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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
5
hits in this display
Target
Somatostatin receptor type 4
(Homo sapiens (Human))
Salk Institute
Curated by
ChEMBL
Ligand
BDBM50136781
(6-amino-12-(4-aminobenzyl)-18-(4-aminobutyl)-9,24-...)
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copy InChI
Affinity Data
IC50: 8.70nM
Assay Description:
Binding affinity at human Somatostatin receptor type 4 by [125I][Leu8,D-Trp22,Tyr25]SRIF-28 displacement.
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2FX7B50
PubMed
Target
Somatostatin receptor type 5
(Homo sapiens (Human))
Salk Institute
Curated by
ChEMBL
Ligand
BDBM50136781
(6-amino-12-(4-aminobenzyl)-18-(4-aminobutyl)-9,24-...)
copy SMILES
copy InChI
Affinity Data
IC50: 101nM
Assay Description:
Binding affinity at human Somatostatin receptor type 5 by [125I][Leu8,D-Trp22,Tyr25]SRIF-28 displacement.
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2FX7B50
PubMed
Target
Somatostatin receptor type 2
(Homo sapiens (Human))
Salk Institute
Curated by
ChEMBL
Ligand
BDBM50136781
(6-amino-12-(4-aminobenzyl)-18-(4-aminobutyl)-9,24-...)
copy SMILES
copy InChI
Affinity Data
IC50: 102nM
Assay Description:
Binding affinity at human Somatostatin receptor type 2 by [125I][Leu8,D-Trp22,Tyr25]SRIF-28 displacement.
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2FX7B50
PubMed
Target
Somatostatin receptor type 3
(Homo sapiens (Human))
Salk Institute
Curated by
ChEMBL
Ligand
BDBM50136781
(6-amino-12-(4-aminobenzyl)-18-(4-aminobutyl)-9,24-...)
copy SMILES
copy InChI
Affinity Data
IC50: 186nM
Assay Description:
Binding affinity at human Somatostatin receptor type 3 by [125I][Leu8,D-Trp22,Tyr25]SRIF-28 displacement.
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2FX7B50
PubMed
Target
Somatostatin receptor type 1
(Homo sapiens (Human))
Salk Institute
Curated by
ChEMBL
Ligand
BDBM50136781
(6-amino-12-(4-aminobenzyl)-18-(4-aminobutyl)-9,24-...)
copy SMILES
copy InChI
Affinity Data
IC50: 1.00E+3nM
Assay Description:
Binding affinity at human Somatostatin receptor type 1 by [125I][Leu8,D-Trp22,Tyr25]SRIF-28 displacement.
More data for this Ligand-Target Pair
Target Info
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2FX7B50
PubMed