Compile Data Set for Download or QSAR
Found 107 with Last Name = 'timmerman' and Initial = 'w'
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50010594(2-Chloro-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b...)copy SMILEScopy InChI
Affinity DataIC50: 2.90nMAssay Description:Binding affinity towards 5-HT2C receptor from rat using [3H]-mesulergine as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)copy SMILEScopy InChI
Affinity DataIC50: 4.90nMAssay Description:Binding affinity towards human Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMedDrugBank
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM22871(13-chloro-10-(4-methylpiperazin-1-yl)-2-oxa-9-azat...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor from rat frontal cortex using [3H]-ketanserin as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50010594(2-Chloro-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of binding of 1.0 nM [3H]-pirenzepine to cloned human Muscarinic acetylcholine receptor M1 expressed in membranes from CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)copy SMILEScopy InChI
Affinity DataIC50: 6.5nMAssay Description:Binding affinity towards human D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)copy SMILEScopy InChI
Affinity DataIC50: 7.5nMAssay Description:Binding affinity towards Dopamine receptor D2 of rat corpus striatum using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50078061(CHEMBL73589 | Trifluoro-methanesulfonic acid 11-(4...)copy SMILEScopy InChI
Affinity DataIC50: 8nMAssay Description:Binding affinity towards human Dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)copy SMILEScopy InChI
Affinity DataIC50: 9.40nMAssay Description:Inhibition of binding of 1.0 nM [3H]-pirenzepine to cloned human Muscarinic acetylcholine receptor M1 expressed in membranes from CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Binding affinity towards human Dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
TargetD(1A) dopamine receptor(RAT)
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50010594(2-Chloro-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Binding affinity towards D1 CNS receptor of rat corpus striatum using [3H]-SCH-23,390 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Binding affinity towards 5-HT2C receptor from rat using [3H]-mesulergine as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50061558(2-Methoxy-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[...)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor from rat frontal cortex using [3H]-ketanserin as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor from rat frontal cortex using [3H]-ketanserin as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50010594(2-Chloro-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b...)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor from rat frontal cortex using [3H]-ketanserin as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50078063(CHEMBL70319 | Trifluoro-methanesulfonic acid 8-chl...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Binding affinity towards 5-HT2C receptor from rat using [3H]-mesulergine as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50010594(2-Chloro-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Binding affinity towards Dopamine receptor D2 of rat corpus striatum using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM22871(13-chloro-10-(4-methylpiperazin-1-yl)-2-oxa-9-azat...)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Compound was tested in vitro for its binding affinity towards human Dopamine receptor D4.2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMedDrugBank
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50061555(8-Methoxy-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[...)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of binding of 1.0 nM [3H]-pirenzepine to cloned human Muscarinic acetylcholine receptor M1 expressed in membranes from CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50061558(2-Methoxy-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[...)copy SMILEScopy InChI
Affinity DataIC50: 21nMAssay Description:Binding affinity towards 5-HT2C receptor from rat using [3H]-mesulergine as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM22871(13-chloro-10-(4-methylpiperazin-1-yl)-2-oxa-9-azat...)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Binding affinity towards human Dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50078063(CHEMBL70319 | Trifluoro-methanesulfonic acid 8-chl...)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor from rat frontal cortex using [3H]-ketanserin as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50078061(CHEMBL73589 | Trifluoro-methanesulfonic acid 11-(4...)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Binding affinity towards human Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
TargetHistamine H1 receptor(RAT)
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Binding affinity towards histamine H1 receptor from rat brain membranes using [3H]-mepyramine as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50061557(11-(4-Methyl-piperazin-1-yl)-5H-dibenzo[b,e][1,4]d...)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Inhibition of binding of 1.0 nM [3H]-pirenzepine to cloned human Muscarinic acetylcholine receptor M1 expressed in membranes from CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50078062(CHEMBL430798 | Trifluoro-methanesulfonic acid 11-(...)copy SMILEScopy InChI
Affinity DataIC50: 29nMAssay Description:Binding affinity towards human Dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50078063(CHEMBL70319 | Trifluoro-methanesulfonic acid 8-chl...)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Binding affinity towards human Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50061559(CHEMBL72292 | Trifluoro-methanesulfonic acid 11-(4...)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:Binding affinity towards Dopamine receptor D2 of rat corpus striatum using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50078061(CHEMBL73589 | Trifluoro-methanesulfonic acid 11-(4...)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Binding affinity towards Dopamine receptor D2 of rat corpus striatum using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50010594(2-Chloro-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[b...)copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:Binding affinity towards human Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50061559(CHEMBL72292 | Trifluoro-methanesulfonic acid 11-(4...)copy SMILEScopy InChI
Affinity DataIC50: 34nMAssay Description:Binding affinity towards 5-HT2C receptor from rat using [3H]-mesulergine as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50061560(CHEMBL310712 | Trifluoro-methanesulfonic acid 11-(...)copy SMILEScopy InChI
Affinity DataIC50: 35nMAssay Description:Inhibition of binding of 1.0 nM [3H]-pirenzepine to cloned human Muscarinic acetylcholine receptor M1 expressed in membranes from CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50061556(11-(4-Methyl-piperazin-1-yl)-5H-dibenzo[b,e][1,4]d...)copy SMILEScopy InChI
Affinity DataIC50: 35nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor from rat frontal cortex using [3H]-ketanserin as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
TargetD(1A) dopamine receptor(RAT)
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)copy SMILEScopy InChI
Affinity DataIC50: 36nMAssay Description:Binding affinity towards D1 CNS receptor of rat corpus striatum using [3H]-SCH-23,390 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50061556(11-(4-Methyl-piperazin-1-yl)-5H-dibenzo[b,e][1,4]d...)copy SMILEScopy InChI
Affinity DataIC50: 37nMAssay Description:Inhibition of binding of 1.0 nM [3H]-pirenzepine to cloned human Muscarinic acetylcholine receptor M1 expressed in membranes from CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50078065(CHEMBL70609 | Methanesulfonic acid 11-(4-methyl-pi...)copy SMILEScopy InChI
Affinity DataIC50: 38nMAssay Description:Inhibition of binding of 1.0 nM [3H]-pirenzepine to cloned human Muscarinic acetylcholine receptor M1 expressed in membranes from CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50061558(2-Methoxy-11-(4-methyl-piperazin-1-yl)-5H-dibenzo[...)copy SMILEScopy InChI
Affinity DataIC50: 39nMAssay Description:Inhibition of binding of 1.0 nM [3H]-pirenzepine to cloned human Muscarinic acetylcholine receptor M1 expressed in membranes from CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50078062(CHEMBL430798 | Trifluoro-methanesulfonic acid 11-(...)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Binding affinity towards Dopamine receptor D2 of rat corpus striatum using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50061559(CHEMBL72292 | Trifluoro-methanesulfonic acid 11-(4...)copy SMILEScopy InChI
Affinity DataIC50: 43nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor from rat frontal cortex using [3H]-ketanserin as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50078063(CHEMBL70319 | Trifluoro-methanesulfonic acid 8-chl...)copy SMILEScopy InChI
Affinity DataIC50: 43nMAssay Description:Binding affinity towards Dopamine receptor D2 of rat corpus striatum using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
TargetHistamine H1 receptor(RAT)
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50061559(CHEMBL72292 | Trifluoro-methanesulfonic acid 11-(4...)copy SMILEScopy InChI
Affinity DataIC50: 47nMAssay Description:Binding affinity towards histamine H1 receptor from rat brain membranes using [3H]-mepyramine as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50078062(CHEMBL430798 | Trifluoro-methanesulfonic acid 11-(...)copy SMILEScopy InChI
Affinity DataIC50: 48nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor from rat frontal cortex using [3H]-ketanserin as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50078062(CHEMBL430798 | Trifluoro-methanesulfonic acid 11-(...)copy SMILEScopy InChI
Affinity DataIC50: 52nMAssay Description:Binding affinity towards human Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50078063(CHEMBL70319 | Trifluoro-methanesulfonic acid 8-chl...)copy SMILEScopy InChI
Affinity DataIC50: 52nMAssay Description:Binding affinity towards human Dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)copy SMILEScopy InChI
Affinity DataIC50: 52nMAssay Description:Binding affinity towards human D4.2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMedDrugBank
TargetD(3) dopamine receptor(Homo sapiens (Human))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50061559(CHEMBL72292 | Trifluoro-methanesulfonic acid 11-(4...)copy SMILEScopy InChI
Affinity DataIC50: 53nMAssay Description:Binding affinity towards human Dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM22871(13-chloro-10-(4-methylpiperazin-1-yl)-2-oxa-9-azat...)copy SMILEScopy InChI
Affinity DataIC50: 54nMAssay Description:Compound was tested in vitro for its binding affinity towards human Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMedDrugBank
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50078063(CHEMBL70319 | Trifluoro-methanesulfonic acid 8-chl...)copy SMILEScopy InChI
Affinity DataIC50: 54nMAssay Description:Inhibition of binding of 1.0 nM [3H]-pirenzepine to cloned human Muscarinic acetylcholine receptor M1 expressed in membranes from CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)copy SMILEScopy InChI
Affinity DataIC50: 55nMAssay Description:Binding affinity towards 5-hydroxytryptamine 2A receptor from rat frontal cortex using [3H]-ketanserin as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
TargetD(1A) dopamine receptor(RAT)
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50061559(CHEMBL72292 | Trifluoro-methanesulfonic acid 11-(4...)copy SMILEScopy InChI
Affinity DataIC50: 64nMAssay Description:Binding affinity towards D1 CNS receptor of rat corpus striatum using [3H]-SCH-23,390 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
TargetD(1A) dopamine receptor(RAT)
University of Göteborg

Curated by ChEMBL
LigandPNGBDBM50078062(CHEMBL430798 | Trifluoro-methanesulfonic acid 11-(...)copy SMILEScopy InChI
Affinity DataIC50: 66nMAssay Description:Binding affinity towards D1 CNS receptor of rat corpus striatum using [3H]-SCH-23,390 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0MH7PubMed
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