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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
30
hits in this display
Target
Proteasome subunit beta type-5
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526813
(CHEMBL4465456)
copy SMILES
copy InChI
Affinity Data
IC50: 38nM
Assay Description:
Inhibition of 20S proteosome beta 5 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2M61PQB
PubMed
Target
Proteasome subunit beta type-5
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526813
(CHEMBL4465456)
copy SMILES
copy InChI
Affinity Data
IC50: 38nM
Assay Description:
Inhibition of 20S proteosome beta 5 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2M61PQB
PubMed
Target
Proteasome subunit beta type-5
(Homo sapiens (Human))
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526813
(CHEMBL4465456)
copy SMILES
copy InChI
Affinity Data
IC50: 39nM
Assay Description:
Inhibition of 20S proteosome beta 5 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2M61PQB
PubMed
Target
Proteasome subunit beta type-5
(Homo sapiens (Human))
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526813
(CHEMBL4465456)
copy SMILES
copy InChI
Affinity Data
IC50: 39nM
Assay Description:
Inhibition of 20S proteosome beta 5 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2M61PQB
PubMed
Target
Proteasome subunit beta type-5
(Homo sapiens (Human))
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526813
(CHEMBL4465456)
copy SMILES
copy InChI
Affinity Data
IC50: 39nM
Assay Description:
Inhibition of 20S proteasome beta 5c (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2154MHB
PubMed
Target
Proteasome subunit beta type-8
(Homo sapiens (Human))
Hangzhou Xixi Hospital
Curated by
ChEMBL
Ligand
BDBM50526813
(CHEMBL4465456)
copy SMILES
copy InChI
Affinity Data
IC50: 49nM
Assay Description:
Inhibition of 20S proteasome beta 5i (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2154MHB
PubMed
Target
Proteasome subunit beta type-8
(Homo sapiens (Human))
Hangzhou Xixi Hospital
Curated by
ChEMBL
Ligand
BDBM50526813
(CHEMBL4465456)
copy SMILES
copy InChI
Affinity Data
IC50: 49nM
Assay Description:
Inhibition of LMP7 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2M61PQB
PubMed
Target
Proteasome subunit beta type-8
(Homo sapiens (Human))
Hangzhou Xixi Hospital
Curated by
ChEMBL
Ligand
BDBM50526813
(CHEMBL4465456)
copy SMILES
copy InChI
Affinity Data
IC50: 49nM
Assay Description:
Inhibition of LMP7 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2M61PQB
PubMed
Target
Proteasome subunit beta type-8
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526813
(CHEMBL4465456)
copy SMILES
copy InChI
Affinity Data
IC50: 56nM
Assay Description:
Inhibition of LMP7 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2M61PQB
PubMed
Target
Proteasome subunit beta type-8
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526813
(CHEMBL4465456)
copy SMILES
copy InChI
Affinity Data
IC50: 56nM
Assay Description:
Inhibition of LMP7 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2M61PQB
PubMed
Target
Proteasome subunit beta type-2
(Homo sapiens (Human))
Hangzhou Xixi Hospital
Curated by
ChEMBL
Ligand
BDBM50526813
(CHEMBL4465456)
copy SMILES
copy InChI
Affinity Data
IC50: 81nM
Assay Description:
Inhibition of 20S proteasome beta 2c (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2154MHB
PubMed
Target
Proteasome subunit beta type-2
(Homo sapiens (Human))
Hangzhou Xixi Hospital
Curated by
ChEMBL
Ligand
BDBM50526813
(CHEMBL4465456)
copy SMILES
copy InChI
Affinity Data
IC50: 81nM
Assay Description:
Inhibition of 20S proteosome beta 2 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2M61PQB
PubMed
Target
Proteasome subunit beta type-2
(Homo sapiens (Human))
Hangzhou Xixi Hospital
Curated by
ChEMBL
Ligand
BDBM50526813
(CHEMBL4465456)
copy SMILES
copy InChI
Affinity Data
IC50: 81nM
Assay Description:
Inhibition of 20S proteosome beta 2 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2M61PQB
PubMed
Target
Proteasome subunit beta type-10
(Homo sapiens (Human))
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526813
(CHEMBL4465456)
copy SMILES
copy InChI
Affinity Data
IC50: 97nM
Assay Description:
Inhibition of MECL1 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2M61PQB
PubMed
Target
Proteasome subunit beta type-10
(Homo sapiens (Human))
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526813
(CHEMBL4465456)
copy SMILES
copy InChI
Affinity Data
IC50: 97nM
Assay Description:
Inhibition of MECL1 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2M61PQB
PubMed
Target
Proteasome subunit beta type-10
(Homo sapiens (Human))
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526813
(CHEMBL4465456)
copy SMILES
copy InChI
Affinity Data
IC50: 97nM
Assay Description:
Inhibition of 20S proteasome beta 2i (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2154MHB
PubMed
Target
Proteasome subunit beta type-2
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526813
(CHEMBL4465456)
copy SMILES
copy InChI
Affinity Data
IC50: 141nM
Assay Description:
Inhibition of 20S proteosome beta 2 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2M61PQB
PubMed
Target
Proteasome subunit beta type-2
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526813
(CHEMBL4465456)
copy SMILES
copy InChI
Affinity Data
IC50: 141nM
Assay Description:
Inhibition of 20S proteosome beta 2 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2M61PQB
PubMed
Target
Proteasome subunit beta type-10
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526813
(CHEMBL4465456)
copy SMILES
copy InChI
Affinity Data
IC50: 159nM
Assay Description:
Inhibition of MECL1 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2M61PQB
PubMed
Target
Proteasome subunit beta type-10
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526813
(CHEMBL4465456)
copy SMILES
copy InChI
Affinity Data
IC50: 159nM
Assay Description:
Inhibition of MECL1 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2M61PQB
PubMed
Target
Proteasome subunit beta type-9
(Homo sapiens (Human))
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526813
(CHEMBL4465456)
copy SMILES
copy InChI
Affinity Data
IC50: 415nM
Assay Description:
Inhibition of LMP2 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2M61PQB
PubMed
Target
Proteasome subunit beta type-9
(Homo sapiens (Human))
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526813
(CHEMBL4465456)
copy SMILES
copy InChI
Affinity Data
IC50: 415nM
Assay Description:
Inhibition of LMP2 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2M61PQB
PubMed
Target
Proteasome subunit beta type-9
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526813
(CHEMBL4465456)
copy SMILES
copy InChI
Affinity Data
IC50: 415nM
Assay Description:
Inhibition of LMP2 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2M61PQB
PubMed
Target
Proteasome subunit beta type-9
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526813
(CHEMBL4465456)
copy SMILES
copy InChI
Affinity Data
IC50: 415nM
Assay Description:
Inhibition of LMP2 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2M61PQB
PubMed
Target
Proteasome subunit beta type-9
(Homo sapiens (Human))
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526813
(CHEMBL4465456)
copy SMILES
copy InChI
Affinity Data
IC50: 425nM
Assay Description:
Inhibition of 20S proteasome beta 1i (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2154MHB
PubMed
Target
Proteasome subunit beta type-1
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526813
(CHEMBL4465456)
copy SMILES
copy InChI
Affinity Data
IC50: 2.50E+5nM
Assay Description:
Inhibition of 20S proteosome beta 1 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2M61PQB
PubMed
Target
Proteasome subunit beta type-1
(Homo sapiens (Human))
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526813
(CHEMBL4465456)
copy SMILES
copy InChI
Affinity Data
IC50: 2.50E+5nM
Assay Description:
Inhibition of 20S proteosome beta 1 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2M61PQB
PubMed
Target
Proteasome subunit beta type-1
(Homo sapiens (Human))
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526813
(CHEMBL4465456)
copy SMILES
copy InChI
Affinity Data
IC50: 2.50E+5nM
Assay Description:
Inhibition of 20S proteasome beta 1c (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2154MHB
PubMed
Target
Proteasome subunit beta type-1
(Homo sapiens (Human))
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526813
(CHEMBL4465456)
copy SMILES
copy InChI
Affinity Data
IC50: 2.50E+5nM
Assay Description:
Inhibition of 20S proteosome beta 1 in human MOLT4 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2M61PQB
PubMed
Target
Proteasome subunit beta type-1
(Mus musculus)
Kezar Life Sciences
Curated by
ChEMBL
Ligand
BDBM50526813
(CHEMBL4465456)
copy SMILES
copy InChI
Affinity Data
IC50: 2.50E+5nM
Assay Description:
Inhibition of 20S proteosome beta 1 in mouse A20 cells by ELISA
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2M61PQB
PubMed