Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetSomatostatin receptor type 2(Homo sapiens (Human))
Ipsen Pharma S.A.S.

US Patent
LigandPNGBDBM144758(US8952128, 16)copy SMILES
Affinity DataKi:  0.0400nM ΔG°:  -59.3kJ/molepH: 7.6 T: 2°CAssay Description:Membranes for in vitro receptor binding assays were obtained by the following procedures. CHO-K1 cells expressing one of the somatostatin receptors w...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2057DNGUS Patent
TargetD(2) dopamine receptor(Homo sapiens (Human))
Ipsen Pharma S.A.S.

US Patent
LigandPNGBDBM144758(US8952128, 16)copy SMILES
Affinity DataKi:  22.5nMpH: 7.6Assay Description:The affinity of a test compound for the human dopamine receptor subtype hDRD2 was determined by radioligand binding assays in CHO-K1 cells stably tra...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2057DNGUS Patent