Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetMAP/microtubule affinity-regulating kinase 3(Homo sapiens (Human))
Merck& Co.

Curated by ChEMBL
LigandPNGBDBM50208912(CHEMBL3883766)copy SMILEScopy InChI
Affinity DataIC50: 738nMAssay Description:Inhibition of full length human MARK3 using biotin labeled peptide substrate by HTRF based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N018JCPubMed
TargetMAP/microtubule affinity-regulating kinase 3(Homo sapiens (Human))
Merck& Co.

Curated by ChEMBL
LigandPNGBDBM50208912(CHEMBL3883766)copy SMILEScopy InChI
Affinity DataIC50: 738nMAssay Description:Inhibition of MARK3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20867B1PubMed
TargetMAP/microtubule affinity-regulating kinase 4(Homo sapiens (Human))
Merck& Co.

Curated by ChEMBL
LigandPNGBDBM50208912(CHEMBL3883766)copy SMILEScopy InChI
Affinity DataIC50: 5.91E+3nMAssay Description:Inhibition of human MARK4 expressed in HEK293T cells coexpressing tau protein assessed as reduction in tau phosphorylation at Ser262 residues by Alph...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N018JCPubMed