Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetMelanocyte-stimulating hormone receptor(Mus musculus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50217789((E)-N-(3-aminopropyl)-2-(1H-indol-3-yl)-N-(2-methy...)copy SMILEScopy InChI
Affinity DataKi:  1.80E+3nMAssay Description:Displacement of [125I]NDP-MSH from MC1 receptor in mouse B16 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X066Q5PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50217789((E)-N-(3-aminopropyl)-2-(1H-indol-3-yl)-N-(2-methy...)copy SMILEScopy InChI
Affinity DataKi:  6.20E+3nMAssay Description:Displacement of [125I]NDP-MSH from human recombinant MC4 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X066Q5PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50217789((E)-N-(3-aminopropyl)-2-(1H-indol-3-yl)-N-(2-methy...)copy SMILEScopy InChI
Affinity DataKi:  9.10E+3nMAssay Description:Displacement of [125I]NDP-MSH from human recombinant MC3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X066Q5PubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50217789((E)-N-(3-aminopropyl)-2-(1H-indol-3-yl)-N-(2-methy...)copy SMILEScopy InChI
Affinity DataKi:  5.80E+4nMAssay Description:Displacement of [125I]NDP-MSH from human recombinant MC5 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X066Q5PubMed