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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
6
hits in this display
Target
Oxytocin receptor
(RAT)
Merck Research Laboratories
Curated by
ChEMBL
Ligand
BDBM50407012
(CHEMBL2112666)
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Affinity Data
IC50: 12nM
Assay Description:
Displacement of [3H]-OT from binding to oxytocin receptor of rat uterus
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
BindingDB Entry DOI:
10.7270/Q21C1VZ0
PubMed
Target
Oxytocin receptor
(RAT)
Merck Research Laboratories
Curated by
ChEMBL
Ligand
BDBM50407012
(CHEMBL2112666)
copy SMILES
copy InChI
Affinity Data
IC50: 12nM
Assay Description:
Inhibition of radioligand [3H]-oxytocin binding at the oxytocin (OT) receptor in rat uterine tissue
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
BindingDB Entry DOI:
10.7270/Q27M070W
PubMed
Target
Vasopressin V1a receptor
(RAT)
Merck Research Laboratories
Curated by
ChEMBL
Ligand
BDBM50407012
(CHEMBL2112666)
copy SMILES
copy InChI
Affinity Data
IC50: 890nM
Assay Description:
Displacement of [3H]AVP from binding to arginine vasopressin 1a (V1a) column of rat liver
More data for this Ligand-Target Pair
Target Info
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
BindingDB Entry DOI:
10.7270/Q21C1VZ0
PubMed
Target
Vasopressin V1a/V1b receptor
(RAT)
Merck Research Laboratories
Curated by
ChEMBL
Ligand
BDBM50407012
(CHEMBL2112666)
copy SMILES
copy InChI
Affinity Data
IC50: 890nM
Assay Description:
Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissue
More data for this Ligand-Target Pair
Target Info
MMDB
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
BindingDB Entry DOI:
10.7270/Q27M070W
PubMed
Target
Vasopressin V2 receptor
(Rattus norvegicus (Rat))
Merck Research Laboratories
Curated by
ChEMBL
Ligand
BDBM50407012
(CHEMBL2112666)
copy SMILES
copy InChI
Affinity Data
IC50: 2.40E+3nM
Assay Description:
Displacement of [3H]-AVP from binding to Vasopressin receptor V2 of rat kidney
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
BindingDB Entry DOI:
10.7270/Q21C1VZ0
PubMed
Target
Vasopressin V2 receptor
(Rattus norvegicus (Rat))
Merck Research Laboratories
Curated by
ChEMBL
Ligand
BDBM50407012
(CHEMBL2112666)
copy SMILES
copy InChI
Affinity Data
IC50: 2.40E+3nM
Assay Description:
Inhibition of radioligand [3H]-AVP binding to the vasopressin V2 receptor in rat kidney tissue
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
BindingDB Entry DOI:
10.7270/Q27M070W
PubMed