Compile Data Set for Download or QSAR
Found 161 with Last Name = 'formosa' and Initial = 'x'
TargetAcetylcholinesterase(Homo sapiens (Human))
Universitat de Barcelona

Curated by ChEMBL
LigandPNGBDBM50379268(CHEMBL3216556)copy SMILEScopy InChI
Affinity DataKi:  1.5nMAssay Description:Competitive inhibition of human recombinant AChE by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26974KHPubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Laboratori de Qu�mica Farmac�utica (Unitat Associada al CSIC)

Curated by ChEMBL
LigandPNGBDBM50271142(6-Chloro-9-[(3-{4-[(5,6-Dimethoxy-1-oxoindan-2-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 0.0900nMAssay Description:Inhibition of bovine erythrocyte AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76DGKPubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universitat de Barcelona

Curated by ChEMBL
LigandPNGBDBM50271142(6-Chloro-9-[(3-{4-[(5,6-Dimethoxy-1-oxoindan-2-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 0.270nMAssay Description:Inhibition of human erythrocyte AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76DGKPubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Laboratori de Qu�mica Farmac�utica (Unitat Associada al CSIC)

Curated by ChEMBL
LigandPNGBDBM50271140(9-[(3-{4-[(5,6-Dimethoxy-1-oxoindan-2-yl)methyl]pi...)copy SMILEScopy InChI
Affinity DataIC50: 0.290nMAssay Description:Inhibition of bovine erythrocyte AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76DGKPubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universitat de Barcelona

Curated by ChEMBL
LigandPNGBDBM10590(3-Chloro-6,7,10,11-tetrahydro-9-methyl-12-{{3-{N-{...)copy SMILEScopy InChI
Affinity DataIC50: 0.290nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21N7ZB6PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universitat de Barcelona

Curated by ChEMBL
LigandPNGBDBM10590(3-Chloro-6,7,10,11-tetrahydro-9-methyl-12-{{3-{N-{...)copy SMILEScopy InChI
Affinity DataIC50: 0.310nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as substrate preincubated for 20 mins prior substrate addition measured after 5 m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26974KHPubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universitat de Barcelona

Curated by ChEMBL
LigandPNGBDBM10586(3-Chloro-6,7,10,11-tetrahydro-9-methyl-12-{{3-{N-{...)copy SMILEScopy InChI
Affinity DataIC50: 0.320nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21N7ZB6PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universitat de Barcelona

Curated by ChEMBL
LigandPNGBDBM10588(3-Chloro-6,7,10,11-tetrahydro-9-methyl-12-{{7-[(6-...)copy SMILEScopy InChI
Affinity DataIC50: 0.330nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21N7ZB6PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universitat de Barcelona

Curated by ChEMBL
LigandPNGBDBM10585(3-Chloro-6,7,10,11-tetrahydro-9-methyl-12-{{8-[(1,...)copy SMILEScopy InChI
Affinity DataIC50: 0.330nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21N7ZB6PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universitat de Barcelona

Curated by ChEMBL
LigandPNGBDBM10584(3-Chloro-6,7,10,11-tetrahydro-9-methyl-12-{{7-[(1,...)copy SMILEScopy InChI
Affinity DataIC50: 0.340nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21N7ZB6PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universitat de Barcelona

Curated by ChEMBL
LigandPNGBDBM10589(3-Chloro-6,7,10,11-tetrahydro-9-methyl-12-{{8-[(6-...)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21N7ZB6PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universitat de Barcelona

Curated by ChEMBL
LigandPNGBDBM10586(3-Chloro-6,7,10,11-tetrahydro-9-methyl-12-{{3-{N-{...)copy SMILEScopy InChI
Affinity DataIC50: 0.420nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as substrate preincubated for 20 mins prior substrate addition measured after 5 m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26974KHPubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universitat de Barcelona

Curated by ChEMBL
LigandPNGBDBM50379273(CHEMBL1994202 | US9238626, (-)-Huprine Y HCl)copy SMILEScopy InChI
Affinity DataIC50: 0.430nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as substrate preincubated for 20 mins prior substrate addition measured after 5 m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26974KHPubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universitat de Barcelona

Curated by ChEMBL
LigandPNGBDBM10587(3-Chloro-6,7,10,11-tetrahydro-9-methyl-12-{{6-[(6-...)copy SMILEScopy InChI
Affinity DataIC50: 0.450nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21N7ZB6PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universitat de Barcelona

Curated by ChEMBL
LigandPNGBDBM10583(3-Chloro-6,7,10,11-tetrahydro-9-methyl-12-{{6-[(1,...)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21N7ZB6PubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Laboratori de Qu�mica Farmac�utica (Unitat Associada al CSIC)

Curated by ChEMBL
LigandPNGBDBM50271141(6-Chloro-9-[(2-{4-[(5,6-dimethoxy-1-oxoindan-2-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 0.570nMAssay Description:Inhibition of bovine erythrocyte AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76DGKPubMed
TargetCholinesterase(Homo sapiens (Human))
Laboratori de Qu�mica Farmac�utica (Unitat Associada al CSIC)

Curated by ChEMBL
LigandPNGBDBM9063(5,6-Dimethoxy-2-{[7-(1,2,3,4-tetrahydro-acridin-9-...)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:Inhibition of human serum BChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76DGKPubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universitat de Barcelona

Curated by ChEMBL
LigandPNGBDBM50271141(6-Chloro-9-[(2-{4-[(5,6-dimethoxy-1-oxoindan-2-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 0.670nMAssay Description:Inhibition of human erythrocyte AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76DGKPubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universitat de Barcelona

Curated by ChEMBL
LigandPNGBDBM50200340((+/-)-huprine Y-HCl | (+/-)-huprineY hydrochloride...)copy SMILEScopy InChI
Affinity DataIC50: 0.690nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as substrate preincubated for 20 mins prior substrate addition measured after 5 m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26974KHPubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universitat de Barcelona

Curated by ChEMBL
LigandPNGBDBM10587(3-Chloro-6,7,10,11-tetrahydro-9-methyl-12-{{6-[(6-...)copy SMILEScopy InChI
Affinity DataIC50: 0.740nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as substrate preincubated for 20 mins prior substrate addition measured after 5 m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26974KHPubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universitat de Barcelona

Curated by ChEMBL
LigandPNGBDBM10592(7-chloro-15-methyl-10-azatetracyclo[11.3.1.0^{2,11...)copy SMILEScopy InChI
Affinity DataIC50: 0.780nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21N7ZB6PubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Laboratori de Qu�mica Farmac�utica (Unitat Associada al CSIC)

Curated by ChEMBL
LigandPNGBDBM50271192(6-Chloro-9-[(3-{4-[(5,6-dimethoxyindan-2-yl)methyl...)copy SMILEScopy InChI
Affinity DataIC50: 0.820nMAssay Description:Inhibition of bovine erythrocyte AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76DGKPubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Laboratori de Qu�mica Farmac�utica (Unitat Associada al CSIC)

Curated by ChEMBL
LigandPNGBDBM50271190(9-[(3-{4-[(5,6-dimethoxyindan-2-yl)methyl]piperidi...)copy SMILEScopy InChI
Affinity DataIC50: 0.820nMAssay Description:Inhibition of bovine erythrocyte AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76DGKPubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universitat de Barcelona

Curated by ChEMBL
LigandPNGBDBM10582(15-ethyl-N-[8-(1,2,3,4-tetrahydroacridin-9-ylamino...)copy SMILEScopy InChI
Affinity DataIC50: 0.820nMpH: 8.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21N7ZB6PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universitat de Barcelona

Curated by ChEMBL
LigandPNGBDBM50271140(9-[(3-{4-[(5,6-Dimethoxy-1-oxoindan-2-yl)methyl]pi...)copy SMILEScopy InChI
Affinity DataIC50: 0.880nMAssay Description:Inhibition of human erythrocyte AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76DGKPubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universitat de Barcelona

Curated by ChEMBL
LigandPNGBDBM10583(3-Chloro-6,7,10,11-tetrahydro-9-methyl-12-{{6-[(1,...)copy SMILEScopy InChI
Affinity DataIC50: 0.890nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as substrate preincubated for 20 mins prior substrate addition measured after 5 m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26974KHPubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universitat de Barcelona

Curated by ChEMBL
LigandPNGBDBM50271192(6-Chloro-9-[(3-{4-[(5,6-dimethoxyindan-2-yl)methyl...)copy SMILEScopy InChI
Affinity DataIC50: 1.06nMAssay Description:Inhibition of human erythrocyte AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76DGKPubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universitat de Barcelona

Curated by ChEMBL
LigandPNGBDBM10589(3-Chloro-6,7,10,11-tetrahydro-9-methyl-12-{{8-[(6-...)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as substrate preincubated for 20 mins prior substrate addition measured after 5 m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26974KHPubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universitat de Barcelona

Curated by ChEMBL
LigandPNGBDBM10585(3-Chloro-6,7,10,11-tetrahydro-9-methyl-12-{{8-[(1,...)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as substrate preincubated for 20 mins prior substrate addition measured after 5 m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26974KHPubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Laboratori de Qu�mica Farmac�utica (Unitat Associada al CSIC)

Curated by ChEMBL
LigandPNGBDBM50377921(SODIUM NITROPRUSSIDE)copy SMILEScopy InChI
Affinity DataIC50: 1.74nMAssay Description:Inhibition of bovine erythrocyte AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76DGKPubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Laboratori de Qu�mica Farmac�utica (Unitat Associada al CSIC)

Curated by ChEMBL
LigandPNGBDBM50271191(6-Chloro-9-[(2-{4-[(5,6-dimethoxyindan-2-yl)methyl...)copy SMILEScopy InChI
Affinity DataIC50: 1.86nMAssay Description:Inhibition of bovine erythrocyte AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76DGKPubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universitat de Barcelona

Curated by ChEMBL
LigandPNGBDBM10584(3-Chloro-6,7,10,11-tetrahydro-9-methyl-12-{{7-[(1,...)copy SMILEScopy InChI
Affinity DataIC50: 1.90nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as substrate preincubated for 20 mins prior substrate addition measured after 5 m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26974KHPubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universitat de Barcelona

Curated by ChEMBL
LigandPNGBDBM50271190(9-[(3-{4-[(5,6-dimethoxyindan-2-yl)methyl]piperidi...)copy SMILEScopy InChI
Affinity DataIC50: 2.16nMAssay Description:Inhibition of human erythrocyte AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76DGKPubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Laboratori de Qu�mica Farmac�utica (Unitat Associada al CSIC)

Curated by ChEMBL
LigandPNGBDBM50271189(9-[(2-{4-[(5,6-Dimethoxyindan-2-yl)methyl]piperidi...)copy SMILEScopy InChI
Affinity DataIC50: 2.28nMAssay Description:Inhibition of bovine erythrocyte AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76DGKPubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universitat de Barcelona

Curated by ChEMBL
LigandPNGBDBM50271191(6-Chloro-9-[(2-{4-[(5,6-dimethoxyindan-2-yl)methyl...)copy SMILEScopy InChI
Affinity DataIC50: 2.60nMAssay Description:Inhibition of human erythrocyte AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76DGKPubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universitat de Barcelona

Curated by ChEMBL
LigandPNGBDBM50027470(CHEMBL3216778)copy SMILEScopy InChI
Affinity DataIC50: 3.30nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as substrate preincubated for 20 mins prior substrate addition measured after 5 m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26974KHPubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universitat de Barcelona

Curated by ChEMBL
LigandPNGBDBM10588(3-Chloro-6,7,10,11-tetrahydro-9-methyl-12-{{7-[(6-...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as substrate preincubated for 20 mins prior substrate addition measured after 5 m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26974KHPubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universitat de Barcelona

Curated by ChEMBL
LigandPNGBDBM50377921(SODIUM NITROPRUSSIDE)copy SMILEScopy InChI
Affinity DataIC50: 4.04nMAssay Description:Inhibition of human erythrocyte AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76DGKPubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universitat de Barcelona

Curated by ChEMBL
LigandPNGBDBM50027471(CHEMBL3216554)copy SMILEScopy InChI
Affinity DataIC50: 4.20nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as substrate preincubated for 20 mins prior substrate addition measured after 5 m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26974KHPubMed
TargetCholinesterase(Homo sapiens (Human))
Laboratori de Qu�mica Farmac�utica (Unitat Associada al CSIC)

Curated by ChEMBL
LigandPNGBDBM10585(3-Chloro-6,7,10,11-tetrahydro-9-methyl-12-{{8-[(1,...)copy SMILEScopy InChI
Affinity DataIC50: 4.74nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21N7ZB6PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universitat de Barcelona

Curated by ChEMBL
LigandPNGBDBM50271189(9-[(2-{4-[(5,6-Dimethoxyindan-2-yl)methyl]piperidi...)copy SMILEScopy InChI
Affinity DataIC50: 5.13nMAssay Description:Inhibition of human erythrocyte AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76DGKPubMed
TargetCholinesterase(Homo sapiens (Human))
Laboratori de Qu�mica Farmac�utica (Unitat Associada al CSIC)

Curated by ChEMBL
LigandPNGBDBM10582(15-ethyl-N-[8-(1,2,3,4-tetrahydroacridin-9-ylamino...)copy SMILEScopy InChI
Affinity DataIC50: 5.55nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21N7ZB6PubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Laboratori de Qu�mica Farmac�utica (Unitat Associada al CSIC)

Curated by ChEMBL
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)copy SMILEScopy InChI
Affinity DataIC50: 5.70nMAssay Description:Inhibition of rat cortex AChEMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Bos taurus (bovine))
Laboratori de Qu�mica Farmac�utica (Unitat Associada al CSIC)

Curated by ChEMBL
LigandPNGBDBM8987(6-chloro-1,2,3,4-tetrahydroacridin-9-amine | 6-chl...)copy SMILEScopy InChI
Affinity DataIC50: 5.73nMpH: 8.0 T: 2°CAssay Description:AChE inhibitory activity was evaluated spectrophotometrically by the method of Ellman, using AChE from bovine or human erythrocytes and acetylthiocho...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2707ZSBPubMed
TargetAcetylcholinesterase(Bos taurus (bovine))
Laboratori de Qu�mica Farmac�utica (Unitat Associada al CSIC)

Curated by ChEMBL
LigandPNGBDBM8987(6-chloro-1,2,3,4-tetrahydroacridin-9-amine | 6-chl...)copy SMILEScopy InChI
Affinity DataIC50: 5.73nMAssay Description:Inhibition of bovine erythrocyte AChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76DGKPubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Laboratori de Qu�mica Farmac�utica (Unitat Associada al CSIC)

Curated by ChEMBL
LigandPNGBDBM8979(CHEMBL486901 | N-[2-(1-benzylpiperidin-4-yl)ethyl]...)copy SMILEScopy InChI
Affinity DataIC50: 6nMAssay Description:Inhibition of rat cortex AChEMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76DGKPubMed
TargetCholinesterase(Homo sapiens (Human))
Laboratori de Qu�mica Farmac�utica (Unitat Associada al CSIC)

Curated by ChEMBL
LigandPNGBDBM10584(3-Chloro-6,7,10,11-tetrahydro-9-methyl-12-{{7-[(1,...)copy SMILEScopy InChI
Affinity DataIC50: 6.70nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21N7ZB6PubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Universitat de Barcelona

Curated by ChEMBL
LigandPNGBDBM31895(Pyrano[3,2-c]quinoline-6-chlorotacrine hybrid, 20....)copy SMILEScopy InChI
Affinity DataIC50: 7.03nMpH: 8.0 T: 2°CAssay Description:AChE inhibitory activity was evaluated spectrophotometrically by the method of Ellman, using AChE from bovine or human erythrocytes and acetylthiocho...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2707ZSBPubMed
TargetCholinesterase(Homo sapiens (Human))
Laboratori de Qu�mica Farmac�utica (Unitat Associada al CSIC)

Curated by ChEMBL
LigandPNGBDBM50271190(9-[(3-{4-[(5,6-dimethoxyindan-2-yl)methyl]piperidi...)copy SMILEScopy InChI
Affinity DataIC50: 7.25nMAssay Description:Inhibition of human serum BChE by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76DGKPubMed
TargetCholinesterase(Homo sapiens (Human))
Laboratori de Qu�mica Farmac�utica (Unitat Associada al CSIC)

Curated by ChEMBL
LigandPNGBDBM10588(3-Chloro-6,7,10,11-tetrahydro-9-methyl-12-{{7-[(6-...)copy SMILEScopy InChI
Affinity DataIC50: 7.38nMAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21N7ZB6PubMed
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