Compile Data Set for Download or QSAR
Found 36 with Last Name = 'iijima' and Initial = 'y'
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Sankyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50024714(2-(4-Carboxymethyl-5-oxo-3-thiophen-2-yl-[1,4]thia...)copy SMILEScopy InChI
Affinity DataIC50: 2.80nMAssay Description:Inhibitory activity against rabbit lung Angiotensin I converting enzyme with 5 mM hippurylhistidylleucine as substrateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2Q52NMJPubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Sankyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50023299(2-(1-Carboxymethyl-2-oxo-6-phenyl-azepan-3-ylamino...)copy SMILEScopy InChI
Affinity DataIC50: 3.10nMAssay Description:Concentration required for 50% inhibition of rabbit lung Angiotensin I converting enzyme with 5 mM hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S75GWHPubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Sankyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50023298(2-(4-Carboxymethyl-5-oxo-3-phenyl-[1,4]thiazepan-6...)copy SMILEScopy InChI
Affinity DataIC50: 3.40nMAssay Description:Inhibitory activity against rabbit lung Angiotensin I converting enzyme with 5 mM hippurylhistidylleucine as substrateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2Q52NMJPubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Sankyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50023298(2-(4-Carboxymethyl-5-oxo-3-phenyl-[1,4]thiazepan-6...)copy SMILEScopy InChI
Affinity DataIC50: 3.40nMAssay Description:Concentration required for 50% inhibition of rabbit lung Angiotensin I converting enzyme with 5 mM hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S75GWHPubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Sankyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50024710(2-(4-Carboxymethyl-5-oxo-2-thiophen-2-yl-[1,4]thia...)copy SMILEScopy InChI
Affinity DataIC50: 3.60nMAssay Description:Inhibitory activity against rabbit lung Angiotensin I converting enzyme with 5 mM hippurylhistidylleucine as substrateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2Q52NMJPubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Sankyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50023296(2-(1-Carboxymethyl-2-oxo-7-phenyl-azepan-3-ylamino...)copy SMILEScopy InChI
Affinity DataIC50: 3.60nMAssay Description:Concentration required for 50% inhibition of rabbit lung Angiotensin I converting enzyme with 5 mM hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S75GWHPubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Sankyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50023295(2-(4-Carboxymethyl-5-oxo-2-phenyl-[1,4]thiazepan-6...)copy SMILEScopy InChI
Affinity DataIC50: 3.70nMAssay Description:Concentration required for 50% inhibition of rabbit lung Angiotensin I converting enzyme with 5 mM hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S75GWHPubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Sankyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50023295(2-(4-Carboxymethyl-5-oxo-2-phenyl-[1,4]thiazepan-6...)copy SMILEScopy InChI
Affinity DataIC50: 3.70nMAssay Description:Inhibitory activity against rabbit lung Angiotensin I converting enzyme with 5 mM hippurylhistidylleucine as substrateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2Q52NMJPubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Sankyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50024713(2-(4-Carboxymethyl-5-oxo-2-thiophen-3-yl-[1,4]thia...)copy SMILEScopy InChI
Affinity DataIC50: 4.10nMAssay Description:Inhibitory activity against rabbit lung Angiotensin I converting enzyme with 5 mM hippurylhistidylleucine as substrateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2Q52NMJPubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Sankyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50023300(2-(1-Carboxymethyl-2-oxo-6-phenyl-azepan-3-ylamino...)copy SMILEScopy InChI
Affinity DataIC50: 4.30nMAssay Description:Concentration required for 50% inhibition of rabbit lung Angiotensin I converting enzyme with 5 mM hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S75GWHPubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Sankyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50367254(ENALAPRILAT)copy SMILEScopy InChI
Affinity DataIC50: 5.70nMAssay Description:Concentration required for 50% inhibition of rabbit lung Angiotensin I converting enzyme with 5 mM hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S75GWHPubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Sankyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50011192((R)-1-[(S)-2-((S)-1-Carboxy-3-phenyl-propylamino)-...)copy SMILEScopy InChI
Affinity DataIC50: 5.70nMAssay Description:Inhibitory activity against rabbit lung Angiotensin I converting enzyme with 5 mM hippurylhistidylleucine as substrateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2Q52NMJPubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Sankyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50023302(2-(1-Carboxymethyl-2-oxo-7-phenyl-azepan-3-ylamino...)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Concentration required for 50% inhibition of rabbit lung Angiotensin I converting enzyme with 5 mM hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S75GWHPubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Sankyo Co. Ltd

Curated by ChEMBL
LigandPNGBDBM50366241(CHEMBL297624 | L-652731)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3T06PubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Sankyo Co. Ltd

Curated by ChEMBL
LigandPNGBDBM50055488(CHEMBL148491 | Carbonic acid methyl ester (E)-(1R,...)copy SMILEScopy InChI
Affinity DataIC50: 26nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3T06PubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Sankyo Co. Ltd

Curated by ChEMBL
LigandPNGBDBM50055491((E)-(1R,2R,3R,5R,12S,13R,16S)-16-(Isoxazol-3-yloxy...)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3T06PubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Sankyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50023303(2-(4-Carboxymethyl-5-oxo-2-phenyl-[1,4]thiazepan-6...)copy SMILEScopy InChI
Affinity DataIC50: 36nMAssay Description:Inhibitory activity against rabbit lung Angiotensin I converting enzyme with 5 mM hippurylhistidylleucine as substrateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2Q52NMJPubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Sankyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50023303(2-(4-Carboxymethyl-5-oxo-2-phenyl-[1,4]thiazepan-6...)copy SMILEScopy InChI
Affinity DataIC50: 36nMAssay Description:Concentration required for 50% inhibition of rabbit lung Angiotensin I converting enzyme with 5 mM hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S75GWHPubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Sankyo Co. Ltd

Curated by ChEMBL
LigandPNGBDBM50055482((E)-(1R,3S,5R,12S,13R,16S)-16-(Isoxazol-3-yloxymet...)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3T06PubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Sankyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50024712(2-(4-Carboxymethyl-5-oxo-2-thiophen-2-yl-[1,4]thia...)copy SMILEScopy InChI
Affinity DataIC50: 65nMAssay Description:Inhibitory activity against rabbit lung Angiotensin I converting enzyme with 5 mM hippurylhistidylleucine as substrateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2Q52NMJPubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Sankyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50023301(2-(4-Carboxymethyl-5-oxo-3-phenyl-[1,4]thiazepan-6...)copy SMILEScopy InChI
Affinity DataIC50: 78nMAssay Description:Concentration required for 50% inhibition of rabbit lung Angiotensin I converting enzyme with 5 mM hippuryl-histidyl-leucine as substrateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2S75GWHPubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Sankyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50023301(2-(4-Carboxymethyl-5-oxo-3-phenyl-[1,4]thiazepan-6...)copy SMILEScopy InChI
Affinity DataIC50: 78nMAssay Description:Inhibitory activity against rabbit lung Angiotensin I converting enzyme with 5 mM hippurylhistidylleucine as substrateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2Q52NMJPubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Sankyo Co. Ltd

Curated by ChEMBL
LigandPNGBDBM50055479(Acetic acid (E)-(1R,2R,3R,5R,12S,13R,16S)-2-hydrox...)copy SMILEScopy InChI
Affinity DataIC50: 80nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3T06PubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Sankyo Co., Ltd.

Curated by ChEMBL
LigandPNGBDBM50024711(2-(4-Carboxymethyl-5-oxo-2-thiophen-3-yl-[1,4]thia...)copy SMILEScopy InChI
Affinity DataIC50: 87nMAssay Description:Inhibitory activity against rabbit lung Angiotensin I converting enzyme with 5 mM hippurylhistidylleucine as substrateMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2Q52NMJPubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Sankyo Co. Ltd

Curated by ChEMBL
LigandPNGBDBM50055489((E)-(1R,3S,5R,12S,13R,16S)-5,9,12,13-Tetramethyl-2...)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3T06PubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Sankyo Co. Ltd

Curated by ChEMBL
LigandPNGBDBM50055493(CHEMBL148549 | Carbonic acid (E)-(1R,2R,3R,5R,12S,...)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3T06PubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Sankyo Co. Ltd

Curated by ChEMBL
LigandPNGBDBM50055495(CHEMBL151075 | Dimethyl-carbamic acid (E)-(1R,2R,3...)copy SMILEScopy InChI
Affinity DataIC50: 180nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3T06PubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Sankyo Co. Ltd

Curated by ChEMBL
LigandPNGBDBM50055483(CHEMBL151310 | Dimethyl-carbamic acid (E)-(1R,3S,5...)copy SMILEScopy InChI
Affinity DataIC50: 180nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3T06PubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Sankyo Co. Ltd

Curated by ChEMBL
LigandPNGBDBM50055492(CHEMBL147337 | Propionic acid (E)-(1R,2R,3R,5R,12S...)copy SMILEScopy InChI
Affinity DataIC50: 340nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3T06PubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Sankyo Co. Ltd

Curated by ChEMBL
LigandPNGBDBM50055487(Acetic acid (E)-(1R,3S,5R,12S,13R,16S)-5,9,12,13-t...)copy SMILEScopy InChI
Affinity DataIC50: 410nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3T06PubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Sankyo Co. Ltd

Curated by ChEMBL
LigandPNGBDBM50055484(CHEMBL421954 | Carbonic acid phenyl ester (E)-(1R,...)copy SMILEScopy InChI
Affinity DataIC50: 550nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3T06PubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Sankyo Co. Ltd

Curated by ChEMBL
LigandPNGBDBM50055494(CHEMBL147079 | Propionic acid (E)-(1R,3S,5R,12S,13...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3T06PubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Sankyo Co. Ltd

Curated by ChEMBL
LigandPNGBDBM50055480((E)-(1R,3S,5R,12S,13R,16S)-16-Hydroxymethyl-5,9,12...)copy SMILEScopy InChI
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3T06PubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Sankyo Co. Ltd

Curated by ChEMBL
LigandPNGBDBM50055485(16-(Isoxazol-3-yloxymethyl)-5,9,12,13-tetramethyl-...)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3T06PubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Sankyo Co. Ltd

Curated by ChEMBL
LigandPNGBDBM50055481(16-(Isoxazol-3-yloxymethyl)-5,9,12,13-tetramethyl-...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3T06PubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Sankyo Co. Ltd

Curated by ChEMBL
LigandPNGBDBM50055486((1R,3S,5R,8S,9S,12S,13R,16S)-8,9-Dihydroxy-16-hydr...)copy SMILEScopy InChI
Affinity DataIC50: 2.80E+5nMAssay Description:Inhibiting Platelet activating factor receptor by radioreceptor binding assay using rabbit platelets and [3H]-PAFMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FF3T06PubMed