1 after 90 mins by IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X580CPubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50322397((S)-N-((3-amino-1-(5-ethyl-7H-pyrrolo[2,3-d]pyrimi...)copy SMILEScopy InChI
Affinity DataIC50: 1.80nMAssay Description:Inhibition of AKT1 after 90 mins by IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X580CPubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM24855(4-{1,2-dihydrospiro[indole-3,4'-piperidine]}-7H-py...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of AKT1 after 90 mins by IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X580CPubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50322402((S)-N-((3-amino-1-(5-chloro-7H-pyrrolo[2,3-d]pyrim...)copy SMILEScopy InChI
Affinity DataIC50: 2.60nMAssay Description:Inhibition of AKT1 after 90 mins by IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X580CPubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50322403((S)-N-((3-amino-1-(5-methyl-7H-pyrrolo[2,3-d]pyrim...)copy SMILEScopy InChI
Affinity DataIC50: 3nMAssay Description:Inhibition of AKT1 after 90 mins by IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X580CPubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50322398((S)-N-((3-amino-1-(5-chloro-7H-pyrrolo[2,3-d]pyrim...)copy SMILEScopy InChI
Affinity DataIC50: 3.30nMAssay Description:Inhibition of AKT1 after 90 mins by IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X580CPubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50322388(5-chloro-4-(2,8-diazaspiro[4.5]decan-2-yl)-7H-pyrr...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of AKT1 after 90 mins by IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X580CPubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50322403((S)-N-((3-amino-1-(5-methyl-7H-pyrrolo[2,3-d]pyrim...)copy SMILEScopy InChI
Affinity DataIC50: 7.40nMAssay Description:Inhibition of AKT1 after 90 mins by IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X580CPubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50322396((S)-N-((3-amino-1-(5-cyano-7H-pyrrolo[2,3-d]pyrimi...)copy SMILEScopy InChI
Affinity DataIC50: 7.70nMAssay Description:Inhibition of AKT1 after 90 mins by IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X580CPubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50322404((S)-N-((3-amino-1-(5-cyano-7H-pyrrolo[2,3-d]pyrimi...)copy SMILEScopy InChI
Affinity DataIC50: 7.80nMAssay Description:Inhibition of AKT1 after 90 mins by IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X580CPubMed
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50322393((S)-N-((3-amino-1-(5-ethyl-7H-pyrrolo[2,3-d]pyrimi...)copy SMILEScopy InChI
Affinity DataIC50: 9nMAssay Description:Inhibition of AKT2 after 90 mins by IMAP assayMore data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50322399((S)-N-((3-amino-1-(5-methyl-7H-pyrrolo[2,3-d]pyrim...)copy SMILEScopy InChI
Affinity DataIC50: 11.4nMAssay Description:Inhibition of AKT1 after 90 mins by IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X580CPubMed
TargetRAC-gamma serine/threonine-protein kinase(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50322393((S)-N-((3-amino-1-(5-ethyl-7H-pyrrolo[2,3-d]pyrimi...)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of AKT3 after 90 mins by IMAP assayMore data for this Ligand-Target Pair
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50322412(CHEMBL1171840 | phenyl(3-amino-1-(5-methyl-7H-pyrr...)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibition of AKT1 after 90 mins by IMAP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24X580CPubMed
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