Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetSomatostatin receptor type 2(Homo sapiens (Human))
Technische Universit£t M£nchen

Curated by ChEMBL
LigandPNGBDBM50165172(4-[(4R,7S,10S,13R,16S)-19-(2-azaniumyl-3-phenylpro...)copy SMILEScopy InChI
Affinity DataIC50: 1.60nMAssay Description:In vitro inhibition of [125I][Leu8,D-Trp22,Tyr25] somatostatin 28 binding to human somatostatin receptor type 2 expressed in CCL39 cells; (n=5)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0ND0PubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Technische Universit£t M£nchen

Curated by ChEMBL
LigandPNGBDBM50165172(4-[(4R,7S,10S,13R,16S)-19-(2-azaniumyl-3-phenylpro...)copy SMILEScopy InChI
Affinity DataIC50: 65nMAssay Description:In vitro inhibition of [125I][Leu8,D-Trp22,Tyr25] somatostatin 28 binding to human somatostatin receptor type 5 expressed in CHO-K1 cells; (n=5)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0ND0PubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Technische Universit£t M£nchen

Curated by ChEMBL
LigandPNGBDBM50165172(4-[(4R,7S,10S,13R,16S)-19-(2-azaniumyl-3-phenylpro...)copy SMILEScopy InChI
Affinity DataIC50: 186nMAssay Description:In vitro inhibition of [125I][Leu8,D-Trp22,Tyr25] somatostatin 28 binding to human somatostatin receptor type 3 expressed in CCL39 cells; (n=5)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0ND0PubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Technische Universit£t M£nchen

Curated by ChEMBL
LigandPNGBDBM50165172(4-[(4R,7S,10S,13R,16S)-19-(2-azaniumyl-3-phenylpro...)copy SMILEScopy InChI
Affinity DataIC50: 729nMAssay Description:In vitro inhibition of [125I][Leu8,D-Trp22,Tyr25] somatostatin 28 binding to human somatostatin receptor type 4 expressed in CCL39 cells; (n=5)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0ND0PubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Technische Universit£t M£nchen

Curated by ChEMBL
LigandPNGBDBM50165172(4-[(4R,7S,10S,13R,16S)-19-(2-azaniumyl-3-phenylpro...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro inhibition of [125I][Leu8,D-Trp22,Tyr25] somatostatin 28 binding to human somatostatin receptor type 1 expressed in CHO-K1 cells; (n=5)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0ND0PubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Technische Universit£t M£nchen

Curated by ChEMBL
LigandPNGBDBM50165172(4-[(4R,7S,10S,13R,16S)-19-(2-azaniumyl-3-phenylpro...)copy SMILEScopy InChI
Affinity DataEC50:  1nMAssay Description:Relative effective concentration against human somatostatin receptor type 2 expressed in CHO cells; (n=3)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26T0ND0PubMed