Home
About
Info
Download
WebServices
Contact
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
14
hits in this display
Target
Group 10 secretory phospholipase A2
(Homo sapiens (Human))
University of Washington
Curated by
ChEMBL
Ligand
BDBM50262844
(2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2-isobutyl-1H-...)
copy SMILES
copy InChI
Affinity Data
IC50: 50nM
Assay Description:
Inhibition of human group2X phospholipase A2 fluorimetric assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2571BSD
PubMed
Target
Group IID secretory phospholipase A2
(Homo sapiens (Human))
University of Washington
Curated by
ChEMBL
Ligand
BDBM50262844
(2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2-isobutyl-1H-...)
copy SMILES
copy InChI
Affinity Data
IC50: 500nM
Assay Description:
Inhibition of human group2D phospholipase A2 by [3H]oleic acid-labeled Escherichia coli membrane assay
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2571BSD
PubMed
Target
Group IIF secretory phospholipase A2
(Homo sapiens (Human))
University of Washington
Curated by
ChEMBL
Ligand
BDBM50262844
(2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2-isobutyl-1H-...)
copy SMILES
copy InChI
Affinity Data
IC50: 550nM
Assay Description:
Inhibition of human group2F phospholipase A2 fluorimetric assay
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2571BSD
PubMed
Target
Phospholipase A2
(Mus musculus)
University of Washington
Curated by
ChEMBL
Ligand
BDBM50262844
(2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2-isobutyl-1H-...)
copy SMILES
copy InChI
Affinity Data
IC50: 580nM
Assay Description:
Inhibition of mouse group1B phospholipase A2 fluorimetric assay
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2571BSD
PubMed
Target
Group IIE secretory phospholipase A2
(Homo sapiens (Human))
University of Washington
Curated by
ChEMBL
Ligand
BDBM50262844
(2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2-isobutyl-1H-...)
copy SMILES
copy InChI
Affinity Data
IC50: 1.30E+3nM
Assay Description:
Inhibition of human group2E phospholipase A2 fluorimetric assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2571BSD
PubMed
Target
Group IID secretory phospholipase A2
(Mus musculus)
University of Washington
Curated by
ChEMBL
Ligand
BDBM50262844
(2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2-isobutyl-1H-...)
copy SMILES
copy InChI
Affinity Data
IC50: 1.60E+3nM
Assay Description:
Inhibition of mouse group2D phospholipase A2 fluorimetric assay
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2571BSD
PubMed
Target
Group 10 secretory phospholipase A2
(Mus musculus)
University of Washington
Curated by
ChEMBL
Ligand
BDBM50262844
(2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2-isobutyl-1H-...)
copy SMILES
copy InChI
Affinity Data
IC50: 1.60E+3nM
Assay Description:
Inhibition of mouse group2X phospholipase A2 fluorimetric assay
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2571BSD
PubMed
Target
Group IIE secretory phospholipase A2
(Mus musculus)
University of Washington
Curated by
ChEMBL
Ligand
BDBM50262844
(2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2-isobutyl-1H-...)
copy SMILES
copy InChI
Affinity Data
IC50: 1.60E+3nM
Assay Description:
Inhibition of mouse group2E phospholipase A2 fluorimetric assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2571BSD
PubMed
Target
Phospholipase A2, membrane associated
(Homo sapiens (Human))
University of Washington
Curated by
ChEMBL
Ligand
BDBM50262844
(2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2-isobutyl-1H-...)
copy SMILES
copy InChI
Affinity Data
IC50: 1.60E+3nM
Assay Description:
Inhibition of human group2A phospholipase A2 fluorimetric assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2571BSD
PubMed
Target
Phospholipase A2, membrane associated
(Mus musculus)
University of Washington
Curated by
ChEMBL
Ligand
BDBM50262844
(2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2-isobutyl-1H-...)
copy SMILES
copy InChI
Affinity Data
IC50: 1.60E+3nM
Assay Description:
Inhibition of mouse group2A phospholipase A2 fluorimetric assay
More data for this Ligand-Target Pair
Target Info
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2571BSD
PubMed
Target
Phospholipase A2 group V
(Homo sapiens (Human))
University of Washington
Curated by
ChEMBL
Ligand
BDBM50262844
(2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2-isobutyl-1H-...)
copy SMILES
copy InChI
Affinity Data
IC50: 1.60E+3nM
Assay Description:
Inhibition of human group2V phospholipase A2 fluorimetric assay
More data for this Ligand-Target Pair
Target Info
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2571BSD
PubMed
Target
Phospholipase A2 group V
(Mus musculus)
University of Washington
Curated by
ChEMBL
Ligand
BDBM50262844
(2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2-isobutyl-1H-...)
copy SMILES
copy InChI
Affinity Data
IC50: 1.60E+3nM
Assay Description:
Inhibition of mouse group2V phospholipase A2 fluorimetric assay
More data for this Ligand-Target Pair
Target Info
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2571BSD
PubMed
Target
Phospholipase A2
(Homo sapiens (Human))
University of Washington
Curated by
ChEMBL
Ligand
BDBM50262844
(2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2-isobutyl-1H-...)
copy SMILES
copy InChI
Affinity Data
IC50: 1.60E+3nM
Assay Description:
Inhibition of human group1B phospholipase A2 fluorimetric assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2571BSD
PubMed
Target
Group IIF secretory phospholipase A2
(Mus musculus)
University of Washington
Curated by
ChEMBL
Ligand
BDBM50262844
(2-(3-(2-amino-2-oxoacetyl)-1-benzyl-2-isobutyl-1H-...)
copy SMILES
copy InChI
Affinity Data
IC50: 1.60E+3nM
Assay Description:
Inhibition of mouse group2F phospholipase A2 fluorimetric assay
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2571BSD
PubMed