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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
5
hits in this display
Target
Somatostatin receptor type 4
(Homo sapiens (Human))
Salk Institute
Curated by
ChEMBL
Ligand
BDBM50136804
(CHEMBL439077 | Somatostatin analogue)
copy SMILES
copy InChI
Affinity Data
IC50: 1.20nM
Assay Description:
Binding affinity towards human somatostatin receptor type 4 using [125I]-[Leu8,DTrp22,Tyr25]SRIF-28 as radioligand.
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2MK6C9X
PubMed
Target
Somatostatin receptor type 5
(Homo sapiens (Human))
Salk Institute
Curated by
ChEMBL
Ligand
BDBM50136804
(CHEMBL439077 | Somatostatin analogue)
copy SMILES
copy InChI
Affinity Data
IC50: 34nM
Assay Description:
Binding affinity towards human somatostatin receptor type 5 using [125I]-[Leu8,DTrp22,Tyr25]SRIF-28 as radioligand.
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2MK6C9X
PubMed
Target
Somatostatin receptor type 2
(Homo sapiens (Human))
Salk Institute
Curated by
ChEMBL
Ligand
BDBM50136804
(CHEMBL439077 | Somatostatin analogue)
copy SMILES
copy InChI
Affinity Data
IC50: 56nM
Assay Description:
Binding affinity towards human somatostatin receptor type 2 using [125I]-[Leu8,DTrp22,Tyr25]SRIF-28 as radioligand.
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2MK6C9X
PubMed
Target
Somatostatin receptor type 3
(Homo sapiens (Human))
Salk Institute
Curated by
ChEMBL
Ligand
BDBM50136804
(CHEMBL439077 | Somatostatin analogue)
copy SMILES
copy InChI
Affinity Data
IC50: 263nM
Assay Description:
Binding affinity towards human somatostatin receptor type 3 using [125I]-[Leu8,DTrp22,Tyr25]SRIF-28 as radioligand.
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2MK6C9X
PubMed
Target
Somatostatin receptor type 1
(Homo sapiens (Human))
Salk Institute
Curated by
ChEMBL
Ligand
BDBM50136804
(CHEMBL439077 | Somatostatin analogue)
copy SMILES
copy InChI
Affinity Data
IC50: 517nM
Assay Description:
Binding affinity towards human somatostatin receptor type 1 using [125I]-[Leu8,DTrp22,Tyr25]SRIF-28 as radioligand.
More data for this Ligand-Target Pair
Target Info
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2MK6C9X
PubMed