Affinity DataKi: 9.43E+3nMAssay Description:Inhibition of 5-carboxyfluorescein-labeled Flu-Bak-BH3 peptide binding to Bcl-w by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.08E+4nMAssay Description:Inhibition of 5-carboxyfluorescein-labeled Flu-Bak-BH3 peptide binding to Bcl-w by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.30E+4nMAssay Description:Inhibition of 5-carboxyfluorescein-labeled Flu-Bak-BH3 peptide binding to Bcl-w by fluorescence polarization assayMore data for this Ligand-Target Pair
Target1D-myo-inositol 2-acetamido-2-deoxy-alpha-D-glucopyranoside deacetylase(Mycobacterium tuberculosis)
University of Cape Town
Curated by ChEMBL
University of Cape Town
Curated by ChEMBL
Affinity DataKi: 1.68E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis MshB expressed in Escherichia coli BL21 after 10 mins by HPLC analysisMore data for this Ligand-Target Pair
Target1D-myo-inositol 2-acetamido-2-deoxy-alpha-D-glucopyranoside deacetylase(Mycobacterium tuberculosis)
University of Cape Town
Curated by ChEMBL
University of Cape Town
Curated by ChEMBL
Affinity DataKi: 9.40E+4nMAssay Description:Inhibition of Mycobacterium tuberculosis MshB expressed in Escherichia coli BL21 after 10 mins by HPLC analysisMore data for this Ligand-Target Pair
Target1D-myo-inositol 2-acetamido-2-deoxy-alpha-D-glucopyranoside deacetylase(Mycobacterium tuberculosis)
University of Cape Town
Curated by ChEMBL
University of Cape Town
Curated by ChEMBL
Affinity DataKi: 1.67E+5nMAssay Description:Inhibition of Mycobacterium tuberculosis MshB expressed in Escherichia coli BL21 after 10 mins by HPLC analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Antagonistic activity against RAR gamma in transcriptional activation assay with 3.2 nM TTNPBMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Antagonistic activity against RAR gamma in transcriptional activation assay with 3.2 nM TTNPBMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Binding affinity of [3H]- RA to baculovirus expressed human Retinoic acid receptor betaMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Binding affinity of [3H]- RA to baculovirus expressed human Retinoic acid receptor betaMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Antagonistic activity against RAR alpha in transcriptional activation assay with 32 nM TTNPBMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 2nMAssay Description:Antagonistic activity against RAR beta in transcriptional activation assay with 10 nM TTNPBMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Antagonistic activity against RAR gamma in transcriptional activation assay with 3.2 nM TTNPBMore data for this Ligand-Target Pair
Affinity DataIC50: 5.5nMAssay Description:Binding affinity of [3H]- RA to baculovirus expressed human RAR alphaMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 6.5nMAssay Description:Antagonistic activity against RAR beta in transcriptional activation assay with 10 nM TTNPBMore data for this Ligand-Target Pair
Affinity DataIC50: 6.5nMAssay Description:Antagonistic activity against RAR alpha in transcriptional activation assay with 32 nM TTNPBMore data for this Ligand-Target Pair
Affinity DataIC50: 7.5nMAssay Description:Antagonistic activity against RAR beta in transcriptional activation assay with 10 nM TTNPBMore data for this Ligand-Target Pair
In DepthDetails
In DepthDetails
In DepthDetails
Affinity DataIC50: 15nMAssay Description:Antagonistic activity against RAR gamma in transcriptional activation assay with 3.2 nM TTNPBMore data for this Ligand-Target Pair
In DepthDetails
Affinity DataIC50: 20nMAssay Description:Antagonistic activity against RAR alpha in transcriptional activation assay with 32 nM TTNPBMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Antagonistic activity against RAR beta in transcriptional activation assay with 10 nM TTNPBMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Antagonistic activity against RAR beta in transcriptional activation assay with 10 nM TTNPBMore data for this Ligand-Target Pair
In DepthDetails
In DepthDetails
In DepthDetails
In DepthDetails
In DepthDetails
In DepthDetails
In DepthDetails
In DepthDetails
In DepthDetails
In DepthDetails
In DepthDetails
In DepthDetails
In DepthDetails
In DepthDetails
In DepthDetails
In DepthDetails
In DepthDetails
In DepthDetails
In DepthDetails
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Morphochem AG
Curated by ChEMBL
Morphochem AG
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory concentration against ProteaseMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Morphochem AG
Curated by ChEMBL
Morphochem AG
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Evaluated for inhibition of Protease after after resynthesis and purificationMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Morphochem AG
Curated by ChEMBL
Morphochem AG
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Evaluated for inhibition of Protease after after resynthesis and purificationMore data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Morphochem AG
Curated by ChEMBL
Morphochem AG
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Evaluated for inhibition of Protease after CLND/MS correction from the crude mixtureMore data for this Ligand-Target Pair