Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetProteasome subunit beta type-5(Homo sapiens (Human))
Universit£ Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464962(CHEMBL4290574)copy SMILEScopy InChI
Affinity DataIC50: 7.10nMAssay Description:Inhibition of human 20S constitutive proteasome beta-5 using Suc-LLVY-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959M74PubMed
TargetProteasome subunit beta type-8(Homo sapiens (Human))
Universit£ Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464962(CHEMBL4290574)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of human 20S immunoproteasome beta-5 using Suc-LLVY-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959M74PubMed
TargetProteasome subunit beta type-10(Homo sapiens (Human))
Universit£ Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464962(CHEMBL4290574)copy SMILEScopy InChI
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibition of human 20S immunoproteasome beta-2 using BocLRR-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959M74PubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Universit£ Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464962(CHEMBL4290574)copy SMILEScopy InChI
Affinity DataIC50: 1.32E+4nMAssay Description:Inhibition of human 20S constitutive proteasome beta-2 using BocLRR-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959M74PubMed
TargetProteasome subunit beta type-9(Homo sapiens (Human))
Universit£ Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464962(CHEMBL4290574)copy SMILEScopy InChI
Affinity DataIC50: 2.38E+4nMAssay Description:Inhibition of human 20S immunoproteasome beta-1 using Ac-PAL-AMC as substrate incubated for 15 mins measured for 45 mins by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959M74PubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Universit£ Rennes 1

Curated by ChEMBL
LigandPNGBDBM50464962(CHEMBL4290574)copy SMILEScopy InChI
Affinity DataIC50: 3.19E+4nMAssay Description:Inhibition of human 20S constitutive proteasome beta-1 using Z-LLE-betaNA as substrate incubated for 15 mins measured for 45 mins by fluorescence ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959M74PubMed