Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetRelaxin-3 receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50558044(CHEMBL4796474)copy SMILES
Affinity DataKi:  23nMAssay Description:Displacement of europium-labeled Eu(A)-mINSL5 from human RXFP4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC3624PubMed
TargetRelaxin-3 receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50558044(CHEMBL4796474)copy SMILES
Affinity DataKi:  23nMAssay Description:Displacement of europium-labeled Eu(A)-mINSL5 from human RXFP4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC3624PubMed
TargetRelaxin-3 receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50558044(CHEMBL4796474)copy SMILES
Affinity DataEC50:  40nMAssay Description:Agonist activity at human RXFP4 expressed in CHO-K1 cells assessed as reduction in forskolin-induced cAMP production by pCRE beta-galactosidase repor...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC3624PubMed
TargetRelaxin-3 receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50558044(CHEMBL4796474)copy SMILES
Affinity DataEC50:  40nMAssay Description:Agonist activity at human RXFP4 expressed in CHO-K1 cells assessed as reduction in forskolin-induced cAMP production by pCRE beta-galactosidase repor...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PC3624PubMed