Compile Data Set for Download or QSAR
Found 152 with Last Name = 'nagano' and Initial = 'y'
TargetProtein kinase C zeta type(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542127(CHEMBL4635482)copy SMILEScopy InChI
Affinity DataIC50: 0.100nMAssay Description:Inhibition of recombinant human PKCzeta using biotin-KKKKRFSFKKSFK substrate and ATP incubated for 30 mins by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542123(CHEMBL4636488)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:Inhibition of recombinant human PKCzeta using biotin-KKKKRFSFKKSFK substrate and ATP incubated for 30 mins by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542116(CHEMBL4646995)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Inhibition of recombinant human PKCzeta using biotin-KKKKRFSFKKSFK substrate and ATP incubated for 30 mins by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542119(CHEMBL4644939)copy SMILEScopy InChI
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant human PKCzeta using biotin-KKKKRFSFKKSFK substrate and ATP incubated for 30 mins by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542128(CHEMBL4636337)copy SMILEScopy InChI
Affinity DataIC50: 0.800nMAssay Description:Inhibition of recombinant human PKCzeta using biotin-KKKKRFSFKKSFK substrate and ATP incubated for 30 mins by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542132(CHEMBL4632523)copy SMILEScopy InChI
Affinity DataIC50: 0.900nMAssay Description:Inhibition of recombinant human PKCzeta using biotin-KKKKRFSFKKSFK substrate and ATP incubated for 30 mins by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542133(CHEMBL4643553)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Inhibition of recombinant human PKCzeta using biotin-KKKKRFSFKKSFK substrate and ATP incubated for 30 mins by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542126(CHEMBL4642166)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:Inhibition of recombinant human PKCzeta using biotin-KKKKRFSFKKSFK substrate and ATP incubated for 30 mins by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542129(CHEMBL4637452)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:Inhibition of recombinant human PKCzeta using biotin-KKKKRFSFKKSFK substrate and ATP incubated for 30 mins by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542134(CHEMBL4647780)copy SMILEScopy InChI
Affinity DataIC50: 3.40nMAssay Description:Inhibition of recombinant human PKCzeta using biotin-KKKKRFSFKKSFK substrate and ATP incubated for 30 mins by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542125(CHEMBL4643470)copy SMILEScopy InChI
Affinity DataIC50: 4.10nMAssay Description:Inhibition of recombinant human PKCzeta using biotin-KKKKRFSFKKSFK substrate and ATP incubated for 30 mins by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542121(CHEMBL4641918)copy SMILEScopy InChI
Affinity DataIC50: 6.40nMAssay Description:Inhibition of recombinant human PKCzeta using biotin-KKKKRFSFKKSFK substrate and ATP incubated for 30 mins by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542130(CHEMBL4632384)copy SMILEScopy InChI
Affinity DataIC50: 9.70nMAssay Description:Inhibition of recombinant human PKCzeta using biotin-KKKKRFSFKKSFK substrate and ATP incubated for 30 mins by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542122(CHEMBL4642061)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant human PKCzeta using biotin-KKKKRFSFKKSFK substrate and ATP incubated for 30 mins by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542111(CHEMBL4644763)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant human PKCzeta using biotin-KKKKRFSFKKSFK substrate and ATP incubated for 30 mins by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542131(CHEMBL4634517)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of recombinant human PKCzeta using biotin-KKKKRFSFKKSFK substrate and ATP incubated for 30 mins by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetSerine/threonine-protein kinase D2(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542119(CHEMBL4644939)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Inhibition of PKD2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542100(CHEMBL4645728)copy SMILEScopy InChI
Affinity DataIC50: 33nMAssay Description:Inhibition of recombinant human PKCzeta using biotin-KKKKRFSFKKSFK substrate and ATP incubated for 30 mins by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542124(CHEMBL4641607)copy SMILEScopy InChI
Affinity DataIC50: 35nMAssay Description:Inhibition of recombinant human PKCzeta using biotin-KKKKRFSFKKSFK substrate and ATP incubated for 30 mins by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542127(CHEMBL4635482)copy SMILEScopy InChI
Affinity DataIC50: 45nMAssay Description:Inhibition of PKCzeta in human THP1 cells assessed as reduction in LPS-induced TNFalpha production pre-incubated for 60 mins before LPS simulations f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542120(CHEMBL4648006)copy SMILEScopy InChI
Affinity DataIC50: 54nMAssay Description:Inhibition of recombinant human PKCzeta using biotin-KKKKRFSFKKSFK substrate and ATP incubated for 30 mins by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetHistone deacetylase(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50475239(CHEMBL112234)copy SMILEScopy InChI
Affinity DataIC50: 72nMAssay Description:Inhibitory concentration against human histone deacetylaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3P70PubMed
TargetHistone deacetylase(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50475246(CHEMBL320323)copy SMILEScopy InChI
Affinity DataIC50: 75nMAssay Description:Inhibitory concentration against human histone deacetylaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3P70PubMed
TargetHistone deacetylase(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50475237(CHEMBL112105)copy SMILEScopy InChI
Affinity DataIC50: 79nMAssay Description:Inhibitory concentration against human histone deacetylaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3P70PubMed
TargetHistone deacetylase(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50475250(CHEMBL113421)copy SMILEScopy InChI
Affinity DataIC50: 85nMAssay Description:Inhibitory concentration against human histone deacetylaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3P70PubMed
TargetHistone deacetylase(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50475236(CHEMBL113159)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibitory concentration against human histone deacetylaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3P70PubMed
TargetSerine/threonine-protein kinase D2(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542117(CHEMBL4640042)copy SMILEScopy InChI
Affinity DataIC50: 102nMAssay Description:Inhibition of PKD2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542114(CHEMBL4646074)copy SMILEScopy InChI
Affinity DataIC50: 109nMAssay Description:Inhibition of recombinant human PKCzeta using biotin-KKKKRFSFKKSFK substrate and ATP incubated for 30 mins by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetHistone deacetylase(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50223653(CHEMBL332246)copy SMILEScopy InChI
Affinity DataIC50: 110nMAssay Description:Inhibitory concentration against human histone deacetylaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3P70PubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542103(CHEMBL4639268)copy SMILEScopy InChI
Affinity DataIC50: 141nMAssay Description:Inhibition of recombinant human PKCzeta using biotin-KKKKRFSFKKSFK substrate and ATP incubated for 30 mins by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542101(CHEMBL4641149)copy SMILEScopy InChI
Affinity DataIC50: 142nMAssay Description:Inhibition of recombinant human PKCzeta using biotin-KKKKRFSFKKSFK substrate and ATP incubated for 30 mins by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetSerine/threonine-protein kinase D2(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542123(CHEMBL4636488)copy SMILEScopy InChI
Affinity DataIC50: 144nMAssay Description:Inhibition of PKD2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542102(CHEMBL4633764)copy SMILEScopy InChI
Affinity DataIC50: 147nMAssay Description:Inhibition of recombinant human PKCzeta using biotin-KKKKRFSFKKSFK substrate and ATP incubated for 30 mins by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542118(CHEMBL4645229)copy SMILEScopy InChI
Affinity DataIC50: 153nMAssay Description:Inhibition of recombinant human PKCzeta using biotin-KKKKRFSFKKSFK substrate and ATP incubated for 30 mins by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542117(CHEMBL4640042)copy SMILEScopy InChI
Affinity DataIC50: 162nMAssay Description:Inhibition of recombinant human PKCzeta using biotin-KKKKRFSFKKSFK substrate and ATP incubated for 30 mins by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetHistone deacetylase(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM19131(CHEMBL419758 | JMC505425 Compound 7 | N-(4-phenyl-...)copy SMILEScopy InChI
Affinity DataIC50: 170nMAssay Description:Inhibitory concentration against human histone deacetylaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3P70PubMed
TargetSerine/threonine-protein kinase D2(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542118(CHEMBL4645229)copy SMILEScopy InChI
Affinity DataIC50: 187nMAssay Description:Inhibition of PKD2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetSerine/threonine-protein kinase D2(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542125(CHEMBL4643470)copy SMILEScopy InChI
Affinity DataIC50: 202nMAssay Description:Inhibition of PKD2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetHistone deacetylase(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM152692(Thiol-SAHA (t-SAHA))copy SMILEScopy InChI
Affinity DataIC50: 210nMAssay Description:Inhibitory concentration against human histone deacetylaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3P70PubMed
TargetHistone deacetylase(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50223648(CHEMBL322504)copy SMILEScopy InChI
Affinity DataIC50: 210nMAssay Description:Inhibitory concentration against human histone deacetylaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3P70PubMed
TargetSerine/threonine-protein kinase D2(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542116(CHEMBL4646995)copy SMILEScopy InChI
Affinity DataIC50: 246nMAssay Description:Inhibition of PKD2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetSerine/threonine-protein kinase D2(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542121(CHEMBL4641918)copy SMILEScopy InChI
Affinity DataIC50: 261nMAssay Description:Inhibition of PKD2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetSerine/threonine-protein kinase D2(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542120(CHEMBL4648006)copy SMILEScopy InChI
Affinity DataIC50: 263nMAssay Description:Inhibition of PKD2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetHistone deacetylase(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)copy SMILEScopy InChI
Affinity DataIC50: 280nMAssay Description:Inhibitory concentration against human histone deacetylaseMore data for this Ligand-Target Pair
TargetHistone deacetylase(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)copy SMILEScopy InChI
Affinity DataIC50: 280nMAssay Description:In vitro inhibitory activity against histone deacetylase (HDAC) isolated from HeLa nuclear extractMore data for this Ligand-Target Pair
TargetProtein kinase C zeta type(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542112(CHEMBL4638383)copy SMILEScopy InChI
Affinity DataIC50: 321nMAssay Description:Inhibition of recombinant human PKCzeta using biotin-KKKKRFSFKKSFK substrate and ATP incubated for 30 mins by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetHistone deacetylase(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50475243(CHEMBL178779)copy SMILEScopy InChI
Affinity DataIC50: 340nMAssay Description:Inhibitory concentration against human histone deacetylaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3P70PubMed
TargetHistone deacetylase(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50221784(CHEMBL112211)copy SMILEScopy InChI
Affinity DataIC50: 340nMAssay Description:Inhibitory concentration against human histone deacetylaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3P70PubMed
TargetProtein kinase C zeta type(Homo sapiens (Human))
Asahi Kasei Pharma Corporation

Curated by ChEMBL
LigandPNGBDBM50542108(CHEMBL4641174)copy SMILEScopy InChI
Affinity DataIC50: 356nMAssay Description:Inhibition of recombinant human PKCzeta using biotin-KKKKRFSFKKSFK substrate and ATP incubated for 30 mins by TR-FRET methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6NWXPubMed
TargetHistone deacetylase(Homo sapiens (Human))
Nagoya City University

Curated by ChEMBL
LigandPNGBDBM50223650(CHEMBL112364)copy SMILEScopy InChI
Affinity DataIC50: 360nMAssay Description:Inhibitory concentration against human histone deacetylaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3P70PubMed
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