Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetMelanocortin receptor 4(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50089424(CHEMBL3577979)copy SMILEScopy InChI
Affinity DataKi:  160nMAssay Description:Displacement of MTII from mouse MC4R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T155C9PubMed
TargetMelanocortin receptor 3(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50089424(CHEMBL3577979)copy SMILEScopy InChI
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of MTII from mouse MC3R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T155C9PubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50089424(CHEMBL3577979)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+8nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by cAMP functional bioassayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T155C9PubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50089424(CHEMBL3577979)copy SMILEScopy InChI
Affinity DataEC50:  1.76E+4nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by cAMP functional bioassayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2T155C9PubMed