Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50422958(CHEMBL2304246)copy SMILEScopy InChI
Affinity DataEC50:  5.27E+3nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2VZKPubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University of Florida

Curated by ChEMBL
LigandPNGBDBM50422958(CHEMBL2304246)copy SMILEScopy InChI
Affinity DataEC50:  1.98E+4nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2VZKPubMed
TargetMelanocortin receptor 3(Mus musculus)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50422958(CHEMBL2304246)copy SMILEScopy InChI
Affinity DataEC50:  2.26E+4nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2VZKPubMed
TargetMelanocortin receptor 4(Mus musculus)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50422958(CHEMBL2304246)copy SMILEScopy InChI
Affinity DataEC50:  8.33E+3nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells by beta-galactosidase assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2VZKPubMed