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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
5
hits in this display
Target
Interleukin-1 receptor-associated kinase 3
(Homo sapiens (Human))
TBA
Ligand
BDBM50560886
(CHEMBL4744403)
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Affinity Data
IC50: 6nM
Assay Description:
Inhibition of kinase tracer 236 binding to recombinant human full-length GST-tagged IRAK3 expressed in insect cells by Lanthascreen Eu kinase binding...
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2P84GMZ
PubMed
Target
Cyclin-C/Cyclin-dependent kinase 19
(Homo sapiens (Human))
TBA
Ligand
BDBM50560886
(CHEMBL4744403)
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Affinity Data
IC50: 70nM
Assay Description:
Inhibition of CDK11/cyclin C (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2P84GMZ
PubMed
Target
Serine/threonine-protein kinase haspin
(Homo sapiens (Human))
TBA
Ligand
BDBM50560886
(CHEMBL4744403)
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Affinity Data
IC50: 150nM
Assay Description:
Inhibition of GSG2 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2P84GMZ
PubMed
Target
Interleukin-1 receptor-associated kinase 4
(Homo sapiens (Human))
TBA
Ligand
BDBM50560886
(CHEMBL4744403)
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Affinity Data
IC50: 1.00E+3nM
Assay Description:
Inhibition of recombinant human full-length His-tagged IRAK4 expressed in baculovirus expression system using 5-FAM-IPTSPITTTYFFFKKK-COOH as substrat...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2P84GMZ
PubMed
Target
Interleukin-1 receptor-associated kinase 1
(Homo sapiens (Human))
TBA
Ligand
BDBM50560886
(CHEMBL4744403)
copy SMILES
Affinity Data
IC50: 1.30E+3nM
Assay Description:
Inhibition of recombinant human N-terminal GST-tagged IRAK1 (194 to 712 residues) expressed in baculovirus expression system using 5-FAM-KKKVSRSGLYRS...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2P84GMZ
PubMed