Compile Data Set for Download or QSAR
Found 177 with Last Name = 'karoli' and Initial = 't'
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals Limited

Curated by ChEMBL
LigandPNGBDBM50388329(CHEMBL2059500)copy SMILEScopy InChI
Affinity DataKi:  3.70nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G161WNPubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals Limited

Curated by ChEMBL
LigandPNGBDBM50388343(CHEMBL2059243)copy SMILEScopy InChI
Affinity DataKi:  5.5nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G161WNPubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals Limited

Curated by ChEMBL
LigandPNGBDBM50388341(CHEMBL2059241)copy SMILEScopy InChI
Affinity DataKi:  5.80nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G161WNPubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals Limited

Curated by ChEMBL
LigandPNGBDBM50388342(CHEMBL2059242)copy SMILEScopy InChI
Affinity DataKi:  6nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G161WNPubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals Limited

Curated by ChEMBL
LigandPNGBDBM50388331(CHEMBL2059499)copy SMILEScopy InChI
Affinity DataKi:  6.10nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G161WNPubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals Limited

Curated by ChEMBL
LigandPNGBDBM50388345(CHEMBL2059245)copy SMILEScopy InChI
Affinity DataKi:  6.40nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G161WNPubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals Limited

Curated by ChEMBL
LigandPNGBDBM50378647(CHEMBL1627122 | PI-88)copy SMILEScopy InChI
Affinity DataKi:  7.90nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G161WNPubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals Limited

Curated by ChEMBL
LigandPNGBDBM50388332(CHEMBL2059498)copy SMILEScopy InChI
Affinity DataKi:  8.40nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G161WNPubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals Limited

Curated by ChEMBL
LigandPNGBDBM50388346(CHEMBL2059246)copy SMILEScopy InChI
Affinity DataKi:  8.5nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G161WNPubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals Limited

Curated by ChEMBL
LigandPNGBDBM50388336(CHEMBL2059504)copy SMILEScopy InChI
Affinity DataKi:  9.10nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G161WNPubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals Limited

Curated by ChEMBL
LigandPNGBDBM50388335(CHEMBL2059503)copy SMILEScopy InChI
Affinity DataKi:  9.10nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G161WNPubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals Limited

Curated by ChEMBL
LigandPNGBDBM50388330(CHEMBL2059247)copy SMILEScopy InChI
Affinity DataKi:  10.5nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G161WNPubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals Limited

Curated by ChEMBL
LigandPNGBDBM50388328(CHEMBL2059505)copy SMILEScopy InChI
Affinity DataKi:  11.3nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G161WNPubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals Limited

Curated by ChEMBL
LigandPNGBDBM50388334(CHEMBL2059501)copy SMILEScopy InChI
Affinity DataKi:  16nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G161WNPubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals Limited

Curated by ChEMBL
LigandPNGBDBM50388333(CHEMBL2059502)copy SMILEScopy InChI
Affinity DataKi:  20nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G161WNPubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals Limited

Curated by ChEMBL
LigandPNGBDBM50388344(CHEMBL2059244)copy SMILEScopy InChI
Affinity DataKi:  22.3nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G161WNPubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals Limited

Curated by ChEMBL
LigandPNGBDBM50388340(CHEMBL2059510)copy SMILEScopy InChI
Affinity DataKi:  30nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G161WNPubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals Limited

Curated by ChEMBL
LigandPNGBDBM50388338(CHEMBL2059508)copy SMILEScopy InChI
Affinity DataKi:  111nMAssay Description:Inhibition of human recombinant heparanase after 2 to 24 hrs by WST1 dye based fondaparinux assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G161WNPubMed
TargetIsoleucyl-tRNA synthetase(Rattus norvegicus)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50093001((4aR,6S,7R,7aS)-7-[2-((S)-2-Amino-3-methyl-butyryl...)copy SMILEScopy InChI
Affinity DataIC50: 2.90nMAssay Description:Compound was evaluated for its inhibitory activity against Isoleucyl-tRNA synthetase from rat liverMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN94W3PubMed
TargetIsoleucyl-tRNA synthetase(Rattus norvegicus)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50093003((4aR,6S,7R,7aS)-7-[2-((2S,3S)-2-Amino-3-methyl-pen...)copy SMILEScopy InChI
Affinity DataIC50: 4.20nMAssay Description:Compound was evaluated for its inhibitory activity against Isoleucyl-tRNA synthetase from rat liverMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN94W3PubMed
TargetIsoleucine--tRNA ligase(Staphylococcus aureus)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50093003((4aR,6S,7R,7aS)-7-[2-((2S,3S)-2-Amino-3-methyl-pen...)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Compound was evaluated for its inhibitory activity against Isoleucyl-tRNA synthetase from staphylococcus aureus WCUH29More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN94W3PubMed
TargetLeucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Australian National University

Curated by ChEMBL
LigandPNGBDBM50093005((4aR,6S,7R,7aS)-7-[2-((S)-2-Amino-4-methyl-pentano...)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Compound was evaluated for its inhibitory activity against Leucyl-tRNA synthetase from staphylococcus aureus WCUH29More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN94W3PubMed
TargetIsoleucyl-tRNA synthetase(Rattus norvegicus)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50093004((4aR,6S,7R,7aS)-7-[2-((2S,3S)-2-Amino-3-methyl-pen...)copy SMILEScopy InChI
Affinity DataIC50: 17nMAssay Description:Compound was evaluated for its inhibitory activity against Isoleucyl-tRNA synthetase from rat liverMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN94W3PubMed
TargetIsoleucyl-tRNA synthetase(Rattus norvegicus)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50093002((4aR,6S,7R,7aS)-7-[2-((2S,3S)-2-Amino-3-methyl-pen...)copy SMILEScopy InChI
Affinity DataIC50: 25nMAssay Description:Compound was evaluated for its inhibitory activity against Isoleucyl-tRNA synthetase from rat liverMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN94W3PubMed
TargetValine--tRNA ligase(Homo sapiens (Human))
Australian National University

Curated by ChEMBL
LigandPNGBDBM50093001((4aR,6S,7R,7aS)-7-[2-((S)-2-Amino-3-methyl-butyryl...)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Compound was evaluated for its inhibitory activity against VRS (valyl tRNA synthetase) from staphylococcus aureus WCUH29More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN94W3PubMed
TargetIsoleucine--tRNA ligase(Staphylococcus aureus)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50093001((4aR,6S,7R,7aS)-7-[2-((S)-2-Amino-3-methyl-butyryl...)copy SMILEScopy InChI
Affinity DataIC50: 37nMAssay Description:Compound was evaluated for its inhibitory activity against Isoleucyl-tRNA synthetase from staphylococcus aureus WCUH29More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN94W3PubMed
TargetIsoleucine--tRNA ligase(Staphylococcus aureus)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50093004((4aR,6S,7R,7aS)-7-[2-((2S,3S)-2-Amino-3-methyl-pen...)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Compound was evaluated for its inhibitory activity against Isoleucyl-tRNA synthetase from staphylococcus aureus WCUH29More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN94W3PubMed
TargetIsoleucyl-tRNA synthetase(Rattus norvegicus)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50093005((4aR,6S,7R,7aS)-7-[2-((S)-2-Amino-4-methyl-pentano...)copy SMILEScopy InChI
Affinity DataIC50: 68nMAssay Description:Compound was evaluated for its inhibitory activity against Isoleucyl-tRNA synthetase from rat liverMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN94W3PubMed
TargetIsoleucine--tRNA ligase(Staphylococcus aureus)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50093002((4aR,6S,7R,7aS)-7-[2-((2S,3S)-2-Amino-3-methyl-pen...)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Compound was evaluated for its inhibitory activity against Isoleucyl-tRNA synthetase from staphylococcus aureus WCUH29More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN94W3PubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
University of Queensland

Curated by ChEMBL
LigandPNGBDBM18069(5-[(3,4,5-trimethoxyphenyl)methyl]pyrimidine-2,4-d...)copy SMILEScopy InChI
Affinity DataIC50: 123nMAssay Description:Inhibition of DHFR using dihydrofolate as substrate following 3 mins substrate preincubation measured after 3 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetValine--tRNA ligase(Homo sapiens (Human))
Australian National University

Curated by ChEMBL
LigandPNGBDBM50093003((4aR,6S,7R,7aS)-7-[2-((2S,3S)-2-Amino-3-methyl-pen...)copy SMILEScopy InChI
Affinity DataIC50: 126nMAssay Description:Compound was evaluated for its inhibitory activity against VRS (valyl tRNA synthetase) from staphylococcus aureus WCUH29More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN94W3PubMed
TargetFibroblast growth factor 1(Homo sapiens (Human))
Progen Pharmaceuticals Limited

Curated by ChEMBL
LigandPNGBDBM50374504(CHEMBL258321)copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Binding affinity at FGF1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24B326ZPubMed
TargetValine--tRNA ligase(Homo sapiens (Human))
Australian National University

Curated by ChEMBL
LigandPNGBDBM50093005((4aR,6S,7R,7aS)-7-[2-((S)-2-Amino-4-methyl-pentano...)copy SMILEScopy InChI
Affinity DataIC50: 290nMAssay Description:Compound was evaluated for its inhibitory activity against VRS (valyl tRNA synthetase) from staphylococcus aureus WCUH29More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN94W3PubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50380095(CHEMBL2012911)copy SMILEScopy InChI
Affinity DataIC50: 340nMAssay Description:Inhibition of DHFR using dihydrofolate as substrate following 3 mins substrate preincubation measured after 3 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27082FGPubMed
TargetIsoleucyl-tRNA synthetase(Rattus norvegicus)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50093006((4aR,6S,7R,7aS)-6-((2S,3S)-2-Benzyloxycarbonylamin...)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Compound was evaluated for its inhibitory activity against Isoleucyl-tRNA synthetase from rat liverMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN94W3PubMed
TargetIsoleucine--tRNA ligase(Staphylococcus aureus)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50093005((4aR,6S,7R,7aS)-7-[2-((S)-2-Amino-4-methyl-pentano...)copy SMILEScopy InChI
Affinity DataIC50: 910nMAssay Description:Compound was evaluated for its inhibitory activity against Isoleucyl-tRNA synthetase from staphylococcus aureus WCUH29More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN94W3PubMed
TargetLeucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Australian National University

Curated by ChEMBL
LigandPNGBDBM50093003((4aR,6S,7R,7aS)-7-[2-((2S,3S)-2-Amino-3-methyl-pen...)copy SMILEScopy InChI
Affinity DataIC50: 1.55E+3nMAssay Description:Compound was evaluated for its inhibitory activity against Leucyl-tRNA synthetase from staphylococcus aureus WCUH29More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN94W3PubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals Limited

Curated by ChEMBL
LigandPNGBDBM50179253((2R,3S,4S,5S,6R)-2-{[(2R,3S,4S,5R,6R)-2-{[(2R,3S,4...)copy SMILEScopy InChI
Affinity DataIC50: 1.64E+3nMAssay Description:Inhibitory activity against human platelet heparanase by Microcon ultrafiltration assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MG7P2VPubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals Limited

Curated by ChEMBL
LigandPNGBDBM50179254((2R,3S,4S,5S,6R)-2-{[(2R,3S,4S,5R,6R)-2-{[(2R,3S,4...)copy SMILEScopy InChI
Affinity DataIC50: 1.83E+3nMAssay Description:Inhibitory activity against human platelet heparanase by Microcon ultrafiltration assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MG7P2VPubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals Limited

Curated by ChEMBL
LigandPNGBDBM50179256(6-{5-[(3aS,4S,6aR)-2-oxo-hexahydro-1H-thieno[3,4-d...)copy SMILEScopy InChI
Affinity DataIC50: 1.85E+3nMAssay Description:Inhibitory activity against human platelet heparanase by Microcon ultrafiltration assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MG7P2VPubMed
TargetHeparanase(Homo sapiens (Human))
Progen Pharmaceuticals Limited

Curated by ChEMBL
LigandPNGBDBM50179255(CHEMBL265885 | N-[(2S,3S,4S,5S,6R)-3-{[(2R,3S,4S,5...)copy SMILEScopy InChI
Affinity DataIC50: 2.02E+3nMAssay Description:Inhibitory activity against human platelet heparanase by Microcon ultrafiltration assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MG7P2VPubMed
TargetLeucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Australian National University

Curated by ChEMBL
LigandPNGBDBM50093001((4aR,6S,7R,7aS)-7-[2-((S)-2-Amino-3-methyl-butyryl...)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+3nMAssay Description:Compound was evaluated for its inhibitory activity against Leucyl-tRNA synthetase from staphylococcus aureus WCUH29More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN94W3PubMed
TargetIsoleucine--tRNA ligase(Staphylococcus aureus)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50093008((4aR,6S,7R,7aS)-4-Carbamoyl-6-hydroxy-2-methyl-7-[...)copy SMILEScopy InChI
Affinity DataIC50: 3.27E+3nMAssay Description:Compound was evaluated for its inhibitory activity against Isoleucyl-tRNA synthetase from staphylococcus aureus WCUH29More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN94W3PubMed
TargetIsoleucyl-tRNA synthetase(Rattus norvegicus)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50093007((4aR,6S,7R,7aS)-4-Carbamoyl-2-methyl-6-((S)-3-meth...)copy SMILEScopy InChI
Affinity DataIC50: 6.10E+3nMAssay Description:Compound was evaluated for its inhibitory activity against Isoleucyl-tRNA synthetase from rat liverMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN94W3PubMed
TargetIsoleucine--tRNA ligase(Staphylococcus aureus)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50093007((4aR,6S,7R,7aS)-4-Carbamoyl-2-methyl-6-((S)-3-meth...)copy SMILEScopy InChI
Affinity DataIC50: 1.46E+4nMAssay Description:Compound was evaluated for its inhibitory activity against Isoleucyl-tRNA synthetase from staphylococcus aureus WCUH29More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN94W3PubMed
TargetIsoleucyl-tRNA synthetase(Rattus norvegicus)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50093008((4aR,6S,7R,7aS)-4-Carbamoyl-6-hydroxy-2-methyl-7-[...)copy SMILEScopy InChI
Affinity DataIC50: 2.23E+4nMAssay Description:Compound was evaluated for its inhibitory activity against Isoleucyl-tRNA synthetase from rat liverMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN94W3PubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50380092(CHEMBL2012918)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of DHFR using dihydrofolate as substrate following 3 mins substrate preincubation measured after 3 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27082FGPubMed
TargetLeucine--tRNA ligase, cytoplasmic(Homo sapiens (Human))
Australian National University

Curated by ChEMBL
LigandPNGBDBM50093004((4aR,6S,7R,7aS)-7-[2-((2S,3S)-2-Amino-3-methyl-pen...)copy SMILEScopy InChI
Affinity DataIC50: 1.86E+5nMAssay Description:Compound was evaluated for its inhibitory activity against Leucyl-tRNA synthetase from staphylococcus aureus WCUH29More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PN94W3PubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50380096(CHEMBL2012916)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibition of DHFR using dihydrofolate as substrate following 3 mins substrate preincubation measured after 3 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27082FGPubMed
TargetDihydrofolate reductase(Homo sapiens (Human))
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50380094(CHEMBL2012914)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibition of DHFR using dihydrofolate as substrate following 3 mins substrate preincubation measured after 3 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27082FGPubMed
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