Compile Data Set for Download or QSAR
Found 346 with Last Name = 'gopinatth' and Initial = 'v'
TargetP2Y purinoceptor 14(Homo sapiens (Human))TBA
LigandPNGBDBM50456168(CHEMBL1800685)copy SMILEScopy InChI
Affinity DataKi:  0.430nMAssay Description:Antagonist activity at human P2Y14 expressed in CHO cells assessed as inhibition of forskolin-induced increase of cAMP accumulation incubated for 15 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
TargetD(3) dopamine receptor(Homo sapiens)TBA
LigandPNGBDBM50584888(CHEMBL5085145)copy SMILES
Affinity DataKi:  330nMAssay Description:Inhibition of dopamine D3 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
TargetSigma intracellular receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50584882(CHEMBL5087121)copy SMILES
Affinity DataKi:  390nMAssay Description:Inhibition of sigma 2 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
TargetTranslocator protein(Homo sapiens (Human))TBA
LigandPNGBDBM50541998(CHEMBL4642592)copy SMILEScopy InChI
Affinity DataKi:  508nMAssay Description:Binding affinity to TSPO (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ69SPPubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50566377(CHEMBL4848380)copy SMILES
Affinity DataKi:  520nMAssay Description:Binding affinity to D1 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ69SPPubMed
TargetSigma intracellular receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50566410(CHEMBL4854018)copy SMILES
Affinity DataKi:  590nMAssay Description:Binding affinity to sigma 2 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ69SPPubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50405423(CHEMBL5283362)copy SMILEScopy InChI
Affinity DataKi:  600nMAssay Description:Histamine H2 receptor antagonistic activity on the isolated spontaneously beating guinea pig right atriumMore data for this Ligand-Target Pair
In DepthDetails
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50569565(CHEMBL4845850)copy SMILES
Affinity DataKi:  650nMAssay Description:Inhibition of alpha2a adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C2516QPubMed
TargetSigma intracellular receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50584891(CHEMBL5085823)copy SMILES
Affinity DataKi:  650nMAssay Description:Inhibition of sigma 2 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
TargetSigma intracellular receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50584891(CHEMBL5085823)copy SMILES
Affinity DataKi:  710nMAssay Description:Inhibition of sigma 2 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
TargetTranslocator protein(Homo sapiens (Human))TBA
LigandPNGBDBM50566402(CHEMBL4853466)copy SMILES
Affinity DataKi:  751nMAssay Description:Binding affinity to TSPO (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ69SPPubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50566377(CHEMBL4848380)copy SMILES
Affinity DataKi:  759nMAssay Description:Binding affinity to sigma 1 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ69SPPubMed
TargetD(3) dopamine receptor(Homo sapiens)TBA
LigandPNGBDBM50405421(CHEMBL5279730)copy SMILEScopy InChI
Affinity DataKi:  780nMAssay Description:Histamine H2 receptor antagonistic activity on the isolated spontaneously beating guinea pig right atriumMore data for this Ligand-Target Pair
In DepthDetails
TargetSigma intracellular receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50584887(CHEMBL5094034)copy SMILES
Affinity DataKi:  860nMAssay Description:Inhibition of sigma 2 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50541998(CHEMBL4642592)copy SMILEScopy InChI
Affinity DataKi:  860nMAssay Description:Binding affinity to beta3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ69SPPubMed
TargetSigma intracellular receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50566389(CHEMBL4854060)copy SMILES
Affinity DataKi:  931nMAssay Description:Binding affinity to sigma 2 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ69SPPubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50569557(CHEMBL4856060)copy SMILES
Affinity DataKi:  940nMAssay Description:Inhibition of alpha2a adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C2516QPubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50584888(CHEMBL5085145)copy SMILES
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of adrenergic alpha 2B receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))TBA
LigandPNGBDBM50584882(CHEMBL5087121)copy SMILES
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of SERT receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))TBA
LigandPNGBDBM50584882(CHEMBL5087121)copy SMILES
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of muscarinic M1 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50584883(CHEMBL5074765)copy SMILES
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of dopamine D5 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50584884(CHEMBL5075741)copy SMILES
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of dopamine D5 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50584885(CHEMBL5079653)copy SMILES
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of dopamine D5 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50584886(CHEMBL5090079)copy SMILES
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of dopamine D5 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
TargetSigma intracellular receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50584893(CHEMBL5083619)copy SMILES
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of sigma 2 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
TargetSigma intracellular receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50584896(CHEMBL5087295)copy SMILES
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of sigma 2 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
TargetSigma intracellular receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50584886(CHEMBL5090079)copy SMILES
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of sigma 2 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
TargetD(3) dopamine receptor(Homo sapiens)TBA
LigandPNGBDBM50584883(CHEMBL5074765)copy SMILES
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of dopamine D3 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50569559(CHEMBL4857492)copy SMILES
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of alpha2b adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C2516QPubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50584885(CHEMBL5079653)copy SMILES
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of adrenergic alpha 2B receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50584889(CHEMBL5083773)copy SMILES
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of adrenergic alpha 2B receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50584894(CHEMBL5076127)copy SMILES
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of adrenergic alpha 2B receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50584884(CHEMBL5075741)copy SMILES
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of adrenergic alpha 2B receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50584883(CHEMBL5074765)copy SMILES
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of adrenergic alpha 2B receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50584891(CHEMBL5085823)copy SMILES
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of adrenergic alpha 2B receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50584888(CHEMBL5085145)copy SMILES
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of adrenergic beta 3 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50584885(CHEMBL5079653)copy SMILES
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of adrenergic beta 3 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50584894(CHEMBL5076127)copy SMILES
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of adrenergic beta 3 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50584883(CHEMBL5074765)copy SMILES
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of adrenergic beta 3 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50584891(CHEMBL5085823)copy SMILES
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of adrenergic beta 3 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))TBA
LigandPNGBDBM50584892(CHEMBL5077671)copy SMILES
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of serotonin 5HT2C receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))TBA
LigandPNGBDBM50584892(CHEMBL5077671)copy SMILES
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of serotonin 5HT1D receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))TBA
LigandPNGBDBM50584882(CHEMBL5087121)copy SMILES
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of serotonin 5HT1D receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))TBA
LigandPNGBDBM50584888(CHEMBL5085145)copy SMILES
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of serotonin 5HT1D receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))TBA
LigandPNGBDBM50584885(CHEMBL5079653)copy SMILES
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of serotonin 5HT1D receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50584898(CHEMBL5094130)copy SMILES
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of KOR (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))TBA
LigandPNGBDBM50584883(CHEMBL5074765)copy SMILES
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of serotonin 5HT1D receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2611470PubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50569559(CHEMBL4857492)copy SMILES
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of dopamine D1 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C2516QPubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50569555(CHEMBL4848838)copy SMILES
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of dopamine D5 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C2516QPubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50405434(CHEMBL5274312)copy SMILEScopy InChI
Affinity DataKi:  1.10E+3nMAssay Description:Histamine H2 receptor antagonistic activity on the isolated spontaneously beating guinea pig right atriumMore data for this Ligand-Target Pair
In DepthDetails
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