Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hits in this display   

TargetSolute carrier family 12 member 5(Rattus norvegicus)
UCB Pharma SA

Curated by ChEMBL
LigandPNGBDBM50315369(CHEMBL1090183 | benzyl 1-acetyl-2-(4-fluoro-2-(tri...)copy SMILEScopy InChI
Affinity DataIC50: 4.00E+3nMAssay Description:Antagonist activity of rat KCC2 transporter expressed in human SK-Hep cells assessed as inhibition of N-ethylmaleimide-mediated Rb+ influx after 10 m...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BZ665CPubMed