Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetThromboxane A2 receptor(Homo sapiens (Human))
Boehringer Ingelheim Pharma KG

Curated by ChEMBL

LigandBDBM50075646(5-{3-[1-(tert-butylamino)-2-cyano-(Z)-1-iminomethy...)copy SMILEScopy InChI

Affinity DataIC50: 81nMAssay Description:In vitro activity on thromboxane A2 receptor antagonism in gel filtered human platelets.More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41QMSPubMed

TargetThromboxane-A synthase(Homo sapiens (Human))
Boehringer Ingelheim Pharma KG

Curated by ChEMBL

LigandBDBM50075646(5-{3-[1-(tert-butylamino)-2-cyano-(Z)-1-iminomethy...)copy SMILEScopy InChI

Affinity DataIC50: 400nMAssay Description:In vitro activity on thromboxane A2 synthase inhibition in gel filtered human platelets.More data for this Ligand-Target Pair

Target InfoKEGG
UniProtKB/SwissProt
DrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H41QMSPubMed