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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Melanocortin receptor 3
(Mus musculus)
University of Minnesota
Curated by
ChEMBL
Ligand
BDBM50258957
(CHEMBL4066929)
copy SMILES
copy InChI
Affinity Data
EC50: >1.00E+5nM
Assay Description:
Agonist activity at mouse melanocortin receptor 3 expressed in HEK293 cells assessed as increase in cAMP accumulation after 2 hrs by AlphaScreen assa...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2DN47H1
PubMed
Target
Melanocortin receptor 4
(Mus musculus)
University of Minnesota
Curated by
ChEMBL
Ligand
BDBM50258957
(CHEMBL4066929)
copy SMILES
copy InChI
Affinity Data
EC50: >1.00E+5nM
Assay Description:
Agonist activity at mouse melanocortin receptor 4 expressed in HEK293 cells assessed as increase in cAMP accumulation after 2 hrs by AlphaScreen assa...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2DN47H1
PubMed
Target
Melanocyte-stimulating hormone receptor
(Mus musculus)
University of Minnesota
Curated by
ChEMBL
Ligand
BDBM50258957
(CHEMBL4066929)
copy SMILES
copy InChI
Affinity Data
EC50: >1.00E+5nM
Assay Description:
Agonist activity at mouse melanocortin receptor 1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 2 hrs by AlphaScreen assa...
More data for this Ligand-Target Pair
Target Info
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2DN47H1
PubMed