Compile Data Set for Download or QSAR
Found 28 with Last Name = 'zhang' and Initial = 'yf'
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50387918(CHEMBL2058680 | US9283222, 459)copy SMILEScopy InChI
In DepthDetails
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556717(CHEMBL4780703)copy SMILES
Affinity DataIC50: 630nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P9327PubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556698(CHEMBL2375494)copy SMILES
Affinity DataIC50: 650nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P9327PubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556715(CHEMBL4782344)copy SMILES
Affinity DataIC50: 880nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P9327PubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556716(CHEMBL4796964)copy SMILES
Affinity DataIC50: 910nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P9327PubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556721(CHEMBL4790746)copy SMILES
Affinity DataIC50: 1.01E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P9327PubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556719(CHEMBL4782590)copy SMILES
Affinity DataIC50: 1.08E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P9327PubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556710(CHEMBL4741257)copy SMILES
Affinity DataIC50: 1.23E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P9327PubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556706(CHEMBL4797370)copy SMILES
Affinity DataIC50: 1.49E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P9327PubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556718(CHEMBL4787771)copy SMILES
Affinity DataIC50: 1.52E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P9327PubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556699(CHEMBL4746541)copy SMILES
Affinity DataIC50: 1.64E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P9327PubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556705(CHEMBL4793323)copy SMILES
Affinity DataIC50: 1.72E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P9327PubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556708(CHEMBL4795327)copy SMILES
Affinity DataIC50: 1.76E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P9327PubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556722(CHEMBL4791780)copy SMILES
Affinity DataIC50: 1.81E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P9327PubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556700(CHEMBL4761208)copy SMILES
Affinity DataIC50: 1.81E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P9327PubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556720(CHEMBL4745132)copy SMILES
Affinity DataIC50: 1.82E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P9327PubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556709(CHEMBL4783011)copy SMILES
Affinity DataIC50: 2.37E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P9327PubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556703(CHEMBL4761078)copy SMILES
Affinity DataIC50: 2.57E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P9327PubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556701(CHEMBL4746014)copy SMILES
Affinity DataIC50: 2.63E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P9327PubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556702(CHEMBL4763588)copy SMILES
Affinity DataIC50: 2.82E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P9327PubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556704(CHEMBL4740701)copy SMILES
Affinity DataIC50: 3.02E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P9327PubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556713(CHEMBL4748854)copy SMILES
Affinity DataIC50: 3.29E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P9327PubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556714(CHEMBL4777734)copy SMILES
Affinity DataIC50: 3.54E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P9327PubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556707(CHEMBL4762863)copy SMILES
Affinity DataIC50: 3.87E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P9327PubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556723(CHEMBL240484)copy SMILES
Affinity DataIC50: 5.45E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P9327PubMed
LigandPNGBDBM50353952(CHEMBL1831185)copy SMILEScopy InChI
Affinity DataIC50: 5.60E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556712(CHEMBL4798117)copy SMILES
Affinity DataIC50: 7.64E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P9327PubMed
TargetG-protein coupled receptor 52(Homo sapiens (Human))TBA
LigandPNGBDBM50556711(CHEMBL4755423)copy SMILES
Affinity DataIC50: 8.13E+3nMAssay Description:Antagonist activity at GPR52 (unknown origin) expressed in HEK293 cells assessed as inhibition of WO459-induced cAMP accumulation preincubated for 15...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P9327PubMed