Compile Data Set for Download or QSAR
Found 14 with Last Name = 'kubota' and Initial = 'y'
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Institute of Microbial Chemistry (BIKAKEN)

Curated by ChEMBL
LigandPNGBDBM50428367(CHEMBL2332119 | Vegfrecine)copy SMILEScopy InChI
Affinity DataIC50: 1.80nMAssay Description:Inhibition of Flt4 (unknown origin) after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ12BHPubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Institute of Microbial Chemistry (BIKAKEN)

Curated by ChEMBL
LigandPNGBDBM50428367(CHEMBL2332119 | Vegfrecine)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of KDR (unknown origin) after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ12BHPubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Institute of Microbial Chemistry (BIKAKEN)

Curated by ChEMBL
LigandPNGBDBM50428367(CHEMBL2332119 | Vegfrecine)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:Inhibition of GST-Flt1 kinase domain (unknown origin) expressed in baculovirus infected Sf9 cells after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ12BHPubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Institute of Microbial Chemistry (BIKAKEN)

Curated by ChEMBL
LigandPNGBDBM4810((3Z)-3-[(3,5-dimethyl-1H-pyrrol-2-yl)methylidene]-...)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Inhibition of PDGFR-alpha (unknown origin) after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ12BHPubMed
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Institute of Microbial Chemistry (BIKAKEN)

Curated by ChEMBL
LigandPNGBDBM4810((3Z)-3-[(3,5-dimethyl-1H-pyrrol-2-yl)methylidene]-...)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Inhibition of PDGFR-beta (unknown origin) after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ12BHPubMed
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Institute of Microbial Chemistry (BIKAKEN)

Curated by ChEMBL
LigandPNGBDBM50428367(CHEMBL2332119 | Vegfrecine)copy SMILEScopy InChI
Affinity DataIC50: 480nMAssay Description:Inhibition of PDGFR-beta (unknown origin) after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ12BHPubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Institute of Microbial Chemistry (BIKAKEN)

Curated by ChEMBL
LigandPNGBDBM4810((3Z)-3-[(3,5-dimethyl-1H-pyrrol-2-yl)methylidene]-...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibition of Flt4 (unknown origin) after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ12BHPubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Institute of Microbial Chemistry (BIKAKEN)

Curated by ChEMBL
LigandPNGBDBM4810((3Z)-3-[(3,5-dimethyl-1H-pyrrol-2-yl)methylidene]-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of KDR (unknown origin) after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ12BHPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Institute of Microbial Chemistry (BIKAKEN)

Curated by ChEMBL
LigandPNGBDBM50428367(CHEMBL2332119 | Vegfrecine)copy SMILEScopy InChI
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of EGFR (unknown origin) after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ12BHPubMed
TargetVascular endothelial growth factor receptor 1(Homo sapiens (Human))
Institute of Microbial Chemistry (BIKAKEN)

Curated by ChEMBL
LigandPNGBDBM4810((3Z)-3-[(3,5-dimethyl-1H-pyrrol-2-yl)methylidene]-...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of GST-Flt1 kinase domain (unknown origin) expressed in baculovirus infected Sf9 cells after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ12BHPubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
Institute of Microbial Chemistry (BIKAKEN)

Curated by ChEMBL
LigandPNGBDBM50428367(CHEMBL2332119 | Vegfrecine)copy SMILEScopy InChI
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of PDGFR-alpha (unknown origin) after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ12BHPubMed
TargetCellular tumor antigen p53(Homo sapiens (Human))
Institute of Microbial Chemistry (BIKAKEN)

Curated by ChEMBL
LigandPNGBDBM50080457(CHEMBL3422268)copy SMILEScopy InChI
Affinity DataIC50: 6.20E+3nMAssay Description:Induction of p53-dependent growth suppression of human LNZTA3 cells after 72 hrs by MTT assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B046ZPubMed
TargetCellular tumor antigen p53(Homo sapiens (Human))
Institute of Microbial Chemistry (BIKAKEN)

Curated by ChEMBL
LigandPNGBDBM50080451(CHEMBL3422267)copy SMILEScopy InChI
Affinity DataIC50: 6.20E+3nMAssay Description:Induction of p53-dependent growth suppression of human LNZTA3 cells after 72 hrs by MTT assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B046ZPubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Institute of Microbial Chemistry (BIKAKEN)

Curated by ChEMBL
LigandPNGBDBM4810((3Z)-3-[(3,5-dimethyl-1H-pyrrol-2-yl)methylidene]-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of EGFR (unknown origin) after 20 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JQ12BHPubMed