Affinity DataKi: 0.430nMAssay Description:Antagonist activity at human P2Y14 expressed in CHO cells assessed as inhibition of forskolin-induced increase of cAMP accumulation incubated for 15 ...More data for this Ligand-Target Pair
Affinity DataKi: 330nMAssay Description:Inhibition of dopamine D3 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Affinity DataKi: 390nMAssay Description:Inhibition of sigma 2 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Affinity DataKi: 508nMAssay Description:Binding affinity to TSPO (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 520nMAssay Description:Binding affinity to D1 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 590nMAssay Description:Binding affinity to sigma 2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 600nMAssay Description:Histamine H2 receptor antagonistic activity on the isolated spontaneously beating guinea pig right atriumMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataKi: 650nMAssay Description:Inhibition of alpha2a adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 650nMAssay Description:Inhibition of sigma 2 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Affinity DataKi: 710nMAssay Description:Inhibition of sigma 2 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Affinity DataKi: 751nMAssay Description:Binding affinity to TSPO (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 759nMAssay Description:Binding affinity to sigma 1 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 780nMAssay Description:Histamine H2 receptor antagonistic activity on the isolated spontaneously beating guinea pig right atriumMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataKi: 860nMAssay Description:Inhibition of sigma 2 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Affinity DataKi: 860nMAssay Description:Binding affinity to beta3 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 931nMAssay Description:Binding affinity to sigma 2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 940nMAssay Description:Inhibition of alpha2a adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of adrenergic alpha 2B receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of SERT receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of muscarinic M1 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of dopamine D5 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of dopamine D5 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of dopamine D5 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of dopamine D5 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Inhibition of sigma 2 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Inhibition of sigma 2 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Inhibition of sigma 2 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Inhibition of dopamine D3 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Inhibition of alpha2b adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of adrenergic alpha 2B receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of adrenergic alpha 2B receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of adrenergic alpha 2B receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of adrenergic alpha 2B receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of adrenergic alpha 2B receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of adrenergic alpha 2B receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of adrenergic beta 3 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of adrenergic beta 3 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of adrenergic beta 3 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of adrenergic beta 3 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of adrenergic beta 3 receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of serotonin 5HT2C receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of serotonin 5HT1D receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of serotonin 5HT1D receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of serotonin 5HT1D receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of serotonin 5HT1D receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of KOR (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of serotonin 5HT1D receptor (unknown origin) assessed as binding constantMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:Inhibition of dopamine D1 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:Inhibition of dopamine D5 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:Histamine H2 receptor antagonistic activity on the isolated spontaneously beating guinea pig right atriumMore data for this Ligand-Target Pair
In DepthDetails
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