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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
6
hits in this display
Target
Melanocortin receptor 4
(Mus musculus)
University of Minnesota
Curated by
ChEMBL
Ligand
BDBM50514457
(CHEMBL4565367)
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copy InChI
Affinity Data
IC50: 8.20nM
Assay Description:
Displacement of [125I]-NDP-MSH from mouse melanocortin receptor 4 expressed in HEK293 cell mebranes incubated for 1 hr by automatic gamma counting me...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q25142KG
PubMed
Target
Melanocortin receptor 4
(Homo sapiens (Human))
University of Minnesota
Curated by
ChEMBL
Ligand
BDBM50514457
(CHEMBL4565367)
copy SMILES
copy InChI
Affinity Data
IC50: 32nM
Assay Description:
Displacement of [125I]-NDP-MSH from human melanocortin receptor 4 expressed in HEK293 cell mebranes incubated for 1 hr by automatic gamma counting me...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q25142KG
PubMed
Target
Melanocortin receptor 5
(Mus musculus (Mouse))
University of Minnesota
Curated by
ChEMBL
Ligand
BDBM50514457
(CHEMBL4565367)
copy SMILES
copy InChI
Affinity Data
IC50: 2.70E+3nM
Assay Description:
Displacement of [125I]-NDP-MSH from mouse melanocortin receptor 5 expressed in HEK293 cell mebranes incubated for 1 hr by automatic gamma counting me...
More data for this Ligand-Target Pair
Target Info
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q25142KG
PubMed
Target
Melanocyte-stimulating hormone receptor
(Mus musculus)
University of Minnesota
Curated by
ChEMBL
Ligand
BDBM50514457
(CHEMBL4565367)
copy SMILES
copy InChI
Affinity Data
IC50: 8.00E+3nM
Assay Description:
Displacement of [125I]-NDP-MSH from mouse melanocortin receptor 1 expressed in HEK293 cell mebranes incubated for 1 hr by automatic gamma counting me...
More data for this Ligand-Target Pair
Target Info
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q25142KG
PubMed
Target
Melanocortin receptor 3
(Mus musculus)
University of Minnesota
Curated by
ChEMBL
Ligand
BDBM50514457
(CHEMBL4565367)
copy SMILES
copy InChI
Affinity Data
IC50: 1.00E+4nM
Assay Description:
Displacement of [125I]-NDP-MSH from mouse melanocortin receptor 3 expressed in HEK293 cell mebranes incubated for 1 hr by automatic gamma counting me...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q25142KG
PubMed
Target
Melanocortin receptor 5
(Mus musculus (Mouse))
University of Minnesota
Curated by
ChEMBL
Ligand
BDBM50514457
(CHEMBL4565367)
copy SMILES
copy InChI
Affinity Data
EC50: >1.00E+5nM
Assay Description:
Agonist activity at mouse melanocortin receptor 5 expressed in HEK293 cells assessed as stimulation of cAMP accumulation incubated for 2 hrs by cAMP ...
More data for this Ligand-Target Pair
Target Info
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q25142KG
PubMed