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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
6
hits in this display
Target
Somatostatin receptor type 3
(Homo sapiens (Human))
Salk Institute
Curated by
ChEMBL
Ligand
BDBM50352480
(CHEMBL1824051)
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Affinity Data
IC50: 1.5nM
Assay Description:
Displacement of 125I-[LTT]-SRIF-28 from human sst3 receptor in CCL39 cells after 2 hrs by autoradiography
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2BV7H1N
PubMed
Target
Somatostatin receptor type 1
(Homo sapiens (Human))
Salk Institute
Curated by
ChEMBL
Ligand
BDBM50352480
(CHEMBL1824051)
copy SMILES
copy InChI
Affinity Data
IC50: 2.70nM
Assay Description:
Displacement of 125I-[LTT]-SRIF-28 from human sst1 receptor in CHO cells after 2 hrs by autoradiography
More data for this Ligand-Target Pair
Target Info
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2BV7H1N
PubMed
Target
Somatostatin receptor type 4
(Homo sapiens (Human))
Salk Institute
Curated by
ChEMBL
Ligand
BDBM50352480
(CHEMBL1824051)
copy SMILES
copy InChI
Affinity Data
IC50: 12nM
Assay Description:
Displacement of 125I-[LTT]-SRIF-28 from human sst4 receptor in CCL39 cells after 2 hrs by autoradiography
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2BV7H1N
PubMed
Target
Somatostatin receptor type 2
(Homo sapiens (Human))
Salk Institute
Curated by
ChEMBL
Ligand
BDBM50352480
(CHEMBL1824051)
copy SMILES
copy InChI
Affinity Data
IC50: 15nM
Assay Description:
Displacement of 125I-[LTT]-SRIF-28 from human sst2 receptor in CCL39 cells after 2 hrs by autoradiography
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2BV7H1N
PubMed
Target
Somatostatin receptor type 5
(Homo sapiens (Human))
Salk Institute
Curated by
ChEMBL
Ligand
BDBM50352480
(CHEMBL1824051)
copy SMILES
copy InChI
Affinity Data
IC50: 69nM
Assay Description:
Displacement of 125I-[LTT]-SRIF-28 from human sst5 receptor in HEK293 cells after 2 hrs by autoradiography
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2BV7H1N
PubMed
Target
Somatostatin receptor type 3
(Homo sapiens (Human))
Salk Institute
Curated by
ChEMBL
Ligand
BDBM50352480
(CHEMBL1824051)
copy SMILES
copy InChI
Affinity Data
EC50: 0.350nM
Assay Description:
Agonist activity at human sst3 receptor expressed in CCL39 cells after 5 hrs by luciferase reporter gene assay
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2BV7H1N
PubMed