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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
8
hits in this display
Target
Melanocyte-stimulating hormone receptor
(Homo sapiens (Human))
The University of Queensland
Curated by
ChEMBL
Ligand
BDBM50263821
(CHEMBL4080223)
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Affinity Data
Ki: 4.68E+3nM
Assay Description:
Displacement of [125I]-NDP-alpha-MSH from human MC1R LBD expressed in HEK293 cell membranes incubated for 16 to 23 hrs in dark by scintillation proxi...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2736TCZ
PubMed
Target
Melanocortin receptor 4
(Homo sapiens (Human))
The University of Queensland
Curated by
ChEMBL
Ligand
BDBM50263821
(CHEMBL4080223)
copy SMILES
copy InChI
Affinity Data
Ki: 6.31E+3nM
Assay Description:
Displacement of [125I]-NDP-alpha-MSH from human MC4R LBD expressed in HEK293 cell membranes incubated for 16 to 23 hrs in dark by scintillation proxi...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2736TCZ
PubMed
Target
Melanocortin receptor 3
(Homo sapiens (Human))
The University of Queensland
Curated by
ChEMBL
Ligand
BDBM50263821
(CHEMBL4080223)
copy SMILES
copy InChI
Affinity Data
Ki: 3.89E+4nM
Assay Description:
Displacement of [125I]-NDP-alpha-MSH from human MC3R LBD expressed in HEK293 cell membranes incubated for 16 to 23 hrs in dark by scintillation proxi...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2736TCZ
PubMed
Target
Melanocortin receptor 5
(Homo sapiens (Human))
The University of Queensland
Curated by
ChEMBL
Ligand
BDBM50263821
(CHEMBL4080223)
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copy InChI
Affinity Data
IC50: 1.12E+4nM
Assay Description:
Displacement of [125I]-NDP-alpha-MSH from human MC5R LBD expressed in HEK293 cell membranes incubated for 16 to 23 hrs in dark by scintillation proxi...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2736TCZ
PubMed
Target
Melanocortin receptor 4
(Homo sapiens (Human))
The University of Queensland
Curated by
ChEMBL
Ligand
BDBM50263821
(CHEMBL4080223)
copy SMILES
copy InChI
Affinity Data
EC50: 1.05E+3nM
Assay Description:
Agonist activity at human MC4R expressed in high doxycyclin-treated HEK293 cell membranes assessed as increase in cAMP production after 15 mins by HT...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2736TCZ
PubMed
Target
Melanocortin receptor 4
(Homo sapiens (Human))
The University of Queensland
Curated by
ChEMBL
Ligand
BDBM50263821
(CHEMBL4080223)
copy SMILES
copy InChI
Affinity Data
EC50: 1.07E+4nM
Assay Description:
Agonist activity at human MC4R expressed in low doxycyclin-treated HEK293 cell membranes assessed as increase in cAMP production after 45 mins by HTR...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2736TCZ
PubMed
Target
Melanocortin receptor 3
(Homo sapiens (Human))
The University of Queensland
Curated by
ChEMBL
Ligand
BDBM50263821
(CHEMBL4080223)
copy SMILES
copy InChI
Affinity Data
EC50: 7.41E+3nM
Assay Description:
Agonist activity at human MC3R expressed in low doxycyclin-treated HEK293 cell membranes assessed as increase in cAMP production after 45 mins by HTR...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2736TCZ
PubMed
Target
Melanocyte-stimulating hormone receptor
(Homo sapiens (Human))
The University of Queensland
Curated by
ChEMBL
Ligand
BDBM50263821
(CHEMBL4080223)
copy SMILES
copy InChI
Affinity Data
EC50: 1.32E+3nM
Assay Description:
Agonist activity at human MC1R expressed in low doxycyclin-treated HEK293 cell membranes assessed as increase in cAMP production after 45 mins by HTR...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2736TCZ
PubMed