Compile Data Set for Download or QSAR
Found 41 with Last Name = 'nikulin' and Initial = 'vi'
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470923(CHEMBL122757)copy SMILEScopy InChI
Affinity DataKi:  0.302nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52SBMPubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470917(CHEMBL120278)copy SMILEScopy InChI
Affinity DataKi:  1.5nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52SBMPubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470918(CHEMBL123596)copy SMILEScopy InChI
Affinity DataKi:  1.5nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52SBMPubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM82487(TMQ, 3',5'-Diiodo)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Binding Affinity against human beta-2 adrenergic receptor expressed in Chinese hamster ovary(CHO) cells was measured by using [125I]ICYP radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057JN4PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470916(CHEMBL121704)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52SBMPubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM82487(TMQ, 3',5'-Diiodo)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52SBMPubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470924(CHEMBL122990)copy SMILEScopy InChI
Affinity DataKi:  6.5nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52SBMPubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470919(CHEMBL332964)copy SMILEScopy InChI
Affinity DataKi:  7.80nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52SBMPubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470922(CHEMBL122992)copy SMILEScopy InChI
Affinity DataKi:  8.70nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52SBMPubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470920(CHEMBL121964)copy SMILEScopy InChI
Affinity DataKi:  12nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52SBMPubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
University of Tennessee

Curated by ChEMBL
LigandPNGBDBM82487(TMQ, 3',5'-Diiodo)copy SMILEScopy InChI
Affinity DataKi:  21nMAssay Description:Binding Affinity against human Beta-3 adrenergic receptor expressed in Chinese hamster ovary(CHO) cells was measured by using [125I]ICYP radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057JN4PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50019355(1-(3,4,5-Trimethoxy-benzyl)-1,2,3,4-tetrahydro-iso...)copy SMILEScopy InChI
Affinity DataKi:  44nMAssay Description:Binding Affinity against human beta-2 adrenergic receptor expressed in Chinese hamster ovary(CHO) cells was measured by using [125I]ICYP radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057JN4PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50019355(1-(3,4,5-Trimethoxy-benzyl)-1,2,3,4-tetrahydro-iso...)copy SMILEScopy InChI
Affinity DataKi:  44nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52SBMPubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM82487(TMQ, 3',5'-Diiodo)copy SMILEScopy InChI
Affinity DataKi:  47nMAssay Description:Binding affinity for human Platelet Thromboxane A2 / Prostaglandin (TP), by radioligand competition binding assays using [3H]-SQ 29548 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52SBMPubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
University of Tennessee

Curated by ChEMBL
LigandPNGBDBM82487(TMQ, 3',5'-Diiodo)copy SMILEScopy InChI
Affinity DataKi:  79nMAssay Description:Binding Affinity against human Beta-1 adrenergic receptor expressed in Chinese hamster ovary(CHO) cells was measured by using [125I]ICYP radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057JN4PubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
University of Tennessee

Curated by ChEMBL
LigandPNGBDBM82487(TMQ, 3',5'-Diiodo)copy SMILEScopy InChI
Affinity DataKi:  79nMAssay Description:Binding affinity for human Beta-1 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52SBMPubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
University of Tennessee

Curated by ChEMBL
LigandPNGBDBM82487(TMQ, 3',5'-Diiodo)copy SMILEScopy InChI
Affinity DataKi:  79.4nMAssay Description:Binding affinity for human Beta-1 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52SBMPubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50019355(1-(3,4,5-Trimethoxy-benzyl)-1,2,3,4-tetrahydro-iso...)copy SMILEScopy InChI
Affinity DataKi:  162nMAssay Description:Binding affinity for human Platelet Thromboxane A2 / Prostaglandin (TP), by radioligand competition binding assays using [3H]-SQ 29548 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52SBMPubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470923(CHEMBL122757)copy SMILEScopy InChI
Affinity DataKi:  178nMAssay Description:Binding affinity for human Platelet Thromboxane A2 / Prostaglandin (TP), by radioligand competition binding assays using [3H]-SQ 29548 as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52SBMPubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
University of Tennessee

Curated by ChEMBL
LigandPNGBDBM50470923(CHEMBL122757)copy SMILEScopy InChI
Affinity DataKi:  182nMAssay Description:Binding affinity for human Beta-1 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52SBMPubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470918(CHEMBL123596)copy SMILEScopy InChI
Affinity DataKi:  186nMAssay Description:Binding affinity for human Platelet Thromboxane A2 / Prostaglandin (TP), by radioligand competition binding assays using [3H]-SQ 29548 as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52SBMPubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
University of Tennessee

Curated by ChEMBL
LigandPNGBDBM50019355(1-(3,4,5-Trimethoxy-benzyl)-1,2,3,4-tetrahydro-iso...)copy SMILEScopy InChI
Affinity DataKi:  324nMAssay Description:Binding affinity for human Beta-1 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52SBMPubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
University of Tennessee

Curated by ChEMBL
LigandPNGBDBM50019355(1-(3,4,5-Trimethoxy-benzyl)-1,2,3,4-tetrahydro-iso...)copy SMILEScopy InChI
Affinity DataKi:  324nMAssay Description:Binding Affinity against human Beta-1 adrenergic receptor expressed in Chinese hamster ovary(CHO) cells was measured by using [125I]ICYP radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057JN4PubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470922(CHEMBL122992)copy SMILEScopy InChI
Affinity DataKi:  355nMAssay Description:Binding affinity for human Platelet Thromboxane A2 / Prostaglandin (TP), by radioligand competition binding assays using [3H]-SQ 29548 as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52SBMPubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50093039(4-(3,5-Diiodo-4-methoxy-benzyl)-4,5,6,7-tetrahydro...)copy SMILEScopy InChI
Affinity DataKi:  427nMAssay Description:Binding Affinity against human Beta-2 adrenergic receptor expressed in Chinese hamster ovary(CHO) cells was measured by using [125I]ICYP radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057JN4PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50472299(CHEMBL73917)copy SMILEScopy InChI
Affinity DataKi:  617nMAssay Description:Binding Affinity against human beta-2 adrenergic receptor expressed in Chinese hamster ovary(CHO) cells was measured by using [125I]ICYP radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057JN4PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM25392(4-[1-hydroxy-2-(isopropylamino)ethyl]pyrocatechol;...)copy SMILEScopy InChI
Affinity DataKi:  676nMAssay Description:Binding Affinity against human beta-2 adrenergic receptor expressed in Chinese hamster ovary(CHO) cells was measured by using [125I]ICYP radioligandMore data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
University of Tennessee

Curated by ChEMBL
LigandPNGBDBM50093039(4-(3,5-Diiodo-4-methoxy-benzyl)-4,5,6,7-tetrahydro...)copy SMILEScopy InChI
Affinity DataKi:  724nMAssay Description:Binding Affinity against human Beta-1 adrenergic receptor expressed in Chinese hamster ovary(CHO) cells was measured by using [125I]ICYP radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057JN4PubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470924(CHEMBL122990)copy SMILEScopy InChI
Affinity DataKi:  1.00E+3nMAssay Description:Binding affinity for human Platelet Thromboxane A2 / Prostaglandin (TP), by radioligand competition binding assays using [3H]-SQ 29548 as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52SBMPubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
University of Tennessee

Curated by ChEMBL
LigandPNGBDBM50093039(4-(3,5-Diiodo-4-methoxy-benzyl)-4,5,6,7-tetrahydro...)copy SMILEScopy InChI
Affinity DataKi:  1.48E+3nMAssay Description:Binding Affinity against human Beta-3 adrenergic receptor expressed in Chinese hamster ovary(CHO) cells was measured by using [125I]ICYP radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057JN4PubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470919(CHEMBL332964)copy SMILEScopy InChI
Affinity DataKi:  1.48E+3nMAssay Description:Binding affinity for human Platelet Thromboxane A2 / Prostaglandin (TP), by radioligand competition binding assays using [3H]-SQ 29548 as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52SBMPubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
University of Tennessee

Curated by ChEMBL
LigandPNGBDBM25392(4-[1-hydroxy-2-(isopropylamino)ethyl]pyrocatechol;...)copy SMILEScopy InChI
Affinity DataKi:  1.59E+3nMAssay Description:Binding Affinity against human Beta-1 adrenergic receptor expressed in Chinese hamster ovary(CHO) cells was measured by using [125I]ICYP radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057JN4PubMedDrugBank
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
University of Tennessee

Curated by ChEMBL
LigandPNGBDBM50019355(1-(3,4,5-Trimethoxy-benzyl)-1,2,3,4-tetrahydro-iso...)copy SMILEScopy InChI
Affinity DataKi:  3.72E+3nMAssay Description:Binding Affinity against human Beta-3 adrenergic receptor expressed in Chinese hamster ovary(CHO) cells was measured by using [125I]ICYP radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057JN4PubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470921(CHEMBL333438)copy SMILEScopy InChI
Affinity DataKi:  4.37E+3nMAssay Description:Binding affinity for human Beta-2 adrenergic receptor expressed in CHO cells by radioligand competition binding assays using [125I]iodocyanopindolol ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52SBMPubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470916(CHEMBL121704)copy SMILEScopy InChI
Affinity DataKi:  5.37E+3nMAssay Description:Binding affinity for human Platelet Thromboxane A2 / Prostaglandin (TP), by radioligand competition binding assays using [3H]-SQ 29548 as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52SBMPubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
University of Tennessee

Curated by ChEMBL
LigandPNGBDBM50472299(CHEMBL73917)copy SMILEScopy InChI
Affinity DataKi:  6.17E+3nMAssay Description:Binding Affinity against human Beta-1 adrenergic receptor expressed in Chinese hamster ovary(CHO) cells was measured by using [125I]ICYP radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057JN4PubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
University of Tennessee

Curated by ChEMBL
LigandPNGBDBM25392(4-[1-hydroxy-2-(isopropylamino)ethyl]pyrocatechol;...)copy SMILEScopy InChI
Affinity DataKi:  1.86E+4nMAssay Description:Binding Affinity against human Beta-3 adrenergic receptor expressed in Chinese hamster ovary(CHO) cells was measured by using [125I]ICYP radioligandMore data for this Ligand-Target Pair
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470920(CHEMBL121964)copy SMILEScopy InChI
Affinity DataKi:  1.91E+4nMAssay Description:Binding affinity for human Platelet Thromboxane A2 / Prostaglandin (TP), by radioligand competition binding assays using [3H]-SQ 29548 as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52SBMPubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470917(CHEMBL120278)copy SMILEScopy InChI
Affinity DataKi:  6.03E+4nMAssay Description:Binding affinity for human Platelet Thromboxane A2 / Prostaglandin (TP), by radioligand competition binding assays using [3H]-SQ 29548 as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52SBMPubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
University of Tennessee

Curated by ChEMBL
LigandPNGBDBM50472299(CHEMBL73917)copy SMILEScopy InChI
Affinity DataKi:  6.76E+4nMAssay Description:Binding Affinity against human Beta-3 adrenergic receptor expressed in Chinese hamster ovary(CHO) cells was measured by using [125I]ICYP radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057JN4PubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University of Tennessee-Memphis

Curated by ChEMBL
LigandPNGBDBM50470921(CHEMBL333438)copy SMILEScopy InChI
Affinity DataKi:  8.32E+4nMAssay Description:Binding affinity for human Platelet Thromboxane A2 / Prostaglandin (TP), by radioligand competition binding assays using [3H]-SQ 29548 as radioligandMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52SBMPubMed