Compile Data Set for Download or QSAR
Found 315 with Last Name = 'guarino' and Initial = 'vr'
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM176023(US10047103, 56 | US9688695, 56)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM176082(US10047103, 115 | US9688695, 115)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetRho-associated protein kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM252182(US9458110, 254)copy SMILES
Affinity DataIC50: 0.300nMAssay Description:Inhibition of ROCK2 (unknown origin) using FITC-AHA-AKRRRLSSLRA-OH peptide substrate by caliper assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J969Z7PubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM175970(US10047103, 3 | US9605024, Example 3 | US9688695, ...)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetRho-associated protein kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM251935(US9458110, 7)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMAssay Description:Inhibition of ROCK2 (unknown origin) using FITC-AHA-AKRRRLSSLRA-OH peptide substrate by caliper assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J969Z7PubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM176053(US10047103, 86 | US9688695, 86)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM176039(US10047103, 72 | US9688695, 72)copy SMILEScopy InChI
Affinity DataIC50: 0.300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetRho-associated protein kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50546544(CHEMBL4791701)copy SMILES
Affinity DataIC50: 0.400nMAssay Description:Inhibition of ROCK2 (unknown origin) using FITC-AHA-AKRRRLSSLRA-OH peptide substrate by caliper assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J969Z7PubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM175988(US10047103, 21 | US9688695, 21)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM50600792(CHEMBL5189522)copy SMILES
Affinity DataIC50: 0.400nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM176061(US10047103, 94 | US9688695, 94)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM50600788(CHEMBL5206065)copy SMILES
Affinity DataIC50: 0.400nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM176007(US10047103, 40 | US9688695, 40)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM176003(US10047103, 36 | US9688695, 36)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM286424(US9518064, Example 40)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM286418(US9518064, Example 34)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM176026(US10047103, 59 | US9688695, 59)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM176019(US10047103, 52 | US9688695, 52)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM286419(US9518064, Example 35)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM286427(US9518064, Example 43)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM175990(US10047103, 23 | US9688695, 23)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM176258(US10047103, 291 | US9688695, 291)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM176268(US10047103, 301 | US9688695, 301)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM176059(US10047103, 92 | US9688695, 92)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM50600791(CHEMBL5177223)copy SMILES
Affinity DataIC50: 0.600nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM176063(US10047103, 96 | US9688695, 96)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM175972(US10047103, 5 | US9688695, 5)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM50600784(CHEMBL5184586)copy SMILES
Affinity DataIC50: 0.630nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM286431(US9518064, Example 47)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM175989(US10047103, 22 | US9688695, 22)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM50600790(CHEMBL5171201)copy SMILES
Affinity DataIC50: 0.700nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetRho-associated protein kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM252032(US9458110, 103)copy SMILES
Affinity DataIC50: 0.700nMAssay Description:Inhibition of ROCK2 (unknown origin) using FITC-AHA-AKRRRLSSLRA-OH peptide substrate by caliper assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J969Z7PubMed
TargetRho-associated protein kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50546544(CHEMBL4791701)copy SMILES
Affinity DataIC50: 0.800nMAssay Description:Inhibition of ROCK1 (unknown origin) using FITC-AHA-AKRRRLSSLRA-OH peptide substrate by caliper assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J969Z7PubMed
TargetRho-associated protein kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM252182(US9458110, 254)copy SMILES
Affinity DataIC50: 0.800nMAssay Description:Inhibition of ROCK1 (unknown origin) using FITC-AHA-AKRRRLSSLRA-OH peptide substrate by caliper assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J969Z7PubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM176048(US10047103, 81 | US9688695, 81)copy SMILEScopy InChI
Affinity DataIC50: 0.800nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM286394(US9518064, Example 6)copy SMILEScopy InChI
Affinity DataIC50: 0.800nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM50600785(CHEMBL5173906)copy SMILES
Affinity DataIC50: 0.800nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM176032(US10047103, 65 | US9688695, 65)copy SMILEScopy InChI
Affinity DataIC50: 0.800nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM50528302(CHEMBL4551932)copy SMILEScopy InChI
Affinity DataIC50: 0.810nMAssay Description:Antagonist activity at full-length human PAR4 expressed in HEK293 cells assessed as inhibition of AYPGKF-induced intracellular calcium mobilization p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QC06ZZPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM50528303(CHEMBL4462511)copy SMILEScopy InChI
Affinity DataIC50: 0.890nMAssay Description:Antagonist activity at full-length human PAR4 expressed in HEK293 cells assessed as inhibition of AYPGKF-induced intracellular calcium mobilization p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QC06ZZPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM286482(2-Methoxy-6-(6-methoxy-4-((2-phenylpyrimidin-4-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 0.900nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetRho-associated protein kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM251935(US9458110, 7)copy SMILEScopy InChI
Affinity DataIC50: 0.900nMAssay Description:Inhibition of ROCK1 (unknown origin) using FITC-AHA-AKRRRLSSLRA-OH peptide substrate by caliper assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J969Z7PubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM50528281(CHEMBL4457190)copy SMILEScopy InChI
Affinity DataIC50: 0.980nMAssay Description:Antagonist activity at full-length human PAR4 expressed in HEK293 cells assessed as inhibition of AYPGKF-induced intracellular calcium mobilization p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QC06ZZPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM364615(US9862730, Example 73)copy SMILEScopy InChI
Affinity DataIC50: 0.990nMAssay Description:Antagonist activity at full-length human PAR4 expressed in HEK293 cells assessed as inhibition of AYPGKF-induced intracellular calcium mobilization p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QC06ZZPubMed
TargetRho-associated protein kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM252039(US9458110, 110)copy SMILES
Affinity DataIC50: 1nMAssay Description:Inhibition of ROCK2 (unknown origin) using FITC-AHA-AKRRRLSSLRA-OH peptide substrate by caliper assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J969Z7PubMed
TargetRho-associated protein kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM252036(US9458110, 107)copy SMILES
Affinity DataIC50: 1nMAssay Description:Inhibition of ROCK2 (unknown origin) using FITC-AHA-AKRRRLSSLRA-OH peptide substrate by caliper assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J969Z7PubMed
TargetRho-associated protein kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM251982(US9458110, 55)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Inhibition of ROCK2 (unknown origin) using FITC-AHA-AKRRRLSSLRA-OH peptide substrate by caliper assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J969Z7PubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM50600793(CHEMBL5205126)copy SMILES
Affinity DataIC50: 1.10nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM175971(US10047103, 4 | US9688695, 4)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
TargetProteinase-activated receptor 4(Homo sapiens (Human))TBA
LigandPNGBDBM286387(2-Methoxy-6-(6-methoxy-4-((3-(pyrimidin-5-yl)benzy...)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SWMPubMed
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