Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 4 hits in this display
BDBM572249((5S)-2-(3-pyrimidin-4-yl-1H-pyrrolo[2,3-b]pyridin-...)copy SMILES
BDBM572249((5S)-2-(3-pyrimidin-4-yl-1H-pyrrolo[2,3-b]pyridin-...)copy SMILES
Ki: 0.0650nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
BDBM572249((5S)-2-(3-pyrimidin-4-yl-1H-pyrrolo[2,3-b]pyridin-...)copy SMILES
Ki: 4.41nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
BDBM572249((5S)-2-(3-pyrimidin-4-yl-1H-pyrrolo[2,3-b]pyridin-...)copy SMILES
Ki: 10.6nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair