Affinity DataKi: 5nMAssay Description:Binding affinity against Purine nucleoside Phosphorylase from calf spleenMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 8.70nMAssay Description:Inhibition of Purine nucleoside Phosphorylase from calf spleen at 1 mM PO4More data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 8.70nMAssay Description:Binding affinity against hydrophobic pocket of Purine nucleoside PhosphorylaseMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 8.70nMAssay Description:Inhibition of Purine nucleoside Phosphorylase from calf spleen at 1 mM PO4More data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Bos taurus (bovine))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Inhibition of purine nucleoside phosphorylase against the enzyme from calf spleen in 1 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Bos taurus (bovine))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from calf spleen in 1 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Bos taurus (bovine))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 45nMAssay Description:Inhibition of purine nucleoside phosphorylase against the enzyme from calf spleen in 1 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Bos taurus (bovine))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 90nMAssay Description:Inhibition of purine nucleoside phosphorylase against the enzyme from calf spleen in 1 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Bos taurus (bovine))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from calf spleen in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 170nMAssay Description:Inhibition of human erythrocytic PNP (purine nucleoside phosphorylase) in 1 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 210nMAssay Description:Inhibition of human erythrocytic PNP (purine nucleoside phosphorylase) in 1 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMAssay Description:Inhibition of human erythrocytic PNP (purine nucleoside phosphorylase) in 1 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Bos taurus (bovine))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from calf spleen in 1 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataKi: 1.10E+5nMAssay Description:Inhibition of human erythrocytic PNP (purine nucleoside phosphorylase) in 1 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 0.0300nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 0.0570nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 0.0670nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Bos taurus (bovine))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 0.0670nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from calf spleen in 1 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 0.0850nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 0.0850nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 0.160nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Bos taurus (bovine))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 0.160nMAssay Description:Inhibition of purine nucleoside phosphorylase against the enzyme from calf spleen in 1 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Bos taurus (bovine))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 0.160nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from calf spleen in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 0.25nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 0.470nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Bos taurus (bovine))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 0.630nMAssay Description:Inhibition of purine nucleoside phosphorylase against the enzyme from calf spleen in 1 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 0.630nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 0.75nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 0.850nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 4.10nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 4.10nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMpH: 6.8 T: 2°CAssay Description:The C-terminal his-tagged AdoMetDC was assayed by measuring the release of 14CO2 from S-adenosyl-L-[carboxy-14C]methionine (Amersham Pharmacia Biotec...More data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 5.90nMAssay Description:Inhibition of Purine nucleoside Phosphorylase from calf spleen at 1 mM PO4More data for this Ligand-Target Pair
Affinity DataIC50: 7nMpH: 6.8 T: 2°CAssay Description:The C-terminal his-tagged AdoMetDC was assayed by measuring the release of 14CO2 from S-adenosyl-L-[carboxy-14C]methionine (Amersham Pharmacia Biotec...More data for this Ligand-Target Pair
Affinity DataIC50: 11nMpH: 6.8 T: 2°CAssay Description:The C-terminal his-tagged AdoMetDC was assayed by measuring the release of 14CO2 from S-adenosyl-L-[carboxy-14C]methionine (Amersham Pharmacia Biotec...More data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Bos taurus (bovine))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:In vitro inhibition of purine nucleoside phosphorylase from calf spleen in 1 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of Purine nucleoside Phosphorylase from calf spleen at 1 mM PO4More data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Bos taurus (bovine))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of purine nucleoside phosphorylase against the enzyme from calf spleen in 1 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of Purine nucleoside Phosphorylase from calf spleen at 1 mM PO4More data for this Ligand-Target Pair
Affinity DataIC50: 15nMpH: 6.8 T: 2°CAssay Description:The C-terminal his-tagged AdoMetDC was assayed by measuring the release of 14CO2 from S-adenosyl-L-[carboxy-14C]methionine (Amersham Pharmacia Biotec...More data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Bos taurus (bovine))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of purine nucleoside phosphorylase against the enzyme from calf spleen in 1 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Bos taurus (bovine))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:In vitro inhibition of purine nucleoside phosphorylase from calf spleen in 1 mM phosphateMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMpH: 6.8 T: 2°CAssay Description:The C-terminal his-tagged AdoMetDC was assayed by measuring the release of 14CO2 from S-adenosyl-L-[carboxy-14C]methionine (Amersham Pharmacia Biotec...More data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from Human erythrocytic in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Homo sapiens (Human))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of Purine nucleoside Phosphorylase from calf spleen at 1 mM PO4More data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Bos taurus (bovine))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of Purine nucleoside phosphorylase was evaluated against the enzyme from calf spleen in 50 mM phosphateMore data for this Ligand-Target Pair
TargetPurine nucleoside phosphorylase(Bos taurus (bovine))
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
BioCryst Pharmaceuticals, Inc.
Curated by ChEMBL
Affinity DataIC50: 21nMAssay Description:Inhibition of purine nucleoside phosphorylase against the enzyme from calf spleen in 1 mM phosphateMore data for this Ligand-Target Pair