Compile Data Set for Download or QSAR
Found 821 with Last Name = 'ramdas' and Initial = 'v'
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457085(CHEMBL4203542)copy SMILEScopy InChI
Affinity DataKi:  0.0500nMAssay Description:Antagonist activity at rat A2A receptor assessed as reduction in CGS-21680-induced cAMP level pretreated for 15 mins followed by CGS-21680 addition m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457098(CHEMBL4217582)copy SMILEScopy InChI
Affinity DataKi:  0.0600nMAssay Description:Antagonist activity at rat A2A receptor assessed as reduction in CGS-21680-induced cAMP level pretreated for 15 mins followed by CGS-21680 addition m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457098(CHEMBL4217582)copy SMILEScopy InChI
Affinity DataKi:  0.0600nMAssay Description:Antagonist activity at human A2A receptor expressed in HEK293 cell membranes assessed as reduction in CGS-21680-induced cAMP level pretreated for 15 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457084(CHEMBL4217248)copy SMILEScopy InChI
Affinity DataKi:  0.0700nMAssay Description:Antagonist activity at human A2A receptor expressed in HEK293 cell membranes assessed as reduction in CGS-21680-induced cAMP level pretreated for 15 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457085(CHEMBL4203542)copy SMILEScopy InChI
Affinity DataKi:  0.150nMAssay Description:Antagonist activity at human A2A receptor expressed in HEK293 cell membranes assessed as reduction in CGS-21680-induced cAMP level pretreated for 15 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50231595(CHEMBL4092832)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Antagonist activity at human adenosine A1 receptor expressed in HEK293 cells assessed as reduction in CPA-mediated inhibition of forskolin-stimulated...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0QKCPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457093(CHEMBL4212821)copy SMILEScopy InChI
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HEK293 cell membranes after 90 mins radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457099(CHEMBL4213177)copy SMILEScopy InChI
Affinity DataKi:  0.210nMAssay Description:Antagonist activity at human A2A receptor expressed in HEK293 cell membranes assessed as reduction in CGS-21680-induced cAMP level pretreated for 15 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457093(CHEMBL4212821)copy SMILEScopy InChI
Affinity DataKi:  0.220nMAssay Description:Antagonist activity at human A2A receptor expressed in HEK293 cell membranes assessed as reduction in CGS-21680-induced cAMP level pretreated for 15 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457097(CHEMBL4205884)copy SMILEScopy InChI
Affinity DataKi:  0.25nMAssay Description:Antagonist activity at human A2A receptor expressed in HEK293 cell membranes assessed as reduction in CGS-21680-induced cAMP level pretreated for 15 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457092(CHEMBL4207914)copy SMILEScopy InChI
Affinity DataKi:  0.260nMAssay Description:Antagonist activity at human A2A receptor expressed in HEK293 cell membranes assessed as reduction in CGS-21680-induced cAMP level pretreated for 15 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457103(CHEMBL4217668)copy SMILEScopy InChI
Affinity DataKi:  0.270nMAssay Description:Antagonist activity at human A2A receptor expressed in HEK293 cell membranes assessed as reduction in CGS-21680-induced cAMP level pretreated for 15 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457087(CHEMBL4205341)copy SMILEScopy InChI
Affinity DataKi:  0.280nMAssay Description:Antagonist activity at rat A2A receptor assessed as reduction in CGS-21680-induced cAMP level pretreated for 15 mins followed by CGS-21680 addition m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50231590(CHEMBL4063997)copy SMILEScopy InChI
Affinity DataKi:  0.280nMAssay Description:Antagonist activity at human adenosine A1 receptor expressed in HEK293 cells assessed as reduction in CPA-mediated inhibition of forskolin-stimulated...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0QKCPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457097(CHEMBL4205884)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HEK293 cell membranes after 90 mins radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457092(CHEMBL4207914)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HEK293 cell membranes after 90 mins radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457105(CHEMBL4212278)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Antagonist activity at human A2A receptor expressed in HEK293 cell membranes assessed as reduction in CGS-21680-induced cAMP level pretreated for 15 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457086(CHEMBL4215754)copy SMILEScopy InChI
Affinity DataKi:  0.400nMAssay Description:Antagonist activity at human A2A receptor expressed in HEK293 cell membranes assessed as reduction in CGS-21680-induced cAMP level pretreated for 15 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457107(CHEMBL4209408)copy SMILEScopy InChI
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HEK293 cell membranes after 90 mins radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457098(CHEMBL4217582)copy SMILEScopy InChI
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HEK293 cell membranes after 90 mins radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457085(CHEMBL4203542)copy SMILEScopy InChI
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HEK293 cell membranes after 90 mins radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457091(CHEMBL4207104)copy SMILEScopy InChI
Affinity DataKi:  0.400nMAssay Description:Antagonist activity at human A2A receptor expressed in HEK293 cell membranes assessed as reduction in CGS-21680-induced cAMP level pretreated for 15 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457104(CHEMBL4217235)copy SMILEScopy InChI
Affinity DataKi:  0.400nMAssay Description:Antagonist activity at human A2A receptor expressed in HEK293 cell membranes assessed as reduction in CGS-21680-induced cAMP level pretreated for 15 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457087(CHEMBL4205341)copy SMILEScopy InChI
Affinity DataKi:  0.420nMAssay Description:Antagonist activity at human A2A receptor expressed in HEK293 cell membranes assessed as reduction in CGS-21680-induced cAMP level pretreated for 15 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457107(CHEMBL4209408)copy SMILEScopy InChI
Affinity DataKi:  0.420nMAssay Description:Antagonist activity at rat A2A receptor assessed as reduction in CGS-21680-induced cAMP level pretreated for 15 mins followed by CGS-21680 addition m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457086(CHEMBL4215754)copy SMILEScopy InChI
Affinity DataKi:  0.440nMAssay Description:Antagonist activity at rat A2A receptor assessed as reduction in CGS-21680-induced cAMP level pretreated for 15 mins followed by CGS-21680 addition m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457091(CHEMBL4207104)copy SMILEScopy InChI
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HEK293 cell membranes after 90 mins radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457101(CHEMBL4210241)copy SMILEScopy InChI
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HEK293 cell membranes after 90 mins radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457094(CHEMBL4204531)copy SMILEScopy InChI
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HEK293 cell membranes after 90 mins radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457101(CHEMBL4210241)copy SMILEScopy InChI
Affinity DataKi:  0.5nMAssay Description:Antagonist activity at human A2A receptor expressed in HEK293 cell membranes assessed as reduction in CGS-21680-induced cAMP level pretreated for 15 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457099(CHEMBL4213177)copy SMILEScopy InChI
Affinity DataKi:  0.580nMAssay Description:Antagonist activity at rat A2A receptor assessed as reduction in CGS-21680-induced cAMP level pretreated for 15 mins followed by CGS-21680 addition m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457105(CHEMBL4212278)copy SMILEScopy InChI
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HEK293 cell membranes after 90 mins radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457108(CHEMBL4216716)copy SMILEScopy InChI
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HEK293 cell membranes after 90 mins radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457104(CHEMBL4217235)copy SMILEScopy InChI
Affinity DataKi:  0.650nMAssay Description:Antagonist activity at rat A2A receptor assessed as reduction in CGS-21680-induced cAMP level pretreated for 15 mins followed by CGS-21680 addition m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457095(CHEMBL4212740)copy SMILEScopy InChI
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HEK293 cell membranes after 90 mins radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457094(CHEMBL4204531)copy SMILEScopy InChI
Affinity DataKi:  0.720nMAssay Description:Antagonist activity at rat A2A receptor assessed as reduction in CGS-21680-induced cAMP level pretreated for 15 mins followed by CGS-21680 addition m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457100(CHEMBL4218105)copy SMILEScopy InChI
Affinity DataKi:  0.740nMAssay Description:Antagonist activity at rat A2A receptor assessed as reduction in CGS-21680-induced cAMP level pretreated for 15 mins followed by CGS-21680 addition m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457102(CHEMBL4205030)copy SMILEScopy InChI
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HEK293 cell membranes after 90 mins radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457089(CHEMBL4212810)copy SMILEScopy InChI
Affinity DataKi:  0.900nMAssay Description:Antagonist activity at human A2A receptor expressed in HEK293 cell membranes assessed as reduction in CGS-21680-induced cAMP level pretreated for 15 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50232062(CHEMBL4068507)copy SMILEScopy InChI
Affinity DataKi:  0.900nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine receptor A2b expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting met...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571F7GPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50232044(CHEMBL4083317)copy SMILEScopy InChI
Affinity DataKi:  0.900nMAssay Description:Antagonist activity at human adenosine receptor A2b expressed in HEK293 cells assessed as inhibition of NECA-induced cAMP level preincubated for 15 m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571F7GPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457099(CHEMBL4213177)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HEK293 cell membranes after 90 mins radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50232044(CHEMBL4083317)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine receptor A2b expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting met...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571F7GPubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50232060(CHEMBL4095766)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Displacement of [3H]-MRS-1754 from human adenosine receptor A2b expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting met...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571F7GPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457084(CHEMBL4217248)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Displacement of [3H]ZM241385 from human A2A receptor expressed in HEK293 cell membranes after 90 mins radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50231595(CHEMBL4092832)copy SMILEScopy InChI
Affinity DataKi:  1nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in HEK293 cell membranes after 90 minsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0QKCPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457100(CHEMBL4218105)copy SMILEScopy InChI
Affinity DataKi:  1.10nMAssay Description:Antagonist activity at human A2A receptor expressed in HEK293 cell membranes assessed as reduction in CGS-21680-induced cAMP level pretreated for 15 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457103(CHEMBL4217668)copy SMILEScopy InChI
Affinity DataKi:  1.10nMAssay Description:Antagonist activity at rat A2A receptor assessed as reduction in CGS-21680-induced cAMP level pretreated for 15 mins followed by CGS-21680 addition m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457102(CHEMBL4205030)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:Antagonist activity at human A2A receptor expressed in HEK293 cell membranes assessed as reduction in CGS-21680-induced cAMP level pretreated for 15 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Advinus Therapeutics Ltd.

Curated by ChEMBL
LigandPNGBDBM50457105(CHEMBL4212278)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:Antagonist activity at rat A2A receptor assessed as reduction in CGS-21680-induced cAMP level pretreated for 15 mins followed by CGS-21680 addition m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571FMDPubMed
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