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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Somatostatin receptor type 2
(Homo sapiens (Human))
Ipsen Pharma S.A.S.
US Patent
Ligand
BDBM144745
(US8952128, 6C)
copy SMILES
Affinity Data
Ki: 0.150nM ΔG°: -56.1kJ/mole
pH: 7.6 T: 2°C
Assay Description:
Membranes for in vitro receptor binding assays were obtained by the following procedures. CHO-K1 cells expressing one of the somatostatin receptors w...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
BindingDB Entry DOI:
10.7270/Q2057DNG
US Patent
Target
D(2) dopamine receptor
(Homo sapiens (Human))
Ipsen Pharma S.A.S.
US Patent
Ligand
BDBM144745
(US8952128, 6C)
copy SMILES
Affinity Data
Ki: 30.3nM
pH: 7.6
Assay Description:
The affinity of a test compound for the human dopamine receptor subtype hDRD2 was determined by radioligand binding assays in CHO-K1 cells stably tra...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
BindingDB Entry DOI:
10.7270/Q2057DNG
US Patent