Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetOxytocin receptor(RAT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50407012(CHEMBL2112666)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Displacement of [3H]-OT from binding to oxytocin receptor of rat uterusMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21C1VZ0PubMed
TargetOxytocin receptor(RAT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50407012(CHEMBL2112666)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of radioligand [3H]-oxytocin binding at the oxytocin (OT) receptor in rat uterine tissueMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27M070WPubMed
TargetVasopressin V1a receptor(RAT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50407012(CHEMBL2112666)copy SMILEScopy InChI
Affinity DataIC50: 890nMAssay Description:Displacement of [3H]AVP from binding to arginine vasopressin 1a (V1a) column of rat liverMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21C1VZ0PubMed
TargetVasopressin V1a/V1b receptor(RAT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50407012(CHEMBL2112666)copy SMILEScopy InChI
Affinity DataIC50: 890nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27M070WPubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50407012(CHEMBL2112666)copy SMILEScopy InChI
Affinity DataIC50: 2.40E+3nMAssay Description:Displacement of [3H]-AVP from binding to Vasopressin receptor V2 of rat kidneyMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21C1VZ0PubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50407012(CHEMBL2112666)copy SMILEScopy InChI
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of radioligand [3H]-AVP binding to the vasopressin V2 receptor in rat kidney tissueMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27M070WPubMed