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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
5
hits in this display
Target
Melanocyte-stimulating hormone receptor
(Homo sapiens (Human))
University of Arizona
Curated by
ChEMBL
Ligand
BDBM50141029
(1N-(1-carbamoyl-2-hydroxypropyl)-15-[3-amino(imino...)
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Affinity Data
EC50: 1.00E+4nM
Assay Description:
Effective concentration required for maximum agonist response at melanocortin 1 receptor from frog skin.
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2XP75PK
PubMed
Target
Melanocortin receptor 4
(Mus musculus)
University of Arizona
Curated by
ChEMBL
Ligand
BDBM50141029
(1N-(1-carbamoyl-2-hydroxypropyl)-15-[3-amino(imino...)
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copy InChI
Affinity Data
EC50: 8.90nM
Assay Description:
Effective concentration for maximum agonist response towards mouse melanocortin 4 receptor
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2XP75PK
PubMed
Target
Melanocortin receptor 5
(Mus musculus (Mouse))
University of Arizona
Curated by
ChEMBL
Ligand
BDBM50141029
(1N-(1-carbamoyl-2-hydroxypropyl)-15-[3-amino(imino...)
copy SMILES
copy InChI
Affinity Data
EC50: 0.550nM
Assay Description:
Maximum agonist response for mouse melanocortin 5 receptor (MC5R)
More data for this Ligand-Target Pair
Target Info
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2XP75PK
PubMed
Target
Melanocyte-stimulating hormone receptor
(Mus musculus)
University of Arizona
Curated by
ChEMBL
Ligand
BDBM50141029
(1N-(1-carbamoyl-2-hydroxypropyl)-15-[3-amino(imino...)
copy SMILES
copy InChI
Affinity Data
EC50: 35nM
Assay Description:
Maximal agonist response of mouse melanocortin 1 receptor (MC1R)
More data for this Ligand-Target Pair
Target Info
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2XP75PK
PubMed
Target
Melanocortin receptor 3
(Rattus norvegicus)
University of Arizona
Curated by
ChEMBL
Ligand
BDBM50141029
(1N-(1-carbamoyl-2-hydroxypropyl)-15-[3-amino(imino...)
copy SMILES
copy InChI
Affinity Data
EC50: 31nM
Assay Description:
Maximal agonist response at rat melanocortin 3 receptor (MC3R)
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2XP75PK
PubMed