Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetInterleukin-1 receptor-associated kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50560886(CHEMBL4744403)copy SMILES
Affinity DataIC50: 6nMAssay Description:Inhibition of kinase tracer 236 binding to recombinant human full-length GST-tagged IRAK3 expressed in insect cells by Lanthascreen Eu kinase binding...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P84GMZPubMed
TargetCyclin-C/Cyclin-dependent kinase 19(Homo sapiens (Human))TBA
LigandPNGBDBM50560886(CHEMBL4744403)copy SMILES
Affinity DataIC50: 70nMAssay Description:Inhibition of CDK11/cyclin C (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P84GMZPubMed
TargetSerine/threonine-protein kinase haspin(Homo sapiens (Human))TBA
LigandPNGBDBM50560886(CHEMBL4744403)copy SMILES
Affinity DataIC50: 150nMAssay Description:Inhibition of GSG2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P84GMZPubMed
TargetInterleukin-1 receptor-associated kinase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50560886(CHEMBL4744403)copy SMILES
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of recombinant human full-length His-tagged IRAK4 expressed in baculovirus expression system using 5-FAM-IPTSPITTTYFFFKKK-COOH as substrat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P84GMZPubMed
TargetInterleukin-1 receptor-associated kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM50560886(CHEMBL4744403)copy SMILES
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged IRAK1 (194 to 712 residues) expressed in baculovirus expression system using 5-FAM-KKKVSRSGLYRS...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P84GMZPubMed