Compile Data Set for Download or QSAR
Found 346 with Last Name = 'tansey' and Initial = 'wp'
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605347(CHEMBL5174178)copy SMILES
Affinity DataKi: <0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605348(CHEMBL5183319)copy SMILES
Affinity DataKi: <0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605346(CHEMBL5177738)copy SMILES
Affinity DataKi: <0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605343(CHEMBL5190556)copy SMILES
Affinity DataKi:  0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605336(CHEMBL5202831)copy SMILES
Affinity DataKi: <0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605332(CHEMBL5195031)copy SMILES
Affinity DataKi: <0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605331(CHEMBL5190578)copy SMILES
Affinity DataKi: <0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605330(CHEMBL5201192)copy SMILES
Affinity DataKi: <0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605325(CHEMBL5199203)copy SMILES
Affinity DataKi: <0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605323(CHEMBL5174357)copy SMILES
Affinity DataKi: <0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50520131(CHEMBL4588661)copy SMILEScopy InChI
Affinity DataKi: <0.0200nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605356(CHEMBL5170071)copy SMILES
Affinity DataKi: <0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605355(CHEMBL5170717)copy SMILES
Affinity DataKi: <0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605350(CHEMBL5177656)copy SMILES
Affinity DataKi: <0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605353(CHEMBL5190717)copy SMILES
Affinity DataKi: <0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605352(CHEMBL5198319)copy SMILES
Affinity DataKi: <0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605350(CHEMBL5177656)copy SMILES
Affinity DataKi: <0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605349(CHEMBL5191181)copy SMILES
Affinity DataKi: <0.0200nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605322(CHEMBL5169425)copy SMILES
Affinity DataKi:  0.0220nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605327(CHEMBL5181314)copy SMILES
Affinity DataKi:  0.0230nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605329(CHEMBL5186072)copy SMILES
Affinity DataKi:  0.0250nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605339(CHEMBL5171051)copy SMILES
Affinity DataKi:  0.0280nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605354(CHEMBL5179388)copy SMILES
Affinity DataKi:  0.0280nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605337(CHEMBL5192283)copy SMILES
Affinity DataKi:  0.0280nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605324(CHEMBL5182982)copy SMILES
Affinity DataKi:  0.0290nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605351(CHEMBL5180435)copy SMILES
Affinity DataKi:  0.0290nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605318(CHEMBL5171315)copy SMILES
Affinity DataKi:  0.0330nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605319(CHEMBL5171953)copy SMILES
Affinity DataKi:  0.0350nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605320(CHEMBL5202878)copy SMILES
Affinity DataKi:  0.0360nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605342(CHEMBL5194215)copy SMILES
Affinity DataKi:  0.0390nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50520121(CHEMBL4441671 | US10844044, Example 1)copy SMILEScopy InChI
Affinity DataKi:  0.0440nMAssay Description:Competitive inhibition of human N-terminal His6-SUMO tagged WDR5 (22 to 334 residues) expressed in Escherichia coli BL21-Gold(DE3) cells using 10-mer...More data for this Ligand-Target Pair
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605326(CHEMBL5206455)copy SMILES
Affinity DataKi:  0.0460nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605321(CHEMBL5182077)copy SMILES
Affinity DataKi:  0.0550nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605345(CHEMBL5190202)copy SMILES
Affinity DataKi:  0.0640nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605328(CHEMBL5199310)copy SMILES
Affinity DataKi:  0.210nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605341(CHEMBL5208340)copy SMILES
Affinity DataKi:  0.230nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605344(CHEMBL5171801)copy SMILES
Affinity DataKi:  0.590nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50465552(CHEMBL4291641 | US10501466, Example B29)copy SMILEScopy InChI
Affinity DataKi:  0.902nMAssay Description:A fluorescence polarization anisotropy (FPA) assay that measures the displacement of either a FITC-labeled MLL-derived peptide or a more potent 10mer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2319Z71US Patent
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50465552(CHEMBL4291641 | US10501466, Example B29)copy SMILEScopy InChI
Affinity DataKi:  0.902nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD21KTPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605317(CHEMBL4116919)copy SMILES
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50465552(CHEMBL4291641 | US10501466, Example B29)copy SMILEScopy InChI
Affinity DataKi: <1nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD21KTPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM423380(US10501466, Example B15)copy SMILEScopy InChI
Affinity DataKi:  2.37nMAssay Description:A fluorescence polarization anisotropy (FPA) assay that measures the displacement of either a FITC-labeled MLL-derived peptide or a more potent 10mer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2319Z71US Patent
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50465585(CHEMBL4279907 | US10501466, Example B11)copy SMILEScopy InChI
Affinity DataKi:  2.5nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD21KTPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50465585(CHEMBL4279907 | US10501466, Example B11)copy SMILEScopy InChI
Affinity DataKi:  2.66nMAssay Description:A fluorescence polarization anisotropy (FPA) assay that measures the displacement of either a FITC-labeled MLL-derived peptide or a more potent 10mer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2319Z71US Patent
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50465585(CHEMBL4279907 | US10501466, Example B11)copy SMILEScopy InChI
Affinity DataKi:  2.70nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD21KTPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50465584(CHEMBL4293572)copy SMILEScopy InChI
Affinity DataKi:  2.80nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD21KTPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM423371(US10501466, Example B6)copy SMILEScopy InChI
Affinity DataKi:  3.35nMAssay Description:A fluorescence polarization anisotropy (FPA) assay that measures the displacement of either a FITC-labeled MLL-derived peptide or a more potent 10mer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2319Z71US Patent
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50605338(CHEMBL5202465)copy SMILES
Affinity DataKi:  3.40nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ153MPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50465593(CHEMBL4283374)copy SMILEScopy InChI
Affinity DataKi:  3.5nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD21KTPubMed
TargetWD repeat-containing protein 5(Homo sapiens (Human))TBA
LigandPNGBDBM50465555(CHEMBL4287817)copy SMILEScopy InChI
Affinity DataKi:  4.90nMAssay Description:Binding affinity to N-terminal 6x-His-SUMO tagged WDR5 delta23 deletion mutant (24 to 334 residues) (unknown origin) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD21KTPubMed
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