Compile Data Set for Download or QSAR
Found 134 with Last Name = 'weinmann' and Initial = 'h'
TargetN-lysine methyltransferase SMYD2(Homo sapiens (Human))
BAYER Pharma AG

Curated by ChEMBL
LigandPNGBDBM50180955(CHEMBL3818617)copy SMILEScopy InChI
Affinity DataKi:  8nMAssay Description:Competitive inhibition of full length 6xHis-tagged SMYD2 (unknown origin) expressed in Escherichia coli using varying levels of Btn-Ahx-GSRAHSSHLKSKK...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN39S5PubMed
TargetN-lysine methyltransferase SMYD2(Homo sapiens (Human))
BAYER Pharma AG

Curated by ChEMBL
LigandPNGBDBM50180955(CHEMBL3818617)copy SMILEScopy InChI
Affinity DataKi:  28nMAssay Description:Uncompetitive inhibition of full length 6xHis-tagged SMYD2 (unknown origin) expressed in Escherichia coli using fixed levels of Btn-Ahx-GSRAHSSHLKSKK...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN39S5PubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
BAYER Pharma AG

Curated by ChEMBL
LigandPNGBDBM50181506(CHEMBL3819038)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Antagonist activity at PAR1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN39S5PubMed
TargetN-lysine methyltransferase SMYD2(Homo sapiens (Human))
BAYER Pharma AG

Curated by ChEMBL
LigandPNGBDBM50075102(CHEMBL3414623)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of SMYD2 (unknown origin) expressed in Escherichia coli BL21 (DE3) using Biotinaminohexanoyl-GSRAHSSHLKSKKGQSTSRH as substrate after 75 mi...More data for this Ligand-Target Pair
TargetN-lysine methyltransferase SMYD2(Homo sapiens (Human))
BAYER Pharma AG

Curated by ChEMBL
LigandPNGBDBM50180967(CHEMBL3818487)copy SMILEScopy InChI
Affinity DataIC50: 19nMAssay Description:Inhibition of SMYD2 (unknown origin) using H4 as substrate after 2hrs in presence 3H-SAM of by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN39S5PubMed
TargetLutropin-choriogonadotropic hormone receptor(Rattus norvegicus)
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50505787(CHEMBL4537998)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Antagonist activity at rat luteinizing hormone receptor expressed in rat ovary granulosa GLHR15 cell suspension assessed as reduction in agonist-indu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P34X6PubMed
TargetN-lysine methyltransferase SMYD2(Homo sapiens (Human))
BAYER Pharma AG

Curated by ChEMBL
LigandPNGBDBM50180955(CHEMBL3818617)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Inhibition of full length 6xHis-tagged SMYD2 (unknown origin) expressed in Escherichia coli using Btn-Ahx GSRAHSSHLKSKKGQSTSRH-amide as substrate aft...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN39S5PubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
BAYER Pharma AG

Curated by ChEMBL
LigandPNGBDBM50181502(CHEMBL3818510)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Antagonist activity at PAR1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN39S5PubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
BAYER Pharma AG

Curated by ChEMBL
LigandPNGBDBM50181504(CHEMBL3818898)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Antagonist activity at PAR1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN39S5PubMed
TargetN-lysine methyltransferase SMYD2(Homo sapiens (Human))
BAYER Pharma AG

Curated by ChEMBL
LigandPNGBDBM50180973(CHEMBL3819284)copy SMILEScopy InChI
Affinity DataIC50: 38nMAssay Description:Inhibition of SMYD2 (unknown origin) using H4 as substrate after 2hrs in presence 3H-SAM of by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN39S5PubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
BAYER Pharma AG

Curated by ChEMBL
LigandPNGBDBM50181505(CHEMBL3819204)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Antagonist activity at PAR1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN39S5PubMed
TargetN-lysine methyltransferase SMYD2(Homo sapiens (Human))
BAYER Pharma AG

Curated by ChEMBL
LigandPNGBDBM50180968(CHEMBL3818080)copy SMILEScopy InChI
Affinity DataIC50: 44nMAssay Description:Inhibition of SMYD2 (unknown origin) using H4 as substrate after 2hrs in presence 3H-SAM of by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN39S5PubMed
TargetLutropin-choriogonadotropic hormone receptor(Rattus norvegicus)
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50505783(CHEMBL4458424)copy SMILEScopy InChI
Affinity DataIC50: 46nMAssay Description:Antagonist activity at rat luteinizing hormone receptor expressed in rat ovary granulosa GLHR15 cell suspension assessed as reduction in agonist-indu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P34X6PubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
BAYER Pharma AG

Curated by ChEMBL
LigandPNGBDBM50181513(CHEMBL3819237)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Antagonist activity at PAR1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN39S5PubMed
TargetN-lysine methyltransferase SMYD2(Homo sapiens (Human))
BAYER Pharma AG

Curated by ChEMBL
LigandPNGBDBM50180971(CHEMBL3818322)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Inhibition of SMYD2 (unknown origin) using H4 as substrate after 2hrs in presence 3H-SAM of by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN39S5PubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
BAYER Pharma AG

Curated by ChEMBL
LigandPNGBDBM50181507(CHEMBL3818421)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Antagonist activity at PAR1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN39S5PubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
BAYER Pharma AG

Curated by ChEMBL
LigandPNGBDBM50181511(CHEMBL3819343)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Antagonist activity at PAR1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN39S5PubMed
TargetN-lysine methyltransferase SMYD2(Homo sapiens (Human))
BAYER Pharma AG

Curated by ChEMBL
LigandPNGBDBM50180955(CHEMBL3818617)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Inhibition of N-terminal 2xc-myc-tagged human SMYD2 transfected in human MDA-MB-231 cells assessed as reduction in AHNAK methylation after 72 hrs by ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN39S5PubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
BAYER Pharma AG

Curated by ChEMBL
LigandPNGBDBM50181509(CHEMBL3817930)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Antagonist activity at PAR1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN39S5PubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
BAYER Pharma AG

Curated by ChEMBL
LigandPNGBDBM50181512(CHEMBL3819277 | US10023539, Example WO 2006/07235...)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:Antagonist activity at PAR1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN39S5PubMed
TargetN-lysine methyltransferase SMYD2(Homo sapiens (Human))
BAYER Pharma AG

Curated by ChEMBL
LigandPNGBDBM50180970(CHEMBL3819554)copy SMILEScopy InChI
Affinity DataIC50: 71nMAssay Description:Inhibition of SMYD2 (unknown origin) using H4 as substrate after 2hrs in presence 3H-SAM of by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN39S5PubMed
TargetLuteinizing hormone/choriogondaotropin receptor(Macaca fascicularis)
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50505787(CHEMBL4537998)copy SMILEScopy InChI
Affinity DataIC50: 78nMAssay Description:Antagonist activity at cynomolgus monkey luteinizing hormone receptor expressed in HEK293 cells assessed as reduction in agonist-induced cAMP product...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P34X6PubMed
TargetN-lysine methyltransferase SMYD2(Homo sapiens (Human))
BAYER Pharma AG

Curated by ChEMBL
LigandPNGBDBM50181508(CHEMBL3818083 | US10023539, Example 4.2)copy SMILEScopy InChI
Affinity DataIC50: 80nMAssay Description:Inhibition of full length 6xHis-tagged SMYD2 (unknown origin) expressed in Escherichia coli using Btn-Ahx GSRAHSSHLKSKKGQSTSRH-amide as substrate aft...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN39S5PubMed
TargetN-lysine methyltransferase SMYD2(Homo sapiens (Human))
BAYER Pharma AG

Curated by ChEMBL
LigandPNGBDBM50180974(CHEMBL3818092 | US10023539, Example 33.2)copy SMILEScopy InChI
Affinity DataIC50: 80nMAssay Description:Inhibition of SMYD2 (unknown origin) using H4 as substrate after 2hrs in presence 3H-SAM of by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN39S5PubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
BAYER Pharma AG

Curated by ChEMBL
LigandPNGBDBM50181510(CHEMBL3818750)copy SMILEScopy InChI
Affinity DataIC50: 80nMAssay Description:Antagonist activity at PAR1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN39S5PubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50505809(CHEMBL4460075)copy SMILEScopy InChI
Affinity DataIC50: 81nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P34X6PubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50383229(CHEMBL2032175)copy SMILEScopy InChI
Affinity DataIC50: 95nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P34X6PubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50505787(CHEMBL4537998)copy SMILEScopy InChI
Affinity DataIC50: 96nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P34X6PubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50505787(CHEMBL4537998)copy SMILEScopy InChI
Affinity DataIC50: 97nMAssay Description:Negative allosteric modulation of human luteinizing hormone receptor assessed as reduction in glycoprotein human luteinizing hormone-induced agonist ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P34X6PubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
BAYER Pharma AG

Curated by ChEMBL
LigandPNGBDBM50180978(CHEMBL3819515)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Antagonist activity at PAR1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN39S5PubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50505791(CHEMBL4587440)copy SMILEScopy InChI
Affinity DataIC50: 102nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P34X6PubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50505799(CHEMBL4573509)copy SMILEScopy InChI
Affinity DataIC50: 107nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P34X6PubMed
TargetN-lysine methyltransferase SMYD2(Homo sapiens (Human))
BAYER Pharma AG

Curated by ChEMBL
LigandPNGBDBM50180969(CHEMBL3818526)copy SMILEScopy InChI
Affinity DataIC50: 119nMAssay Description:Inhibition of SMYD2 (unknown origin) using H4 as substrate after 2hrs in presence 3H-SAM of by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN39S5PubMed
TargetN-lysine methyltransferase SMYD2(Homo sapiens (Human))
BAYER Pharma AG

Curated by ChEMBL
LigandPNGBDBM50396022(CHEMBL2169920)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Inhibition of SMYD2 (unknown origin) expressed in Escherichia coli BL21 (DE3) using Biotinaminohexanoyl-GSRAHSSHLKSKKGQSTSRH as substrate after 75 mi...More data for this Ligand-Target Pair
TargetN-lysine methyltransferase SMYD2(Homo sapiens (Human))
BAYER Pharma AG

Curated by ChEMBL
LigandPNGBDBM50396022(CHEMBL2169920)copy SMILEScopy InChI
Affinity DataIC50: 120nMAssay Description:Inhibition of SMYD2 (unknown origin) expressed in Escherichia coli BL21 (DE3) using Biotinaminohexanoyl-GSRAHSSHLKSKKGQSTSRH as substrate after 75 mi...More data for this Ligand-Target Pair
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50505796(CHEMBL4531781)copy SMILEScopy InChI
Affinity DataIC50: 127nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P34X6PubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
BAYER Pharma AG

Curated by ChEMBL
LigandPNGBDBM50181454(CHEMBL3818932)copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Antagonist activity at PAR1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RN39S5PubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50505785(CHEMBL4443605)copy SMILEScopy InChI
Affinity DataIC50: 174nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P34X6PubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50505783(CHEMBL4458424)copy SMILEScopy InChI
Affinity DataIC50: 185nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P34X6PubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50505811(CHEMBL4461980)copy SMILEScopy InChI
Affinity DataIC50: 193nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P34X6PubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50505787(CHEMBL4537998)copy SMILEScopy InChI
Affinity DataIC50: 200nMAssay Description:Negative allosteric modulation of human luteinizing hormone receptor assessed as reduction in glycoprotein human luteinizing hormone-induced agonist ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P34X6PubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50505797(CHEMBL4522381)copy SMILEScopy InChI
Affinity DataIC50: 207nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P34X6PubMed
TargetLutropin-choriogonadotropic hormone receptor(Rattus norvegicus)
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50505793(CHEMBL4593222)copy SMILEScopy InChI
Affinity DataIC50: 212nMAssay Description:Antagonist activity at rat luteinizing hormone receptor expressed in rat ovary granulosa GLHR15 cell suspension assessed as reduction in agonist-indu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P34X6PubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50505798(CHEMBL4581889)copy SMILEScopy InChI
Affinity DataIC50: 275nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P34X6PubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50505812(CHEMBL4555151)copy SMILEScopy InChI
Affinity DataIC50: 312nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P34X6PubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50505795(CHEMBL4579421)copy SMILEScopy InChI
Affinity DataIC50: 332nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P34X6PubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50505793(CHEMBL4593222)copy SMILEScopy InChI
Affinity DataIC50: 378nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P34X6PubMed
TargetN-lysine methyltransferase SMYD2(Homo sapiens (Human))
BAYER Pharma AG

Curated by ChEMBL
LigandPNGBDBM50075102(CHEMBL3414623)copy SMILEScopy InChI
Affinity DataIC50: 388nMAssay Description:Inhibition of SMYD2 (unknown origin) using H4 as substrate after 2hrs in presence 3H-SAM of by scintillation proximity assayMore data for this Ligand-Target Pair
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50505789(CHEMBL4471621)copy SMILEScopy InChI
Affinity DataIC50: 403nMAssay Description:Antagonist activity at human luteinizing hormone receptor assessed as reduction in agonist-induced cAMP production preincubated for 20 mins followed ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P34X6PubMed
TargetLutropin-choriogonadotropic hormone receptor(Rattus norvegicus)
Bayer AG

Curated by ChEMBL
LigandPNGBDBM50505789(CHEMBL4471621)copy SMILEScopy InChI
Affinity DataIC50: 412nMAssay Description:Antagonist activity at rat luteinizing hormone receptor expressed in rat ovary granulosa GLHR15 cell suspension assessed as reduction in agonist-indu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29P34X6PubMed
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