Compile Data Set for Download or QSAR
Found 12 with Last Name = 'constantinou-kokotou' and Initial = 'v'
TargetCytosolic phospholipase A2(Homo sapiens (Human))
University of Athens

Curated by ChEMBL
LigandPNGBDBM50023445(CHEMBL3329874)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of human recombinant GIVA cPLA2 in vitro vesicle assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7X7CPubMed
TargetCytosolic phospholipase A2(Homo sapiens (Human))
University of Athens

Curated by ChEMBL
LigandPNGBDBM50023444(CHEMBL3329869 | US9597318, Code GK185)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human recombinant GIVA cPLA2 in vitro vesicle assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HD7X7CPubMed
TargetPhospholipase A1 member A(Rattus norvegicus)
Agricultural University of Athens

Curated by ChEMBL
LigandPNGBDBM50470665(CHEMBL3143220)copy SMILEScopy InChI
Affinity DataIC50: 4.94E+4nMAssay Description:IC50 was measured as concentration causing 50% inhibition of lysosomal phospholipase A1 activityMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WW7MD4PubMed
TargetPhospholipase A1 member A(Rattus norvegicus)
Agricultural University of Athens

Curated by ChEMBL
LigandPNGBDBM50470662(CHEMBL357385)copy SMILEScopy InChI
Affinity DataIC50: 7.55E+4nMAssay Description:IC50 was measured as concentration causing 50% inhibition of lysosomal phospholipase A1 activity.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WW7MD4PubMed
TargetPhospholipase A1 member A(Rattus norvegicus)
Agricultural University of Athens

Curated by ChEMBL
LigandPNGBDBM50031282(CHEBI:17630 | Kanamycin)copy SMILEScopy InChI
Affinity DataIC50: 8.04E+4nMAssay Description:IC50 was measured as concentration causing 50% inhibition of lysosomal phospholipase A1 activity.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WW7MD4PubMed
TargetPhospholipase A1 member A(Rattus norvegicus)
Agricultural University of Athens

Curated by ChEMBL
LigandPNGBDBM50470660(CHEMBL142949)copy SMILEScopy InChI
Affinity DataIC50: 9.14E+4nMAssay Description:IC50 was measured as concentration causing 50% inhibition of lysosomal phospholipase A1 activity.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WW7MD4PubMed
TargetPhospholipase A1 member A(Rattus norvegicus)
Agricultural University of Athens

Curated by ChEMBL
LigandPNGBDBM50470660(CHEMBL142949)copy SMILEScopy InChI
Affinity DataIC50: 9.14E+4nMAssay Description:IC50 was measured as concentration causing 50% inhibition of lysosomal phospholipase A1 activity.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WW7MD4PubMed
TargetPhospholipase A1 member A(Rattus norvegicus)
Agricultural University of Athens

Curated by ChEMBL
LigandPNGBDBM50366389(GENTAMICIN)copy SMILEScopy InChI
Affinity DataIC50: 9.42E+4nMAssay Description:IC50 was measured as concentration causing 50% inhibition of lysosomal phospholipase A1 activity.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WW7MD4PubMed
TargetPhospholipase A1 member A(Rattus norvegicus)
Agricultural University of Athens

Curated by ChEMBL
LigandPNGBDBM50470663(CHEMBL3143222)copy SMILEScopy InChI
Affinity DataIC50: 1.01E+5nMAssay Description:IC50 was measured as concentration causing 50% inhibition of lysosomal phospholipase A1 activityMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WW7MD4PubMed
TargetPhospholipase A1 member A(Rattus norvegicus)
Agricultural University of Athens

Curated by ChEMBL
LigandPNGBDBM50470664(Netilmicin)copy SMILEScopy InChI
Affinity DataIC50: 1.15E+5nMAssay Description:IC50 was measured as concentration causing 50% inhibition of lysosomal phospholipase A1 activity.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WW7MD4PubMed
TargetPhospholipase A1 member A(Rattus norvegicus)
Agricultural University of Athens

Curated by ChEMBL
LigandPNGBDBM50470666(CHEMBL143885)copy SMILEScopy InChI
Affinity DataIC50: 1.18E+5nMAssay Description:IC50 was measured as concentration causing 50% inhibition of lysosomal phospholipase A1 activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WW7MD4PubMed
TargetPhospholipase A1 member A(Rattus norvegicus)
Agricultural University of Athens

Curated by ChEMBL
LigandPNGBDBM50470661(CHEMBL356044)copy SMILEScopy InChI
Affinity DataIC50: 1.32E+5nMAssay Description:IC50 was measured as concentration causing 50% inhibition of lysosomal phospholipase A1 activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2WW7MD4PubMed