Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetMelanocortin receptor 5(Mus musculus (Mouse))
University of Florida

Curated by ChEMBL
LigandPNGBDBM50374124(CHEMBL272439)copy SMILEScopy InChI
Affinity DataEC50:  1.70E+4nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0P61PubMed
TargetMelanocortin receptor 3(Mus musculus)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50374124(CHEMBL272439)copy SMILEScopy InChI
Affinity DataEC50:  3.07E+4nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0P61PubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50374124(CHEMBL272439)copy SMILEScopy InChI
Affinity DataEC50:  1.80E+3nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells assessed as forskolin-stimulated response by beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KH0P61PubMed