Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetMelanocortin receptor 4(Mus musculus)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50427678(CHEMBL2323788)copy SMILEScopy InChI
Affinity DataEC50:  705nMAssay Description:Agonist activity at mouse MC4 receptor expressed in HEK293 cells after 6 hrs by cAMP-based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NS0W8SPubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University of Florida

Curated by ChEMBL
LigandPNGBDBM50427678(CHEMBL2323788)copy SMILEScopy InChI
Affinity DataEC50:  690nMAssay Description:Agonist activity at mouse MC5 receptor expressed in HEK293 cells after 6 hrs by cAMP-based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NS0W8SPubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50427678(CHEMBL2323788)copy SMILEScopy InChI
Affinity DataEC50:  52nMAssay Description:Agonist activity at mouse MC1 receptor expressed in HEK293 cells after 6 hrs by cAMP-based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NS0W8SPubMed
TargetMelanocortin receptor 3(Mus musculus)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50427678(CHEMBL2323788)copy SMILEScopy InChI
Affinity DataEC50:  4.02E+3nMAssay Description:Agonist activity at mouse MC3 receptor expressed in HEK293 cells after 6 hrs by cAMP-based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NS0W8SPubMed