Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetMelanocortin receptor 4(Mus musculus)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50409674(CHEMBL2096693)copy SMILEScopy InChI
Affinity DataEC50:  8.50E+3nMAssay Description:Activity in mouse melanocortin-4 receptor stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2Q2410RPubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University of Florida

Curated by ChEMBL
LigandPNGBDBM50409674(CHEMBL2096693)copy SMILEScopy InChI
Affinity DataEC50:  700nMAssay Description:Activity in mouse melanocortin-5 receptor stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2Q2410RPubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50409674(CHEMBL2096693)copy SMILEScopy InChI
Affinity DataEC50:  43nMAssay Description:Activity in mouse melanocortin-1 receptor stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2Q2410RPubMed
TargetMelanocortin receptor 3(Mus musculus)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50409674(CHEMBL2096693)copy SMILEScopy InChI
Affinity DataEC50:  2.32E+4nMAssay Description:Activity in mouse melanocortin-3 receptor (mMC3R) stably expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2Q2410RPubMed