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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Prostaglandin E2 receptor EP1 subtype
(Homo sapiens (Human))
GlaxoSmithKline
Curated by
ChEMBL
Ligand
BDBM50423023
(CHEMBL427844)
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copy InChI
Affinity Data
IC50: 0.400nM
Assay Description:
Displacement of [3H]PGE2 from human recombinant EP1 receptor expressed in CHO cell membranes
More data for this Ligand-Target Pair
Target Info
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2MC91B9
PubMed
Target
Thromboxane A2 receptor
(Homo sapiens (Human))
GlaxoSmithKline
Curated by
ChEMBL
Ligand
BDBM50423023
(CHEMBL427844)
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copy InChI
Affinity Data
IC50: 2.5nM
Assay Description:
Inhibition of TP receptor
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2MC91B9
PubMed
Target
Prostaglandin E2 receptor EP4 subtype
(Homo sapiens (Human))
GlaxoSmithKline
Curated by
ChEMBL
Ligand
BDBM50423023
(CHEMBL427844)
copy SMILES
copy InChI
Affinity Data
IC50: 158nM
Assay Description:
Inhibition of EP4 receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2MC91B9
PubMed