Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 12 hits in this display   

TargetExcitatory amino acid transporter 2(Homo sapiens (Human))
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159150(CHEMBL3787264)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of human EAAT2 assessed as [3H]Asp uptakeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2000408PubMed
TargetExcitatory amino acid transporter 1(Homo sapiens (Human))
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159150(CHEMBL3787264)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of human EAAT1 assessed as [3H]Asp uptakeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2000408PubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159150(CHEMBL3787264)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of human EAAT3 assessed as [3H]Asp uptakeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2000408PubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159150(CHEMBL3787264)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at rat mGlu4 receptor expressed in HEK293 cells assessed as IP1 accumulation by IP-One functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2000408PubMed
TargetMetabotropic glutamate receptor 6(Rattus norvegicus (Rat))
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159150(CHEMBL3787264)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at rat mGlu6 receptor expressed in HEK293 cells assessed as IP1 accumulation by IP-One functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2000408PubMed
TargetMetabotropic glutamate receptor 8(Rattus norvegicus (Rat))
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159150(CHEMBL3787264)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at rat mGlu8 receptor expressed in HEK293 cells assessed as IP1 accumulation by IP-One functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2000408PubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159150(CHEMBL3787264)copy SMILEScopy InChI
Affinity DataEC50:  1.19E+5nMAssay Description:Agonist activity at rat mGlu2 receptor by FRET based mGlu sensor assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2000408PubMed
TargetMetabotropic glutamate receptor 3(Rattus norvegicus (Rat))
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159150(CHEMBL3787264)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at rat mGlu3 receptor by FRET based mGlu sensor assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2000408PubMed
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159150(CHEMBL3787264)copy SMILEScopy InChI
Affinity DataEC50:  3.37E+4nMAssay Description:Agonist activity at rat mGlu2 receptor expressed in HEK293 cells assessed as IP1 accumulation by IP-One functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2000408PubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159150(CHEMBL3787264)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at rat mGlu5 receptor expressed in HEK293 cells assessed as IP1 accumulation by IP-One functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2000408PubMed
TargetMetabotropic glutamate receptor 1(RAT)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159150(CHEMBL3787264)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at rat mGlu1 receptor expressed in HEK293 cells assessed as IP1 accumulation by IP-One functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2000408PubMed
TargetMetabotropic glutamate receptor 7(Rattus norvegicus (Rat))
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50159150(CHEMBL3787264)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at rat mGlu7 receptor expressed in HEK293 cells assessed as IP1 accumulation by IP-One functional assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2000408PubMed