TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez (CIBICAN)
Curated by ChEMBL
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez (CIBICAN)
Curated by ChEMBL
Affinity DataKi: 390nMAssay Description:ATP-competitive inhibition of human CK2-alpha/beta expressed in Escherichia coli BL21(DE3) using RRRDDDSDDD peptide as substrate after 15 mins in pre...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez (CIBICAN)
Curated by ChEMBL
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez (CIBICAN)
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:Inhibition of human CK2-alpha/beta expressed in Escherichia coli BL21(DE3) using RRRDDDSDDD peptide as substrate after 15 mins by capillary electroph...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez (CIBICAN)
Curated by ChEMBL
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez (CIBICAN)
Curated by ChEMBL
Affinity DataIC50: 570nMAssay Description:Inhibition of human CK2-alpha/beta expressed in Escherichia coli BL21(DE3) using RRRDDDSDDD peptide as substrate after 15 mins by capillary electroph...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez (CIBICAN)
Curated by ChEMBL
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez (CIBICAN)
Curated by ChEMBL
Affinity DataIC50: 580nMAssay Description:Inhibition of human CK2-alpha/beta expressed in Escherichia coli BL21(DE3) using RRRDDDSDDD peptide as substrate after 15 mins by capillary electroph...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez (CIBICAN)
Curated by ChEMBL
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez (CIBICAN)
Curated by ChEMBL
Affinity DataIC50: 720nMAssay Description:Inhibition of human CK2-alpha/beta expressed in Escherichia coli BL21(DE3) using RRRDDDSDDD peptide as substrate after 15 mins by capillary electroph...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez (CIBICAN)
Curated by ChEMBL
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez (CIBICAN)
Curated by ChEMBL
Affinity DataIC50: 840nMAssay Description:Inhibition of human CK2-alpha/beta expressed in Escherichia coli BL21(DE3) using RRRDDDSDDD peptide as substrate after 15 mins by capillary electroph...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez (CIBICAN)
Curated by ChEMBL
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez (CIBICAN)
Curated by ChEMBL
Affinity DataIC50: 890nMAssay Description:Inhibition of human CK2-alpha/beta expressed in Escherichia coli BL21(DE3) using RRRDDDSDDD peptide as substrate after 15 mins by capillary electroph...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez (CIBICAN)
Curated by ChEMBL
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez (CIBICAN)
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Inhibition of human CK2-alpha/beta expressed in Escherichia coli BL21(DE3) using RRRDDDSDDD peptide as substrate after 15 mins by capillary electroph...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez (CIBICAN)
Curated by ChEMBL
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez (CIBICAN)
Curated by ChEMBL
Affinity DataIC50: 996nMAssay Description:Inhibition of human CK2-alpha/beta expressed in Escherichia coli BL21(DE3) using RRRDDDSDDD peptide as substrate after 15 mins by capillary electroph...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha 3(Homo sapiens)
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez (CIBICAN)
Curated by ChEMBL
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez (CIBICAN)
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of CK2 (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez (CIBICAN)
Curated by ChEMBL
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez (CIBICAN)
Curated by ChEMBL
Affinity DataIC50: 1.36E+3nMAssay Description:Inhibition of human CK2-alpha/beta expressed in Escherichia coli BL21(DE3) using RRRDDDSDDD peptide as substrate after 15 mins by capillary electroph...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez (CIBICAN)
Curated by ChEMBL
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez (CIBICAN)
Curated by ChEMBL
Affinity DataIC50: 1.38E+3nMAssay Description:Inhibition of human CK2-alpha/beta expressed in Escherichia coli BL21(DE3) using RRRDDDSDDD peptide as substrate after 15 mins by capillary electroph...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez (CIBICAN)
Curated by ChEMBL
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez (CIBICAN)
Curated by ChEMBL
Affinity DataIC50: 1.44E+3nMAssay Description:Inhibition of human CK2-alpha/beta expressed in Escherichia coli BL21(DE3) using RRRDDDSDDD peptide as substrate after 15 mins by capillary electroph...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez (CIBICAN)
Curated by ChEMBL
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez (CIBICAN)
Curated by ChEMBL
Affinity DataIC50: 1.94E+3nMAssay Description:Inhibition of human CK2-alpha/beta expressed in Escherichia coli BL21(DE3) using RRRDDDSDDD peptide as substrate after 15 mins by capillary electroph...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez (CIBICAN)
Curated by ChEMBL
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez (CIBICAN)
Curated by ChEMBL
Affinity DataIC50: 1.99E+3nMAssay Description:Inhibition of human CK2-alpha/beta expressed in Escherichia coli BL21(DE3) using RRRDDDSDDD peptide as substrate after 15 mins by capillary electroph...More data for this Ligand-Target Pair
TargetCasein kinase II subunit alpha/beta(Homo sapiens (Human))
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez (CIBICAN)
Curated by ChEMBL
Instituto Universitario de Bio-Org£nica Antonio Gonz£lez (CIBICAN)
Curated by ChEMBL
Affinity DataIC50: 3.71E+3nMAssay Description:Inhibition of human CK2-alpha/beta expressed in Escherichia coli BL21(DE3) using RRRDDDSDDD peptide as substrate after 15 mins by capillary electroph...More data for this Ligand-Target Pair
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Instituto Universitario de Bio-Org£nica (CIBICAN)
Curated by ChEMBL
Instituto Universitario de Bio-Org£nica (CIBICAN)
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human topoisomerase-2 alpha expressed in baculovirus infected insect cells assessed as reduction in enzyme-meditaed supercoiled pRYG DN...More data for this Ligand-Target Pair
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Instituto Universitario de Bio-Org£nica (CIBICAN)
Curated by ChEMBL
Instituto Universitario de Bio-Org£nica (CIBICAN)
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human topoisomerase-2 alpha expressed in baculovirus infected insect cells assessed as reduction in enzyme-meditaed supercoiled pRYG DN...More data for this Ligand-Target Pair
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Instituto Universitario de Bio-Org£nica (CIBICAN)
Curated by ChEMBL
Instituto Universitario de Bio-Org£nica (CIBICAN)
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human topoisomerase-2 alpha expressed in baculovirus infected insect cells assessed as reduction in enzyme-meditaed supercoiled pRYG DN...More data for this Ligand-Target Pair
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Instituto Universitario de Bio-Org£nica (CIBICAN)
Curated by ChEMBL
Instituto Universitario de Bio-Org£nica (CIBICAN)
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human topoisomerase-2 alpha expressed in baculovirus infected insect cells assessed as reduction in enzyme-meditaed supercoiled pRYG DN...More data for this Ligand-Target Pair
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Instituto Universitario de Bio-Org£nica (CIBICAN)
Curated by ChEMBL
Instituto Universitario de Bio-Org£nica (CIBICAN)
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human topoisomerase-2 alpha expressed in baculovirus infected insect cells assessed as reduction in enzyme-meditaed supercoiled pRYG DN...More data for this Ligand-Target Pair
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Instituto Universitario de Bio-Org£nica (CIBICAN)
Curated by ChEMBL
Instituto Universitario de Bio-Org£nica (CIBICAN)
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human topoisomerase-2 alpha expressed in baculovirus infected insect cells assessed as reduction in enzyme-meditaed supercoiled pRYG DN...More data for this Ligand-Target Pair
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Instituto Universitario de Bio-Org£nica (CIBICAN)
Curated by ChEMBL
Instituto Universitario de Bio-Org£nica (CIBICAN)
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human topoisomerase-2 alpha expressed in baculovirus infected insect cells assessed as reduction in enzyme-meditaed supercoiled pRYG DN...More data for this Ligand-Target Pair
Affinity DataIC50: 1.38E+4nMAssay Description:Inhibition of NLRP3 in mouse J774A.1 cells assessed as inhibition of LPS and nigerecin-induced IL-1beta production pre-stimulated with LPS for 5 hrs ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.87E+4nMAssay Description:Inhibition of NLRP3 in mouse J774A.1 cells assessed as inhibition of LPS and nigerecin-induced IL-1beta production pre-stimulated with LPS for 5 hrs ...More data for this Ligand-Target Pair
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