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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
23
hits in this display
Target
Somatostatin receptor type 5
(Homo sapiens (Human))
Royal Victoria Hospital
Curated by
PDSP K
i
Database
Ligand
BDBM50063839
(BIM 23268 | CHEMBL263606 | H-cyclo[DCys-Phe-Phe-DT...)
copy SMILES
copy InChI
Affinity Data
Ki: 0.370nM
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2CR5RXQ
PubMed
Target
Somatostatin receptor type 5
(Homo sapiens (Human))
Royal Victoria Hospital
Curated by
PDSP K
i
Database
Ligand
BDBM50063839
(BIM 23268 | CHEMBL263606 | H-cyclo[DCys-Phe-Phe-DT...)
copy SMILES
copy InChI
Affinity Data
Ki: 0.370nM
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2H70DCK
PubMed
Target
Somatostatin receptor type 2
(MOUSE)
German Institute of Human Nutrition
Curated by
PDSP K
i
Database
Ligand
BDBM50063839
(BIM 23268 | CHEMBL263606 | H-cyclo[DCys-Phe-Phe-DT...)
copy SMILES
copy InChI
Affinity Data
Ki: 1.49nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q22R3Q6B
PubMed
Target
Somatostatin receptor type 5
(Homo sapiens (Human))
Royal Victoria Hospital
Curated by
PDSP K
i
Database
Ligand
BDBM50063839
(BIM 23268 | CHEMBL263606 | H-cyclo[DCys-Phe-Phe-DT...)
copy SMILES
copy InChI
Affinity Data
Ki: 2.18nM
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q22R3Q6B
PubMed
Target
Somatostatin receptor type 5
(RAT)
German Institute of Human Nutrition
Curated by
PDSP K
i
Database
Ligand
BDBM50063839
(BIM 23268 | CHEMBL263606 | H-cyclo[DCys-Phe-Phe-DT...)
copy SMILES
copy InChI
Affinity Data
Ki: 3.40nM
More data for this Ligand-Target Pair
Target Info
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q22R3Q6B
PubMed
Target
Somatostatin receptor type 3
(RAT)
German Institute of Human Nutrition
Curated by
PDSP K
i
Database
Ligand
BDBM50063839
(BIM 23268 | CHEMBL263606 | H-cyclo[DCys-Phe-Phe-DT...)
copy SMILES
copy InChI
Affinity Data
Ki: 4.10nM
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q22R3Q6B
PubMed
Target
Somatostatin receptor type 2
(MOUSE)
German Institute of Human Nutrition
Curated by
PDSP K
i
Database
Ligand
BDBM50063839
(BIM 23268 | CHEMBL263606 | H-cyclo[DCys-Phe-Phe-DT...)
copy SMILES
copy InChI
Affinity Data
Ki: 11nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q22R3Q6B
PubMed
Target
Somatostatin receptor type 2
(Homo sapiens (Human))
Royal Victoria Hospital
Curated by
PDSP K
i
Database
Ligand
BDBM50063839
(BIM 23268 | CHEMBL263606 | H-cyclo[DCys-Phe-Phe-DT...)
copy SMILES
copy InChI
Affinity Data
Ki: 15.1nM
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2CR5RXQ
PubMed
Target
Somatostatin receptor type 2
(Homo sapiens (Human))
Royal Victoria Hospital
Curated by
PDSP K
i
Database
Ligand
BDBM50063839
(BIM 23268 | CHEMBL263606 | H-cyclo[DCys-Phe-Phe-DT...)
copy SMILES
copy InChI
Affinity Data
Ki: 15.1nM
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2H70DCK
PubMed
Target
Somatostatin receptor type 4
(Homo sapiens (Human))
Cedars-Sinai Research Institute
Curated by
PDSP K
i
Database
Ligand
BDBM50063839
(BIM 23268 | CHEMBL263606 | H-cyclo[DCys-Phe-Phe-DT...)
copy SMILES
copy InChI
Affinity Data
Ki: 16.3nM
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2H70DCK
PubMed
Target
Somatostatin receptor type 4
(Homo sapiens (Human))
Cedars-Sinai Research Institute
Curated by
PDSP K
i
Database
Ligand
BDBM50063839
(BIM 23268 | CHEMBL263606 | H-cyclo[DCys-Phe-Phe-DT...)
copy SMILES
copy InChI
Affinity Data
Ki: 16.3nM
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2CR5RXQ
PubMed
Target
Somatostatin receptor type 1
(Homo sapiens (Human))
Cedars-Sinai Research Institute
Curated by
PDSP K
i
Database
Ligand
BDBM50063839
(BIM 23268 | CHEMBL263606 | H-cyclo[DCys-Phe-Phe-DT...)
copy SMILES
copy InChI
Affinity Data
Ki: 18.4nM
More data for this Ligand-Target Pair
Target Info
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2H70DCK
PubMed
Target
Somatostatin receptor type 1
(Homo sapiens (Human))
Cedars-Sinai Research Institute
Curated by
PDSP K
i
Database
Ligand
BDBM50063839
(BIM 23268 | CHEMBL263606 | H-cyclo[DCys-Phe-Phe-DT...)
copy SMILES
copy InChI
Affinity Data
Ki: 18.4nM
More data for this Ligand-Target Pair
Target Info
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2CR5RXQ
PubMed
Target
Somatostatin receptor type 3
(Homo sapiens (Human))
Royal Victoria Hospital
Curated by
PDSP K
i
Database
Ligand
BDBM50063839
(BIM 23268 | CHEMBL263606 | H-cyclo[DCys-Phe-Phe-DT...)
copy SMILES
copy InChI
Affinity Data
Ki: 61.6nM
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2CR5RXQ
PubMed
Target
Somatostatin receptor type 3
(Homo sapiens (Human))
Royal Victoria Hospital
Curated by
PDSP K
i
Database
Ligand
BDBM50063839
(BIM 23268 | CHEMBL263606 | H-cyclo[DCys-Phe-Phe-DT...)
copy SMILES
copy InChI
Affinity Data
Ki: 61.6nM
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2H70DCK
PubMed
Target
Somatostatin receptor type 2
(RAT)
German Institute of Human Nutrition
Curated by
PDSP K
i
Database
Ligand
BDBM50063839
(BIM 23268 | CHEMBL263606 | H-cyclo[DCys-Phe-Phe-DT...)
copy SMILES
copy InChI
Affinity Data
Ki: 101nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q22R3Q6B
PubMed
Target
Somatostatin receptor type 4
(Homo sapiens (Human))
Cedars-Sinai Research Institute
Curated by
PDSP K
i
Database
Ligand
BDBM50063839
(BIM 23268 | CHEMBL263606 | H-cyclo[DCys-Phe-Phe-DT...)
copy SMILES
copy InChI
Affinity Data
Ki: 174nM
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q22R3Q6B
PubMed
Target
Somatostatin receptor type 1
(Homo sapiens (Human))
Cedars-Sinai Research Institute
Curated by
PDSP K
i
Database
Ligand
BDBM50063839
(BIM 23268 | CHEMBL263606 | H-cyclo[DCys-Phe-Phe-DT...)
copy SMILES
copy InChI
Affinity Data
Ki: 582nM
More data for this Ligand-Target Pair
Target Info
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q22R3Q6B
PubMed
Target
Somatostatin receptor type 3
(Homo sapiens (Human))
Royal Victoria Hospital
Curated by
PDSP K
i
Database
Ligand
BDBM50455449
(CHEMBL2370306)
copy SMILES
copy InChI
Affinity Data
IC50: 5.60nM
Assay Description:
Binding affinity towards cloned human somatostatin 3 (hsst) receptor
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q26W9BS9
PubMed
Target
Somatostatin receptor type 5
(Homo sapiens (Human))
Royal Victoria Hospital
Curated by
PDSP K
i
Database
Ligand
BDBM50455449
(CHEMBL2370306)
copy SMILES
copy InChI
Affinity Data
IC50: 28nM
Assay Description:
Binding affinity towards cloned human somatostatin 5 (hsst) receptor
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q26W9BS9
PubMed
Target
Somatostatin receptor type 2
(Homo sapiens (Human))
Royal Victoria Hospital
Curated by
PDSP K
i
Database
Ligand
BDBM50455449
(CHEMBL2370306)
copy SMILES
copy InChI
Affinity Data
IC50: 35nM
Assay Description:
Binding affinity towards cloned human somatostatin 2 (hsst) receptor
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q26W9BS9
PubMed
Target
Somatostatin receptor type 4
(Homo sapiens (Human))
Cedars-Sinai Research Institute
Curated by
PDSP K
i
Database
Ligand
BDBM50455449
(CHEMBL2370306)
copy SMILES
copy InChI
Affinity Data
IC50: 406nM
Assay Description:
Binding affinity towards cloned human somatostatin 4 (hsst) receptor
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q26W9BS9
PubMed
Target
Somatostatin receptor type 1
(Homo sapiens (Human))
Cedars-Sinai Research Institute
Curated by
PDSP K
i
Database
Ligand
BDBM50455449
(CHEMBL2370306)
copy SMILES
copy InChI
Affinity Data
IC50: 723nM
Assay Description:
Binding affinity towards cloned human somatostatin 1 (hsst) receptor
More data for this Ligand-Target Pair
Target Info
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q26W9BS9
PubMed