Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 10 hits in this display   

TargetSomatostatin receptor type 2(Homo sapiens (Human))
Technische Universit£t M£nchen

Curated by ChEMBL
LigandPNGBDBM50165164(CHEMBL262135 | CHEMBL430066 | Radiolabeled octreot...)copy SMILEScopy InChI
Affinity DataIC50: 0.200nMAssay Description:In vitro inhibition of [125I][Leu8,D-Trp22,Tyr25] somatostatin 28 binding to human somatostatin receptor type 2 expressed in CCL39 cells; (n=3)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0ND0PubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Technische Universit£t M£nchen

Curated by ChEMBL
LigandPNGBDBM50165164(CHEMBL262135 | CHEMBL430066 | Radiolabeled octreot...)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:In vitro inhibition of [125I][Leu8,D-Trp22,Tyr25] somatostatin 28 binding to human somatostatin receptor type 2 expressed in CCL39 cells; (n=3)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0ND0PubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Technische Universit£t M£nchen

Curated by ChEMBL
LigandPNGBDBM50165164(CHEMBL262135 | CHEMBL430066 | Radiolabeled octreot...)copy SMILEScopy InChI
Affinity DataIC50: 187nMAssay Description:In vitro inhibition of [125I][Leu8,D-Trp22,Tyr25] somatostatin 28 binding to human somatostatin receptor type 5 expressed in CHO-K1 cells; (n=3)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0ND0PubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Technische Universit£t M£nchen

Curated by ChEMBL
LigandPNGBDBM50165164(CHEMBL262135 | CHEMBL430066 | Radiolabeled octreot...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:In vitro inhibition of [125I][Leu8,D-Trp22,Tyr25] somatostatin 28 binding to human somatostatin receptor type 4 expressed in CCL39 cells; (n=3)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0ND0PubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Technische Universit£t M£nchen

Curated by ChEMBL
LigandPNGBDBM50165164(CHEMBL262135 | CHEMBL430066 | Radiolabeled octreot...)copy SMILEScopy InChI
Affinity DataIC50: 377nMAssay Description:In vitro inhibition of [125I][Leu8,D-Trp22,Tyr25] somatostatin 28 binding to human somatostatin receptor type 5 expressed in CHO-K1 cells; (n=3)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0ND0PubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Technische Universit£t M£nchen

Curated by ChEMBL
LigandPNGBDBM50165164(CHEMBL262135 | CHEMBL430066 | Radiolabeled octreot...)copy SMILEScopy InChI
Affinity DataIC50: 523nMAssay Description:In vitro inhibition of [125I][Leu8,D-Trp22,Tyr25] somatostatin 28 binding to human somatostatin receptor type 4 expressed in CCL39 cells; (n=3)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0ND0PubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Technische Universit£t M£nchen

Curated by ChEMBL
LigandPNGBDBM50165164(CHEMBL262135 | CHEMBL430066 | Radiolabeled octreot...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro inhibition of [125I][Leu8,D-Trp22,Tyr25] somatostatin 28 binding to human somatostatin receptor type 3 expressed in CCL39 cells; (n=3)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0ND0PubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Technische Universit£t M£nchen

Curated by ChEMBL
LigandPNGBDBM50165164(CHEMBL262135 | CHEMBL430066 | Radiolabeled octreot...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro inhibition of [125I][Leu8,D-Trp22,Tyr25] somatostatin 28 binding to human somatostatin receptor type 3 expressed in CCL39 cells; (n=3)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0ND0PubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Technische Universit£t M£nchen

Curated by ChEMBL
LigandPNGBDBM50165164(CHEMBL262135 | CHEMBL430066 | Radiolabeled octreot...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of [125I][Leu8,D-Trp22,Tyr25] somatostatin 28 binding to human somatostatin receptor type 1 expressed in CHO-K1 cells; (n=4)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0ND0PubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Technische Universit£t M£nchen

Curated by ChEMBL
LigandPNGBDBM50165164(CHEMBL262135 | CHEMBL430066 | Radiolabeled octreot...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of [125I][Leu8,D-Trp22,Tyr25] somatostatin 28 binding to human somatostatin receptor type 1 expressed in CHO-K1 cells; (n=3)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0ND0PubMed