Compile Data Set for Download or QSAR
Found 124 with Last Name = 'li' and Initial = 'xq'
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Dalian University of Technology

Curated by ChEMBL
LigandPNGBDBM50351809(CHEMBL1824190)copy SMILEScopy InChI
Affinity DataKi:  24nMAssay Description:Displacement of FAM-Bid peptide from human Mcl-1 after 30 mins by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6D8WPubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Dalian University of Technology

Curated by ChEMBL
LigandPNGBDBM50336576(3-Thiomorpholin-8-oxo-8H-acenaphtho[1,2-b]pyrrole-...)copy SMILEScopy InChI
Affinity DataKi:  58nMAssay Description:Displacement of FAM-Bid peptide from human Mcl-1 after 30 mins by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6D8WPubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Dalian University of Technology

Curated by ChEMBL
LigandPNGBDBM50336580(CHEMBL1672071 | Isopropyl-3-(4-isopropylphenoxy)-8...)copy SMILEScopy InChI
Affinity DataKi:  99nMAssay Description:Displacement of FAM-Bid peptide from human Mcl-1 after 30 mins by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6D8WPubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Dalian University of Technology

Curated by ChEMBL
LigandPNGBDBM50336579(3-(4-methoxyphenoxy)-8-oxo-8H-acenaphtho[1,2-b]pyr...)copy SMILEScopy InChI
Affinity DataKi:  122nMAssay Description:Displacement of FAM-Bid peptide from human Mcl-1 after 30 mins by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6D8WPubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Dalian University of Technology

Curated by ChEMBL
LigandPNGBDBM50351805(CHEMBL1824188)copy SMILEScopy InChI
Affinity DataKi:  149nMAssay Description:Displacement of FAM-Bid peptide from human Mcl-1 after 30 mins by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6D8WPubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Dalian University of Technology

Curated by ChEMBL
LigandPNGBDBM50351809(CHEMBL1824190)copy SMILEScopy InChI
Affinity DataKi:  158nMAssay Description:Displacement of FAM-Bid peptide from human recombinant Bcl2 after 30 mins by by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6D8WPubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Dalian University of Technology

Curated by ChEMBL
LigandPNGBDBM50336577(3-(p-tolyloxy)-8-oxo-8H-acenaphtho[1,2-b]pyrrole-9...)copy SMILEScopy InChI
Affinity DataKi:  174nMAssay Description:Displacement of FAM-Bid peptide from human Mcl-1 after 30 mins by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6D8WPubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Dalian University of Technology

Curated by ChEMBL
LigandPNGBDBM50351806(CHEMBL1824187)copy SMILEScopy InChI
Affinity DataKi:  213nMAssay Description:Displacement of FAM-Bid peptide from human Mcl-1 after 30 mins by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6D8WPubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Dalian University of Technology

Curated by ChEMBL
LigandPNGBDBM50336580(CHEMBL1672071 | Isopropyl-3-(4-isopropylphenoxy)-8...)copy SMILEScopy InChI
Affinity DataKi:  252nMAssay Description:Displacement of FAM-Bid peptide from human recombinant Bcl2 after 30 mins by by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6D8WPubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Dalian University of Technology

Curated by ChEMBL
LigandPNGBDBM50336578(3-(biphenyl-4-yloxy)-8-oxo-8H-acenaphtho[1,2-b]pyr...)copy SMILEScopy InChI
Affinity DataKi:  278nMAssay Description:Displacement of FAM-Bid peptide from human recombinant Bcl2 after 30 mins by by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6D8WPubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Dalian University of Technology

Curated by ChEMBL
LigandPNGBDBM50336579(3-(4-methoxyphenoxy)-8-oxo-8H-acenaphtho[1,2-b]pyr...)copy SMILEScopy InChI
Affinity DataKi:  304nMAssay Description:Displacement of FAM-Bid peptide from human recombinant Bcl2 after 30 mins by by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6D8WPubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Dalian University of Technology

Curated by ChEMBL
LigandPNGBDBM50336576(3-Thiomorpholin-8-oxo-8H-acenaphtho[1,2-b]pyrrole-...)copy SMILEScopy InChI
Affinity DataKi:  310nMAssay Description:Displacement of FAM-Bid peptide from human recombinant Bcl2 after 30 mins by by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6D8WPubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Dalian University of Technology

Curated by ChEMBL
LigandPNGBDBM50351808(CHEMBL1824189)copy SMILEScopy InChI
Affinity DataKi:  375nMAssay Description:Displacement of FAM-Bid peptide from human Mcl-1 after 30 mins by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6D8WPubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Dalian University of Technology

Curated by ChEMBL
LigandPNGBDBM50351807(CHEMBL1824186)copy SMILEScopy InChI
Affinity DataKi:  445nMAssay Description:Displacement of FAM-Bid peptide from human Mcl-1 after 30 mins by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6D8WPubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Dalian University of Technology

Curated by ChEMBL
LigandPNGBDBM50336577(3-(p-tolyloxy)-8-oxo-8H-acenaphtho[1,2-b]pyrrole-9...)copy SMILEScopy InChI
Affinity DataKi:  445nMAssay Description:Displacement of FAM-Bid peptide from human recombinant Bcl2 after 30 mins by by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6D8WPubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Dalian University of Technology

Curated by ChEMBL
LigandPNGBDBM50351805(CHEMBL1824188)copy SMILEScopy InChI
Affinity DataKi:  886nMAssay Description:Displacement of FAM-Bid peptide from human recombinant Bcl2 after 30 mins by by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6D8WPubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
Dalian University of Technology

Curated by ChEMBL
LigandPNGBDBM50336578(3-(biphenyl-4-yloxy)-8-oxo-8H-acenaphtho[1,2-b]pyr...)copy SMILEScopy InChI
Affinity DataKi:  1.28E+3nMAssay Description:Displacement of FAM-Bid peptide from human Mcl-1 after 30 mins by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6D8WPubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Dalian University of Technology

Curated by ChEMBL
LigandPNGBDBM50351806(CHEMBL1824187)copy SMILEScopy InChI
Affinity DataKi:  1.43E+3nMAssay Description:Displacement of FAM-Bid peptide from human recombinant Bcl2 after 30 mins by by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6D8WPubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Dalian University of Technology

Curated by ChEMBL
LigandPNGBDBM50351807(CHEMBL1824186)copy SMILEScopy InChI
Affinity DataKi:  6.03E+3nMAssay Description:Displacement of FAM-Bid peptide from human recombinant Bcl2 after 30 mins by by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6D8WPubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Dalian University of Technology

Curated by ChEMBL
LigandPNGBDBM50351808(CHEMBL1824189)copy SMILEScopy InChI
Affinity DataKi:  1.66E+4nMAssay Description:Displacement of FAM-Bid peptide from human recombinant Bcl2 after 30 mins by by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MK6D8WPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM23926((E)-resveratrol | 5-[(E)-2-(4-hydroxyphenyl)etheny...)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-AMC as substrate preincubated for 4 secs followed by substrate addition and measured after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ39SVPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM222244(6-Iodo-N3-(3-nitrobenzylidene)-2-phenyl-N4-(thiazo...)copy SMILEScopy InChI
Affinity DataIC50: 0.760nMAssay Description:Inhibition of DPP4 (unknown origin) using H-Gly-Pro-AMC as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ39SVPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50462429(CHEMBL4247480)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Inhibition of DPP4 (unknown origin) using H-Gly-Pro-AMC as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ39SVPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM222254(6-Iodo-N4-(4-methylthiazol-2-yl)-N3-(3-nitrobenzyl...)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMAssay Description:Inhibition of DPP4 (unknown origin) using H-Gly-Pro-AMC as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ39SVPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM222239(N3-(3-Nitrobenzylidene)-2-phenyl-N4-(thiazol-2-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Inhibition of DPP4 (unknown origin) using H-Gly-Pro-AMC as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ39SVPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM222245(6-Iodo-N3-(4-methoxybenzylidene)-2-phenyl-N4-(thia...)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:Inhibition of DPP4 (unknown origin) using H-Gly-Pro-AMC as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ39SVPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50462425(CHEMBL4241283)copy SMILEScopy InChI
Affinity DataIC50: 3.40nMAssay Description:Inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ39SVPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50462419(CHEMBL4250956)copy SMILEScopy InChI
Affinity DataIC50: 6.30nMAssay Description:Inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ39SVPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50462426(CHEMBL4241366)copy SMILEScopy InChI
Affinity DataIC50: 6.90nMAssay Description:Inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ39SVPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM11162((1R)-3-oxo-3-[3-(trifluoroethyl)-5,6-dihydro[1,2,4...)copy SMILEScopy InChI
Affinity DataIC50: 7.80nMAssay Description:Inhibition of recombinant human DPP4 using Gly-Pro-AMC as substrate after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50462415(CHEMBL4250492)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Inhibition of recombinant human DPP4 using Gly-Pro-AMC as substrate after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ39SVPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50462418(CHEMBL4246674)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant human DPP4 pre-incubated for 30 mins before Gly-Pro-Aminomethylcoumarin substrate additionMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ39SVPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM11162((1R)-3-oxo-3-[3-(trifluoroethyl)-5,6-dihydro[1,2,4...)copy SMILEScopy InChI
Affinity DataIC50: 38nMAssay Description:Inhibition of human recombinant C-terminal 6His-tagged DPP-4 expressed in insect cells incubated for 30 mins by TPE-KFPE fluorescent probe-based assa...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory of Technology of Drug Preparation (Zhengzhou University)

Curated by ChEMBL
LigandPNGBDBM50158869(CHEMBL3786182 | US10836743, Compound GSK-2879552 |...)copy SMILEScopy InChI
Affinity DataIC50: 41nMAssay Description:Inhibition of full length recombinant LSD1 (unknown origin) expressed in Escherichia coli BL21(DE) using H3K4me2 as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FQ9ZV3PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50273500(CHEMBL4128052)copy SMILEScopy InChI
Affinity DataIC50: 64nMAssay Description:Inhibition of human recombinant C-terminal 6His-tagged DPP-4 expressed in insect cells incubated for 30 mins by TPE-KFPE fluorescent probe-based assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047Z5PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50273498(CHEMBL4128601)copy SMILEScopy InChI
Affinity DataIC50: 65nMAssay Description:Inhibition of human recombinant C-terminal 6His-tagged DPP-4 expressed in insect cells incubated for 30 mins by TPE-KFPE fluorescent probe-based assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047Z5PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50462427(CHEMBL4250558)copy SMILEScopy InChI
Affinity DataIC50: 95nMAssay Description:Inhibition of recombinant human DPP4 using H-Gly-Pro-AMC as substrate after 30 mins by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ39SVPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM7459(2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4H-chromen-4...)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-AMC as substrate preincubated for 4 secs followed by substrate addition and measured after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ39SVPubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory of Technology of Drug Preparation (Zhengzhou University)

Curated by ChEMBL
LigandPNGBDBM50234620(CHEMBL4099241)copy SMILEScopy InChI
Affinity DataIC50: 121nMAssay Description:Inhibition of recombinant full length LSD1 (unknown origin) expressed in Escherichia coli BL21 (DE) using H3K4me2 substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22R3TX0PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory of Technology of Drug Preparation (Zhengzhou University)

Curated by ChEMBL
LigandPNGBDBM50234626(CHEMBL4072238)copy SMILEScopy InChI
Affinity DataIC50: 124nMAssay Description:Inhibition of recombinant full length LSD1 (unknown origin) expressed in Escherichia coli BL21 (DE) using H3K4me2 substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22R3TX0PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM7458(5,7-dihydroxy-2-(4-hydroxyphenyl)-4H-chromen-4-one...)copy SMILEScopy InChI
Affinity DataIC50: 140nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-AMC as substrate preincubated for 4 secs followed by substrate addition and measured after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ39SVPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50028962(CHEMBL275638 | flavone)copy SMILEScopy InChI
Affinity DataIC50: 170nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-AMC as substrate preincubated for 4 secs followed by substrate addition and measured after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ39SVPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50273499(CHEMBL4129968)copy SMILEScopy InChI
Affinity DataIC50: 189nMAssay Description:Inhibition of human recombinant C-terminal 6His-tagged DPP-4 expressed in insect cells incubated for 30 mins by TPE-KFPE fluorescent probe-based assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M047Z5PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory of Technology of Drug Preparation (Zhengzhou University)

Curated by ChEMBL
LigandPNGBDBM50234629(CHEMBL4089088)copy SMILEScopy InChI
Affinity DataIC50: 193nMAssay Description:Inhibition of recombinant full length LSD1 (unknown origin) expressed in Escherichia coli BL21 (DE) using H3K4me2 substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22R3TX0PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory of Technology of Drug Preparation (Zhengzhou University)

Curated by ChEMBL
LigandPNGBDBM50234625(CHEMBL4093001)copy SMILEScopy InChI
Affinity DataIC50: 197nMAssay Description:Inhibition of recombinant full length LSD1 (unknown origin) expressed in Escherichia coli BL21 (DE) using H3K4me2 substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22R3TX0PubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory of Technology of Drug Preparation (Zhengzhou University)

Curated by ChEMBL
LigandPNGBDBM50234621(CHEMBL4060903)copy SMILEScopy InChI
Affinity DataIC50: 210nMAssay Description:Inhibition of recombinant full length LSD1 (unknown origin) expressed in Escherichia coli BL21 (DE) using H3K4me2 substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22R3TX0PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50462430(CHEMBL4246222)copy SMILEScopy InChI
Affinity DataIC50: 233nMAssay Description:Inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ39SVPubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM23419((2S)-5,7-dihydroxy-2-(4-hydroxyphenyl)-3,4-dihydro...)copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-AMC as substrate preincubated for 4 secs followed by substrate addition and measured after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ39SVPubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Key Laboratory of Technology of Drug Preparation (Zhengzhou University)

Curated by ChEMBL
LigandPNGBDBM50234618(CHEMBL4091505)copy SMILEScopy InChI
Affinity DataIC50: 246nMAssay Description:Inhibition of recombinant full length LSD1 (unknown origin) expressed in Escherichia coli BL21 (DE) using H3K4me2 substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22R3TX0PubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM23418((2S)-5,7-dihydroxy-2-(3-hydroxy-4-methoxyphenyl)-3...)copy SMILEScopy InChI
Affinity DataIC50: 280nMAssay Description:Inhibition of DPP4 (unknown origin) using Gly-Pro-AMC as substrate preincubated for 4 secs followed by substrate addition and measured after 30 mins ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CZ39SVPubMed
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