Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetDiacylglycerol kinase alpha/zeta(Homo sapiens)
Therachem Research Medilab, LLC.

Curated by ChEMBL
LigandPNGBDBM50541810(CHEMBL4645744)copy SMILEScopy InChI
Affinity DataIC50: 43nMAssay Description:Inhibition of DGKA/DGKZ in human CD8 cells assessed as induction of CD8 activation by measuring IFNgamma level after 20 hrs by AlphaLISA assayMore data for this Ligand-Target Pair
Ligand InfoMCE
PC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20868V5PubMed
TargetDiacylglycerol kinase alpha(Homo sapiens)
Therachem Research Medilab, LLC.

Curated by ChEMBL
LigandPNGBDBM50541810(CHEMBL4645744)copy SMILEScopy InChI
Affinity DataIC50: 190nMAssay Description:Inhibition of full-length C-terminal His6 tagged TVMV-pFBgate fused human DGKalpha expressed in baculovirus infected Sf9 insect cells using liposome ...More data for this Ligand-Target Pair
Ligand InfoMCE
PC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20868V5PubMed
TargetDiacylglycerol kinase zeta(Homo sapiens)
Therachem Research Medilab, LLC.

Curated by ChEMBL
LigandPNGBDBM50541810(CHEMBL4645744)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Inhibition of full length C-terminal His6tagged TVMV-His-pFBgate fused human DGK-zeta expressed in baculovirus infected Sf9 insect cells using liposo...More data for this Ligand-Target Pair
Ligand InfoMCE
PC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20868V5PubMed
TargetDiacylglycerol kinase zeta(Homo sapiens)
Therachem Research Medilab, LLC.

Curated by ChEMBL
LigandPNGBDBM50541810(CHEMBL4645744)copy SMILEScopy InChI
Affinity DataIC50: 460nMAssay Description:Inhibition of DGKalpha/zeta in human whole blood assessed as induction of T-cell activation by measuring IFNgamma level preincubated for 1 hr followe...More data for this Ligand-Target Pair
Ligand InfoMCE
PC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20868V5PubMed